JP5383037B2 - 大環状化合物およびそれらを製造し使用する方法 - Google Patents

大環状化合物およびそれらを製造し使用する方法 Download PDF

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Publication number
JP5383037B2
JP5383037B2 JP2007501005A JP2007501005A JP5383037B2 JP 5383037 B2 JP5383037 B2 JP 5383037B2 JP 2007501005 A JP2007501005 A JP 2007501005A JP 2007501005 A JP2007501005 A JP 2007501005A JP 5383037 B2 JP5383037 B2 JP 5383037B2
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group
alkyl
unsaturated
heteroatoms
aromatic
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Expired - Fee Related
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JP2007501005A
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Japanese (ja)
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JP2007525520A (ja
JP2007525520A5 (https=
Inventor
ジェイ ジェイ． ファーマー，
アショク バタチャージー，
イ チェン，
ジョエル エー． ゴールドバーグ，
ジョセフ エー． イッポリト，
ゾルタン エフ． カンヨ，
ロンリャン ロウ，
アデグボイガ ケー． オイレアー，
エドワード シー． シェレアー，
ジョイス エー． サトクリフィー，
デピン ワン，
ユシェン ウー，
ヤンミン デュ，
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Melinta Subsidiary Corp
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Rib X Pharmaceuticals Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10—Laxatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Pain & Pain Management (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Materials For Medical Uses (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP2007501005A 2004-02-27 2005-02-25 大環状化合物およびそれらを製造し使用する方法 Expired - Fee Related JP5383037B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US54828004P 2004-02-27 2004-02-27
US60/548,280 2004-02-27
US57594904P 2004-06-01 2004-06-01
US60/575,949 2004-06-01
PCT/US2005/006082 WO2005085266A2 (en) 2004-02-27 2005-02-25 Macrocyclic compounds and methods of making and using the same

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012034350A Division JP5631909B2 (ja) 2004-02-27 2012-02-20 大環状化合物およびそれらを製造し使用する方法

Publications (3)

Publication Number Publication Date
JP2007525520A JP2007525520A (ja) 2007-09-06
JP2007525520A5 JP2007525520A5 (https=) 2008-04-03
JP5383037B2 true JP5383037B2 (ja) 2014-01-08

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Family Applications (5)

Application Number Title Priority Date Filing Date
JP2007501005A Expired - Fee Related JP5383037B2 (ja) 2004-02-27 2005-02-25 大環状化合物およびそれらを製造し使用する方法
JP2012034350A Expired - Fee Related JP5631909B2 (ja) 2004-02-27 2012-02-20 大環状化合物およびそれらを製造し使用する方法
JP2014161364A Pending JP2014208707A (ja) 2004-02-27 2014-08-07 大環状化合物およびそれらを製造し使用する方法
JP2016136733A Pending JP2017019786A (ja) 2004-02-27 2016-07-11 大環状化合物およびそれらを製造し使用する方法
JP2018009418A Pending JP2018104437A (ja) 2004-02-27 2018-01-24 大環状化合物およびそれらを製造し使用する方法

Family Applications After (4)

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JP2012034350A Expired - Fee Related JP5631909B2 (ja) 2004-02-27 2012-02-20 大環状化合物およびそれらを製造し使用する方法
JP2014161364A Pending JP2014208707A (ja) 2004-02-27 2014-08-07 大環状化合物およびそれらを製造し使用する方法
JP2016136733A Pending JP2017019786A (ja) 2004-02-27 2016-07-11 大環状化合物およびそれらを製造し使用する方法
JP2018009418A Pending JP2018104437A (ja) 2004-02-27 2018-01-24 大環状化合物およびそれらを製造し使用する方法

Country Status (5)

Country Link
US (4) US8202843B2 (https=)
EP (2) EP1723159B1 (https=)
JP (5) JP5383037B2 (https=)
CN (1) CN102816194A (https=)
WO (1) WO2005085266A2 (https=)

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US20080045585A1 (en) 2008-02-21
WO2005085266A8 (en) 2005-12-01
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US20180066007A1 (en) 2018-03-08
CN102816194A (zh) 2012-12-12
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US20150158901A1 (en) 2015-06-11
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US20120252747A1 (en) 2012-10-04
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