JP4809244B2 - ヨードニウム塩のフッ素化におけるラジカル捕捉剤 - Google Patents

ヨードニウム塩のフッ素化におけるラジカル捕捉剤 Download PDF

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Publication number
JP4809244B2
JP4809244B2 JP2006546303A JP2006546303A JP4809244B2 JP 4809244 B2 JP4809244 B2 JP 4809244B2 JP 2006546303 A JP2006546303 A JP 2006546303A JP 2006546303 A JP2006546303 A JP 2006546303A JP 4809244 B2 JP4809244 B2 JP 4809244B2
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Japan
Prior art keywords
fluorine
reaction
labeled compound
mmol
fluoride
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JP2006546303A
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English (en)
Japanese (ja)
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JP2007515465A (ja
JP2007515465A5 (enExample
Inventor
ワッズワース，ハリー・ジョン
ウィッドウソン，デイビッド・アーサー
ウィルソン，エマニュエル
キャロル，マイケル・アンドリュー
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GE Healthcare Ltd
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GE Healthcare Ltd
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Liquid Crystal (AREA)
  • Saccharide Compounds (AREA)
  • Seasonings (AREA)
JP2006546303A 2003-12-23 2004-12-17 ヨードニウム塩のフッ素化におけるラジカル捕捉剤 Expired - Fee Related JP4809244B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0329716.5A GB0329716D0 (en) 2003-12-23 2003-12-23 Radical trap
GB0329716.5 2003-12-23
PCT/GB2004/005304 WO2005061415A1 (en) 2003-12-23 2004-12-17 Radical trap in fluoridation of iodonium salt

Publications (3)

Publication Number Publication Date
JP2007515465A JP2007515465A (ja) 2007-06-14
JP2007515465A5 JP2007515465A5 (enExample) 2008-02-14
JP4809244B2 true JP4809244B2 (ja) 2011-11-09

Family

ID=30776291

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006546303A Expired - Fee Related JP4809244B2 (ja) 2003-12-23 2004-12-17 ヨードニウム塩のフッ素化におけるラジカル捕捉剤

Country Status (9)

Country Link
US (1) US7642373B2 (enExample)
EP (1) EP1697279B1 (enExample)
JP (1) JP4809244B2 (enExample)
CN (1) CN100415696C (enExample)
AT (1) ATE409173T1 (enExample)
DE (1) DE602004016771D1 (enExample)
ES (1) ES2313117T3 (enExample)
GB (1) GB0329716D0 (enExample)
WO (1) WO2005061415A1 (enExample)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0407952D0 (en) * 2004-04-08 2004-05-12 Amersham Plc Fluoridation method
GB0525949D0 (en) * 2005-12-21 2006-02-01 Hammersmith Imanet Ltd Pet radiotracers
EP2192928A4 (en) * 2007-10-03 2011-04-06 Ge Healthcare Ltd PERFLUOR ARYLIODONIUM SALTS IN A NUCLEOPHILIC AROMATIC 18F FLUORATION
RU2475448C2 (ru) * 2008-01-03 2013-02-20 ДжиИ ХЕЛТКЕР ЛИМИТЕД Способ обработки фторида
GB0808986D0 (en) 2008-05-16 2008-06-25 Univ Newcastle Formation of 18F and 19F fluoroarenes bearing reactive functionalities
WO2010015340A1 (en) * 2008-08-06 2010-02-11 Bayer Schering Pharma Aktiengesellschaft Daa-pyridine as peripheral benzodiazepine receptor ligand for diagnostic imaging and pharmaceutical treatment
GB0814893D0 (en) * 2008-08-14 2008-09-17 Ge Healthcare Ltd Improved fluoridation of iodonium salts
ES2861578T3 (es) 2008-10-21 2021-10-06 Nutech Ventures Fluoración de sistemas de anillos aromáticos
US9302990B2 (en) 2008-10-21 2016-04-05 Nutech Ventures Fluorination of aromatic ring systems
GB0905438D0 (en) 2009-03-30 2009-05-13 Ge Healthcare Ltd Radiolabelling reagents and methods
WO2010117435A2 (en) * 2009-04-08 2010-10-14 The Regents Of The University Of California No-carrier-added nucleophilic [f-18] fluorination of aromatic compounds
US8377704B2 (en) 2009-10-20 2013-02-19 Nutech Ventures Detection and quantification of anions
US8546578B2 (en) 2010-02-04 2013-10-01 Nutech Ventures Iodonium Cyclophanes for SECURE arene functionalization
WO2011141515A1 (en) 2010-05-14 2011-11-17 Bayer Pharma Aktiengesellschaft Diagnostic agents for amyloid beta imaging
KR101441406B1 (ko) * 2011-05-25 2014-11-04 주식회사 바이오이미징코리아 디아릴이오도늄 염 전구체를 이용한 플로오린-18이 표지된 플루마제닐의 제조 방법
CA2889575A1 (en) * 2012-10-27 2014-05-01 Ground Fluor Pharmaceuticals, Inc. Processes and reagents for making diaryliodonium salts
EP2821383B1 (en) * 2013-07-02 2017-08-30 Trasis S.A. Stabilization of radiosynthetic intermediates
US10071943B2 (en) * 2014-04-11 2018-09-11 The Regents Of The University Of Michigan Copper catalyzed [18F]fluorination of iodonium salts
CN105237483B (zh) * 2015-11-10 2018-04-20 东华大学 一种对称型嘧啶基碘鎓盐及其制备方法
FR3054445B1 (fr) * 2016-07-26 2019-07-05 Laboratoires Cyclopharma Synthese d'une composition d'agent radioactif
US10695450B2 (en) 2016-07-26 2020-06-30 Laboratoires Cyclopharma Synthesis of a radioactive agent composition
CU20200039A7 (es) 2017-10-24 2021-03-11 Lunella Biotech Inc Mitoflavoscinas: la fijación como objetivo de enzimas que contienen flavina elimina células madre cancerosas (cscs) al inhibir la respiración mitocrondrial
GB201805253D0 (en) * 2018-03-29 2018-05-16 Ge Healthcare Ltd Ip Solid phase extraction
JP7558694B2 (ja) * 2019-07-01 2024-10-01 住友化学株式会社 塩、酸発生剤、レジスト組成物及びレジストパターンの製造方法
JP7556709B2 (ja) * 2019-07-01 2024-09-26 住友化学株式会社 カルボン酸塩、カルボン酸発生剤、レジスト組成物及びレジストパターンの製造方法
JP2021008455A (ja) * 2019-07-01 2021-01-28 住友化学株式会社 カルボン酸塩、カルボン酸発生剤、レジスト組成物及びレジストパターンの製造方法
JP7627551B2 (ja) * 2019-07-01 2025-02-06 住友化学株式会社 塩、酸発生剤、レジスト組成物及びレジストパターンの製造方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS52133994A (en) * 1976-04-29 1977-11-09 Daikin Ind Ltd Method of fluorination
JP3165775B2 (ja) * 1994-08-31 2001-05-14 日本鋼管株式会社 フッ素放射性同位元素標識ｌ−ドーパの製造方法
JP3171036B2 (ja) * 1994-11-16 2001-05-28 日本鋼管株式会社 フッ素放射性同位元素標識ドーパミンの製造方法
GB0115927D0 (en) * 2001-06-29 2001-08-22 Nycomed Amersham Plc Solid-phase nucleophilic fluorination
GB0206750D0 (en) * 2002-03-22 2002-05-01 Amersham Plc Radiofluorination methods
DE10346228B4 (de) * 2003-09-25 2009-04-09 Eberhard-Karls-Universität Tübingen Universitätsklinikum Herstellung von [18F]fluormarkierten aromatischen L-Aminosäuren
GB0407952D0 (en) * 2004-04-08 2004-05-12 Amersham Plc Fluoridation method

Also Published As

Publication number Publication date
EP1697279A1 (en) 2006-09-06
ATE409173T1 (de) 2008-10-15
US7642373B2 (en) 2010-01-05
CN100415696C (zh) 2008-09-03
WO2005061415A1 (en) 2005-07-07
CN1898184A (zh) 2007-01-17
JP2007515465A (ja) 2007-06-14
US20060292060A1 (en) 2006-12-28
DE602004016771D1 (de) 2008-11-06
GB0329716D0 (en) 2004-01-28
EP1697279B1 (en) 2008-09-24
ES2313117T3 (es) 2009-03-01

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