DE602005024518D1 - C10-cyclopentylester-substituierte taxane - Google Patents

C10-cyclopentylester-substituierte taxane

Info

Publication number
DE602005024518D1
DE602005024518D1 DE602005024518T DE602005024518T DE602005024518D1 DE 602005024518 D1 DE602005024518 D1 DE 602005024518D1 DE 602005024518 T DE602005024518 T DE 602005024518T DE 602005024518 T DE602005024518 T DE 602005024518T DE 602005024518 D1 DE602005024518 D1 DE 602005024518D1
Authority
DE
Germany
Prior art keywords
cyclopentylester
substituierte
taxane
substituierte taxane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE602005024518T
Other languages
German (de)
English (en)
Inventor
Robert A Holton
Phong Taxolog Vu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Florida State University Research Foundation Inc
Original Assignee
Florida State University Research Foundation Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Florida State University Research Foundation Inc filed Critical Florida State University Research Foundation Inc
Publication of DE602005024518D1 publication Critical patent/DE602005024518D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Epoxy Compounds (AREA)
DE602005024518T 2004-02-13 2005-02-14 C10-cyclopentylester-substituierte taxane Expired - Lifetime DE602005024518D1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US54475504P 2004-02-13 2004-02-13
US61350304P 2004-09-27 2004-09-27
PCT/US2005/004442 WO2005079319A2 (en) 2004-02-13 2005-02-14 C10 cyclopentyl ester substituted taxanes

Publications (1)

Publication Number Publication Date
DE602005024518D1 true DE602005024518D1 (en) 2010-12-16

Family

ID=34890477

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602005024518T Expired - Lifetime DE602005024518D1 (en) 2004-02-13 2005-02-14 C10-cyclopentylester-substituierte taxane

Country Status (21)

Country Link
US (2) US7589111B2 (https=)
EP (1) EP1713798B1 (https=)
JP (1) JP4879757B2 (https=)
KR (1) KR101169818B1 (https=)
AR (1) AR047704A1 (https=)
AT (1) ATE486596T1 (https=)
AU (1) AU2005214065B2 (https=)
BR (1) BRPI0507671A (https=)
CA (1) CA2556200C (https=)
CR (1) CR8554A (https=)
DE (1) DE602005024518D1 (https=)
EC (1) ECSP066765A (https=)
HN (1) HN2005000054A (https=)
IL (1) IL177372A (https=)
NO (1) NO20064090L (https=)
NZ (1) NZ548769A (https=)
PE (1) PE20050693A1 (https=)
RU (1) RU2006132741A (https=)
SV (1) SV2006002010A (https=)
TW (1) TWI353354B (https=)
WO (1) WO2005079319A2 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1303077C (zh) * 2004-01-16 2007-03-07 桂林晖昂生化药业有限责任公司 合成紫杉烷的制备工艺
JP4833126B2 (ja) * 2007-03-26 2011-12-07 Ｎｔｎ株式会社 潤滑剤劣化検出装置および検出装置付き軸受
CN113209287B (zh) * 2021-02-04 2022-07-08 中国农业科学院农业环境与可持续发展研究所 油包水型纳米疫苗佐剂、制备方法及其应用

Family Cites Families (71)

* Cited by examiner, † Cited by third party
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US5283253A (en) 1991-09-23 1994-02-01 Florida State University Furyl or thienyl carbonyl substituted taxanes and pharmaceutical compositions containing them
US5714513A (en) 1991-09-23 1998-02-03 Florida State University C10 taxane derivatives and pharmaceutical compositions
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US5739362A (en) 1991-09-23 1998-04-14 Florida State University Taxanes having an alkoxy, alkenoxy or aryloxy substituted side-chain and pharmaceutical compositions containing them
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US5430160A (en) 1991-09-23 1995-07-04 Florida State University Preparation of substituted isoserine esters using β-lactams and metal or ammonium alkoxides
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US5274124A (en) 1991-09-23 1993-12-28 Florida State University Metal alkoxides
US5445908A (en) 1991-10-17 1995-08-29 Matsushita Electric Industrial Co., Ltd. Alkaline dry cell
DK0552041T3 (da) 1992-01-15 2000-10-09 Squibb & Sons Inc Enzymatiske fremgangsmåder til spaltning af enantiomerblandinger af forbindelser, der er nyttige som mellemprodukter ved fr
US5272171A (en) 1992-02-13 1993-12-21 Bristol-Myers Squibb Company Phosphonooxy and carbonate derivatives of taxol
US5200534A (en) 1992-03-13 1993-04-06 University Of Florida Process for the preparation of taxol and 10-deacetyltaxol
FR2691460B1 (fr) 1992-05-21 1994-07-22 Rhone Poulenc Rorer Sa Nouveaux derives du taxane, leur preparation et les compositions qui les contiennent.
US5254580A (en) 1993-01-19 1993-10-19 Bristol-Myers Squibb Company 7,8-cyclopropataxanes
CA2100808A1 (en) 1992-10-01 1994-04-02 Vittorio Farina Deoxy paclitaxels
FR2696461B1 (fr) 1992-10-05 1994-11-10 Rhone Poulenc Rorer Sa Nouveaux dérivés d'analogues du taxol, leur préparation et les compositions qui les contiennent.
CA2109861C (en) * 1992-12-04 1999-03-16 Shu-Hui Chen 6,7-modified paclitaxels
IL107950A (en) 1992-12-15 2001-04-30 Upjohn Co 7β, 8β - METHANO-TAXOLS, THEIR PREPARATION AND ANTINEOPLASTIC PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
MX9308012A (es) 1992-12-24 1994-08-31 Bristol Myers Squibb Co Eteres fosfonooximetilicos de derivados de taxano, solubles en agua y composiciones farmaceuticas que los incluyen.
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FR2702212B1 (fr) 1993-03-02 1995-04-07 Rhone Poulenc Rorer Sa Nouveaux taxoïdes, leur préparation et les compositions pharmaceutiques qui les contiennent.
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WO1995004154A1 (en) 1993-07-27 1995-02-09 Nippon Steel Corporation Process for producing taxol and its analogues using microorganisms
CA2129288C (en) 1993-08-17 2000-05-16 Jerzy Golik Phosphonooxymethyl esters of taxane derivatives
DE69507702T2 (de) 1994-07-26 1999-08-26 Indena S.P.A. Semisynthetisch taxal derivate mit antitumor wirkung
US6100411A (en) 1994-10-28 2000-08-08 The Research Foundation Of State University Of New York Taxoid anti-tumor agents and pharmaceutical compositions thereof
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MA23823A1 (fr) 1995-03-27 1996-10-01 Aventis Pharma Sa Nouveaux taxoides, leur preparation et les compositions qui les contiennent
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FR2732968B1 (fr) 1995-04-14 1997-05-16 Rhone Poulenc Rorer Sa Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
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JP2003522171A (ja) 2000-02-02 2003-07-22 フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド 抗腫瘍剤としてのｃ１０カーボネート置換タキサン
HUP0600302A2 (en) 2000-02-02 2006-07-28 Univ Florida State Res Found C10 ester substituted taxanes as antitumor agents
KR20010111580A (ko) 2000-02-02 2001-12-19 플로리다 스테이트 유니버시티 리서치 파운데이션, 인크 개선된 용해도를 갖는 탁산 제형물
CA2367661A1 (en) 2000-02-02 2001-08-09 Robert A. Holton Taxane formulations having improved solubility
IT1319168B1 (it) 2000-03-17 2003-09-26 Indena Spa Derivati di condensazione ad attivita' antitumorale, loro metodo dipreparazione e formulazioni che li contengono.
JP4717252B2 (ja) * 2001-04-25 2011-07-06 株式会社小松製作所 プレスのスライド駆動装置
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CA2808297C (en) * 2010-08-13 2018-09-18 Roilblue Corporation Oil containment assembly and method of using same

Also Published As

Publication number Publication date
AU2005214065A1 (en) 2005-09-01
JP2007522236A (ja) 2007-08-09
EP1713798A2 (en) 2006-10-25
ECSP066765A (es) 2006-12-29
EP1713798B1 (en) 2010-11-03
RU2006132741A (ru) 2008-03-20
US7589111B2 (en) 2009-09-15
KR20060129018A (ko) 2006-12-14
US8003812B2 (en) 2011-08-23
NO20064090L (no) 2006-11-10
CR8554A (es) 2008-04-25
IL177372A (en) 2011-09-27
TWI353354B (en) 2011-12-01
US20050228037A1 (en) 2005-10-13
AU2005214065B2 (en) 2009-11-12
US20100056614A1 (en) 2010-03-04
ATE486596T1 (de) 2010-11-15
BRPI0507671A (pt) 2007-07-17
SV2006002010A (es) 2006-08-23
PE20050693A1 (es) 2005-09-27
HK1097534A1 (en) 2007-06-29
JP4879757B2 (ja) 2012-02-22
NZ548769A (en) 2009-10-30
EP1713798A4 (en) 2007-12-05
CA2556200C (en) 2012-06-26
IL177372A0 (en) 2006-12-10
AR047704A1 (es) 2006-02-08
WO2005079319A3 (en) 2005-11-17
AU2005214065A2 (en) 2005-09-01
TW200530209A (en) 2005-09-16
WO2005079319A2 (en) 2005-09-01
CA2556200A1 (en) 2005-09-01
KR101169818B1 (ko) 2012-07-30
HN2005000054A (es) 2009-02-18

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