JP4725939B2 - １−アルキル−ピラゾール−５−カルボン酸エステルｉｉｉの製造方法 - Google Patents

１−アルキル−ピラゾール−５−カルボン酸エステルｉｉｉの製造方法 Download PDF

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Publication number
JP4725939B2
JP4725939B2 JP2000566252A JP2000566252A JP4725939B2 JP 4725939 B2 JP4725939 B2 JP 4725939B2 JP 2000566252 A JP2000566252 A JP 2000566252A JP 2000566252 A JP2000566252 A JP 2000566252A JP 4725939 B2 JP4725939 B2 JP 4725939B2
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JP
Japan
Prior art keywords
formula
alkyl
represented
pyrazole
ethyl
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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JP2000566252A
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English (en)
Japanese (ja)
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JP2002523401A5 (enExample
JP2002523401A (ja
Inventor
ミユラー，ニコラウス
マツケ，ミヒヤエル
Original Assignee
ランクセス・ドイチュランド・ゲーエムベーハー
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Publication of JP2002523401A publication Critical patent/JP2002523401A/ja
Publication of JP2002523401A5 publication Critical patent/JP2002523401A5/ja
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/67—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
    • C07C69/716—Esters of keto-carboxylic acids or aldehydo-carboxylic acids

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2000566252A 1998-08-17 1999-08-04 １−アルキル−ピラゾール−５−カルボン酸エステルｉｉｉの製造方法 Expired - Fee Related JP4725939B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19837067.9 1998-08-17
DE19837067A DE19837067A1 (de) 1998-08-17 1998-08-17 Verfahren zur Herstellung von 1-Alkyl-pyrazol-5-carbonsäureestern
PCT/EP1999/005641 WO2000010978A1 (de) 1998-08-17 1999-08-04 Verfahren zur herstellung von 1-alkyl-pyrazol-5-carbonsäureestern iii

Publications (3)

Publication Number Publication Date
JP2002523401A JP2002523401A (ja) 2002-07-30
JP2002523401A5 JP2002523401A5 (enExample) 2006-09-28
JP4725939B2 true JP4725939B2 (ja) 2011-07-13

Family

ID=7877651

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000566252A Expired - Fee Related JP4725939B2 (ja) 1998-08-17 1999-08-04 １−アルキル−ピラゾール−５−カルボン酸エステルｉｉｉの製造方法

Country Status (13)

Country Link
US (1) US6444828B1 (enExample)
EP (1) EP1104406B1 (enExample)
JP (1) JP4725939B2 (enExample)
KR (1) KR20010072709A (enExample)
CN (1) CN1192023C (enExample)
AT (1) ATE310730T1 (enExample)
CA (1) CA2340704A1 (enExample)
CZ (1) CZ2001615A3 (enExample)
DE (2) DE19837067A1 (enExample)
HU (1) HUP0103116A3 (enExample)
IL (1) IL141281A0 (enExample)
PL (1) PL346016A1 (enExample)
WO (1) WO2000010978A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0016787D0 (en) 2000-07-07 2000-08-30 Pfizer Ltd Compounds useful in therapy
FR2826592B1 (fr) * 2001-06-27 2003-08-15 Bio Merieux Procede, dispositif, et equipement de separation par voie humide de micro particules magnetiques
CN101977889B (zh) * 2008-03-18 2013-12-04 三井化学Agro株式会社 含氟酰基乙酸衍生物的制备方法、含氟吡唑甲酸酯衍生物的制备方法及含氟吡唑甲酸衍生物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3557095A (en) 1968-05-31 1971-01-19 Parke Davis & Co Pyrazolodiazepinone compounds
ES8203350A1 (es) 1979-11-16 1982-04-01 Morishita Pharma Procedimiento para la fabricacion de derivados del pirazol
JPS5673069A (en) * 1979-11-16 1981-06-17 Morishita Seiyaku Kk Pyrazolecarboxylic acid derivative
JP2743461B2 (ja) 1989-05-08 1998-04-22 三菱化学株式会社 １―メチル―３―アルキル―５―ピラゾールカルボン酸エステル類の製造法
US5250534A (en) 1990-06-20 1993-10-05 Pfizer Inc. Pyrazolopyrimidinone antianginal agents
JP3006091B2 (ja) * 1990-12-25 2000-02-07 日本ヒドラジン工業株式会社 置換ピラゾールの製造方法
GB9114760D0 (en) 1991-07-09 1991-08-28 Pfizer Ltd Therapeutic agents
GB9311920D0 (en) 1993-06-09 1993-07-28 Pfizer Ltd Therapeutic agents
JP3491344B2 (ja) * 1993-08-31 2004-01-26 宇部興産株式会社 １−アルキル−５−ピラゾールカルボン酸エステル類の製法
DE19701277A1 (de) * 1997-01-16 1998-07-23 Bayer Ag Verfahren zur Herstellung von 1-Alkyl-pyrazol-5-carbonsäureestern

Also Published As

Publication number Publication date
HUP0103116A3 (en) 2002-05-28
CZ2001615A3 (cs) 2001-09-12
ATE310730T1 (de) 2005-12-15
CN1312801A (zh) 2001-09-12
KR20010072709A (ko) 2001-07-31
DE59912831D1 (de) 2005-12-29
HUP0103116A2 (hu) 2002-04-29
IL141281A0 (en) 2002-03-10
CA2340704A1 (en) 2000-03-02
EP1104406B1 (de) 2005-11-23
PL346016A1 (en) 2002-01-14
EP1104406A1 (de) 2001-06-06
WO2000010978A8 (de) 2001-05-10
DE19837067A1 (de) 2000-02-24
JP2002523401A (ja) 2002-07-30
WO2000010978A1 (de) 2000-03-02
CN1192023C (zh) 2005-03-09
US6444828B1 (en) 2002-09-03

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