JP5086987B2 - 臭素を使用するピラゾールへの２−ピラゾリンの変換 - Google Patents

臭素を使用するピラゾールへの２−ピラゾリンの変換 Download PDF

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Publication number
JP5086987B2
JP5086987B2 JP2008502077A JP2008502077A JP5086987B2 JP 5086987 B2 JP5086987 B2 JP 5086987B2 JP 2008502077 A JP2008502077 A JP 2008502077A JP 2008502077 A JP2008502077 A JP 2008502077A JP 5086987 B2 JP5086987 B2 JP 5086987B2
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JP
Japan
Prior art keywords
formula
compound
bromine
halogen
haloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP2008502077A
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English (en)
Japanese (ja)
Other versions
JP2008533169A5 (enExample
JP2008533169A (ja
Inventor
フアガン，ポール・ジヨセフ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
EIDP Inc
Original Assignee
EI Du Pont de Nemours and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by EI Du Pont de Nemours and Co filed Critical EI Du Pont de Nemours and Co
Publication of JP2008533169A publication Critical patent/JP2008533169A/ja
Publication of JP2008533169A5 publication Critical patent/JP2008533169A5/ja
Application granted granted Critical
Publication of JP5086987B2 publication Critical patent/JP5086987B2/ja
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Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Chemical Treatment Of Metals (AREA)
  • Enzymes And Modification Thereof (AREA)
JP2008502077A 2005-03-18 2006-03-14 臭素を使用するピラゾールへの２−ピラゾリンの変換 Expired - Lifetime JP5086987B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US66341005P 2005-03-18 2005-03-18
US60/663,410 2005-03-18
PCT/US2006/009617 WO2006102025A1 (en) 2005-03-18 2006-03-14 Conversion of 2-pyrazolines to pyrazoles using bromine

Publications (3)

Publication Number Publication Date
JP2008533169A JP2008533169A (ja) 2008-08-21
JP2008533169A5 JP2008533169A5 (enExample) 2009-04-23
JP5086987B2 true JP5086987B2 (ja) 2012-11-28

Family

ID=36592996

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008502077A Expired - Lifetime JP5086987B2 (ja) 2005-03-18 2006-03-14 臭素を使用するピラゾールへの２−ピラゾリンの変換

Country Status (20)

Country Link
US (1) US7951953B2 (enExample)
EP (1) EP1858878B1 (enExample)
JP (1) JP5086987B2 (enExample)
KR (1) KR101337159B1 (enExample)
CN (1) CN101142207B (enExample)
AT (1) ATE555103T1 (enExample)
AU (1) AU2006227484B2 (enExample)
BR (1) BRPI0609844B1 (enExample)
CA (1) CA2601870C (enExample)
DK (1) DK1858878T3 (enExample)
ES (1) ES2385496T3 (enExample)
IL (1) IL185329A (enExample)
MX (1) MX2007011162A (enExample)
PL (1) PL1858878T3 (enExample)
RS (2) RS20070369A (enExample)
RU (1) RU2410381C2 (enExample)
TW (1) TWI371449B (enExample)
UA (1) UA93869C2 (enExample)
WO (1) WO2006102025A1 (enExample)
ZA (1) ZA200707470B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2008002236A (es) * 2005-08-24 2008-03-27 Du Pont Antranilamidas para controlar plagas de invertebrados.
CN101550130B (zh) * 2008-04-01 2012-11-07 中国中化股份有限公司 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法
CN101863874B (zh) * 2009-04-14 2013-11-06 中国中化股份有限公司 一种吡唑亚胺类化合物及其应用
ES2555260T3 (es) 2010-06-15 2015-12-30 Bayer Intellectual Property Gmbh Derivados de diamida de ácido antranílico
TWI849253B (zh) * 2019-11-11 2024-07-21 美商富曼西公司 用於製備3-溴-1- (3-氯吡啶-2-基) -1h-吡唑-5-羧酸乙酯的方法
TWI884201B (zh) * 2020-01-08 2025-05-21 美商富曼西公司 用於製備3-溴-1-(3-氯吡啶-2-基)-1h-吡唑-5-羧酸乙酯的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5281571A (en) * 1990-10-18 1994-01-25 Monsanto Company Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles
TWI371450B (en) * 2001-08-13 2012-09-01 Du Pont Novel substituted dihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use
MY142967A (en) 2001-08-13 2011-01-31 Du Pont Method for controlling particular insect pests by applying anthranilamide compounds
TWI343376B (en) 2002-07-31 2011-06-11 Du Pont Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles

Also Published As

Publication number Publication date
TWI371449B (en) 2012-09-01
DK1858878T3 (da) 2012-08-06
RU2410381C2 (ru) 2011-01-27
ZA200707470B (en) 2008-12-31
AU2006227484A1 (en) 2006-09-28
PL1858878T3 (pl) 2012-09-28
TW200700407A (en) 2007-01-01
BRPI0609844A2 (pt) 2010-05-04
AU2006227484B2 (en) 2011-08-11
CN101142207A (zh) 2008-03-12
RS20070369A (sr) 2009-01-22
UA93869C2 (en) 2011-03-25
WO2006102025A1 (en) 2006-09-28
KR20070112292A (ko) 2007-11-22
RU2007138552A (ru) 2009-04-27
EP1858878B1 (en) 2012-04-25
CN101142207B (zh) 2011-10-05
BRPI0609844B1 (pt) 2015-06-30
MX2007011162A (es) 2007-10-17
IL185329A0 (en) 2008-02-09
CA2601870A1 (en) 2006-09-28
US7951953B2 (en) 2011-05-31
US20080177078A1 (en) 2008-07-24
EP1858878A1 (en) 2007-11-28
ATE555103T1 (de) 2012-05-15
CA2601870C (en) 2013-06-11
JP2008533169A (ja) 2008-08-21
ES2385496T3 (es) 2012-07-25
RS52344B (sr) 2012-12-31
KR101337159B1 (ko) 2013-12-05
IL185329A (en) 2013-04-30

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