JP5186219B2 - 置換アリールアミン化合物および５−ｈｔ６調節因子としてのその使用 - Google Patents

置換アリールアミン化合物および５−ｈｔ６調節因子としてのその使用 Download PDF

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JP5186219B2
JP5186219B2 JP2007552407A JP2007552407A JP5186219B2 JP 5186219 B2 JP5186219 B2 JP 5186219B2 JP 2007552407 A JP2007552407 A JP 2007552407A JP 2007552407 A JP2007552407 A JP 2007552407A JP 5186219 B2 JP5186219 B2 JP 5186219B2
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phenyl
mmol
piperazin
methylsulfonyl
ethyl
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JP2008528517A (ja
JP2008528517A5 (enExample
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オレン ベッカー，
メルセデス ロベラ，
ローザ イー． メレンデス，
アヌラグ シャラデンドゥ，
ローレンス ウー，
シャン ワイ． ユー，
デール エス． ダノア，
スリニバサ ラオ チェルク，
ヤエル マランツ，
シルビア ノイマン，
メラブ フィヒマン，
ハノヒ センデロウィッツ，
シャロン シャカム，
アシス サハ，
ピニ オーバック，
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エピックス デラウェア， インコーポレイテッド
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
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    • C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
JP2007552407A 2005-01-25 2006-01-25 置換アリールアミン化合物および５−ｈｔ６調節因子としてのその使用 Expired - Fee Related JP5186219B2 (ja)

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US64695705P 2005-01-25 2005-01-25
US60/646,957 2005-01-25
US70185305P 2005-07-22 2005-07-22
US60/701,853 2005-07-22
PCT/US2006/002718 WO2006081332A1 (en) 2005-01-25 2006-01-25 Substituted arylamine compounds and their use as 5-ht6 modulators

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JP5186219B2 true JP5186219B2 (ja) 2013-04-17

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US (2) US7968538B2 (enExample)
EP (1) EP1856075A1 (enExample)
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KR (1) KR20070097590A (enExample)
AU (1) AU2006209216A1 (enExample)
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CA (1) CA2595607C (enExample)
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US8808492B2 (en) 2011-12-20 2014-08-19 Industrial Technology Research Institute Method of joining superconductor materials

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EP1676842A1 (en) * 2004-12-30 2006-07-05 Laboratorios Del Dr. Esteve, S.A. Nitro-substituted phenyl-piperazine compounds, their preparation and use in medicaments
JP5186219B2 (ja) 2005-01-25 2013-04-17 エピックス デラウェア， インコーポレイテッド 置換アリールアミン化合物および５−ｈｔ６調節因子としてのその使用
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