JP4879757B2 - Ｃ１０シクロペンチルエステル置換タキサン - Google Patents

Ｃ１０シクロペンチルエステル置換タキサン Download PDF

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Publication number
JP4879757B2
JP4879757B2 JP2006553281A JP2006553281A JP4879757B2 JP 4879757 B2 JP4879757 B2 JP 4879757B2 JP 2006553281 A JP2006553281 A JP 2006553281A JP 2006553281 A JP2006553281 A JP 2006553281A JP 4879757 B2 JP4879757 B2 JP 4879757B2
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Japan
Prior art keywords
composition
tumor
taxane
administration
dosage unit
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Expired - Fee Related
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JP2006553281A
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English (en)
Japanese (ja)
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JP2007522236A (ja
JP2007522236A5 (https=
Inventor
ロバート・エイ・ホルトン
フォン・ブ
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Florida State University Research Foundation Inc
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Florida State University Research Foundation Inc
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Publication of JP2007522236A5 publication Critical patent/JP2007522236A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Epoxy Compounds (AREA)
JP2006553281A 2004-02-13 2005-02-14 Ｃ１０シクロペンチルエステル置換タキサン Expired - Fee Related JP4879757B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US54475504P 2004-02-13 2004-02-13
US60/544,755 2004-02-13
US61350304P 2004-09-27 2004-09-27
US60/613,503 2004-09-27
PCT/US2005/004442 WO2005079319A2 (en) 2004-02-13 2005-02-14 C10 cyclopentyl ester substituted taxanes

Publications (3)

Publication Number Publication Date
JP2007522236A JP2007522236A (ja) 2007-08-09
JP2007522236A5 JP2007522236A5 (https=) 2008-04-03
JP4879757B2 true JP4879757B2 (ja) 2012-02-22

Family

ID=34890477

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006553281A Expired - Fee Related JP4879757B2 (ja) 2004-02-13 2005-02-14 Ｃ１０シクロペンチルエステル置換タキサン

Country Status (21)

Country Link
US (2) US7589111B2 (https=)
EP (1) EP1713798B1 (https=)
JP (1) JP4879757B2 (https=)
KR (1) KR101169818B1 (https=)
AR (1) AR047704A1 (https=)
AT (1) ATE486596T1 (https=)
AU (1) AU2005214065B2 (https=)
BR (1) BRPI0507671A (https=)
CA (1) CA2556200C (https=)
CR (1) CR8554A (https=)
DE (1) DE602005024518D1 (https=)
EC (1) ECSP066765A (https=)
HN (1) HN2005000054A (https=)
IL (1) IL177372A (https=)
NO (1) NO20064090L (https=)
NZ (1) NZ548769A (https=)
PE (1) PE20050693A1 (https=)
RU (1) RU2006132741A (https=)
SV (1) SV2006002010A (https=)
TW (1) TWI353354B (https=)
WO (1) WO2005079319A2 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1303077C (zh) * 2004-01-16 2007-03-07 桂林晖昂生化药业有限责任公司 合成紫杉烷的制备工艺
JP4833126B2 (ja) * 2007-03-26 2011-12-07 Ｎｔｎ株式会社 潤滑剤劣化検出装置および検出装置付き軸受
CN113209287B (zh) * 2021-02-04 2022-07-08 中国农业科学院农业环境与可持续发展研究所 油包水型纳米疫苗佐剂、制备方法及其应用

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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JP2003055360A (ja) * 2001-07-31 2003-02-26 Florida State Univ Research Foundation Inc Ｃ１０エステル置換タキサン
JP2003521545A (ja) * 2000-02-02 2003-07-15 フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド 改良された溶解性を有するタキサン製剤

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JP2003055360A (ja) * 2001-07-31 2003-02-26 Florida State Univ Research Foundation Inc Ｃ１０エステル置換タキサン

Also Published As

Publication number Publication date
AU2005214065A1 (en) 2005-09-01
JP2007522236A (ja) 2007-08-09
EP1713798A2 (en) 2006-10-25
ECSP066765A (es) 2006-12-29
EP1713798B1 (en) 2010-11-03
RU2006132741A (ru) 2008-03-20
US7589111B2 (en) 2009-09-15
KR20060129018A (ko) 2006-12-14
US8003812B2 (en) 2011-08-23
NO20064090L (no) 2006-11-10
CR8554A (es) 2008-04-25
IL177372A (en) 2011-09-27
TWI353354B (en) 2011-12-01
US20050228037A1 (en) 2005-10-13
AU2005214065B2 (en) 2009-11-12
US20100056614A1 (en) 2010-03-04
ATE486596T1 (de) 2010-11-15
BRPI0507671A (pt) 2007-07-17
SV2006002010A (es) 2006-08-23
PE20050693A1 (es) 2005-09-27
HK1097534A1 (en) 2007-06-29
NZ548769A (en) 2009-10-30
EP1713798A4 (en) 2007-12-05
DE602005024518D1 (en) 2010-12-16
CA2556200C (en) 2012-06-26
IL177372A0 (en) 2006-12-10
AR047704A1 (es) 2006-02-08
WO2005079319A3 (en) 2005-11-17
AU2005214065A2 (en) 2005-09-01
TW200530209A (en) 2005-09-16
WO2005079319A2 (en) 2005-09-01
CA2556200A1 (en) 2005-09-01
KR101169818B1 (ko) 2012-07-30
HN2005000054A (es) 2009-02-18

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