CN1192023C - 制备1-烷基吡唑-5-羧酸酯iii的方法 - Google Patents

制备1-烷基吡唑-5-羧酸酯iii的方法 Download PDF

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Publication number
CN1192023C
CN1192023C CNB998097276A CN99809727A CN1192023C CN 1192023 C CN1192023 C CN 1192023C CN B998097276 A CNB998097276 A CN B998097276A CN 99809727 A CN99809727 A CN 99809727A CN 1192023 C CN1192023 C CN 1192023C
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CN
China
Prior art keywords
formula
alkyl
iii
optionally halogenated
alkylhydrazine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CNB998097276A
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English (en)
Chinese (zh)
Other versions
CN1312801A (zh
Inventor
N·米勒
M·马茨克
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Saltigo GmbH
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of CN1312801A publication Critical patent/CN1312801A/zh
Application granted granted Critical
Publication of CN1192023C publication Critical patent/CN1192023C/zh
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/67Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
    • C07C69/716Esters of keto-carboxylic acids or aldehydo-carboxylic acids

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CNB998097276A 1998-08-17 1999-08-04 制备1-烷基吡唑-5-羧酸酯iii的方法 Expired - Fee Related CN1192023C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19837067.9 1998-08-17
DE19837067A DE19837067A1 (de) 1998-08-17 1998-08-17 Verfahren zur Herstellung von 1-Alkyl-pyrazol-5-carbonsäureestern

Publications (2)

Publication Number Publication Date
CN1312801A CN1312801A (zh) 2001-09-12
CN1192023C true CN1192023C (zh) 2005-03-09

Family

ID=7877651

Family Applications (1)

Application Number Title Priority Date Filing Date
CNB998097276A Expired - Fee Related CN1192023C (zh) 1998-08-17 1999-08-04 制备1-烷基吡唑-5-羧酸酯iii的方法

Country Status (13)

Country Link
US (1) US6444828B1 (enExample)
EP (1) EP1104406B1 (enExample)
JP (1) JP4725939B2 (enExample)
KR (1) KR20010072709A (enExample)
CN (1) CN1192023C (enExample)
AT (1) ATE310730T1 (enExample)
CA (1) CA2340704A1 (enExample)
CZ (1) CZ2001615A3 (enExample)
DE (2) DE19837067A1 (enExample)
HU (1) HUP0103116A3 (enExample)
IL (1) IL141281A0 (enExample)
PL (1) PL346016A1 (enExample)
WO (1) WO2000010978A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0016787D0 (en) 2000-07-07 2000-08-30 Pfizer Ltd Compounds useful in therapy
FR2826592B1 (fr) * 2001-06-27 2003-08-15 Bio Merieux Procede, dispositif, et equipement de separation par voie humide de micro particules magnetiques
CN101977889B (zh) * 2008-03-18 2013-12-04 三井化学Agro株式会社 含氟酰基乙酸衍生物的制备方法、含氟吡唑甲酸酯衍生物的制备方法及含氟吡唑甲酸衍生物的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3557095A (en) 1968-05-31 1971-01-19 Parke Davis & Co Pyrazolodiazepinone compounds
ES8203350A1 (es) 1979-11-16 1982-04-01 Morishita Pharma Procedimiento para la fabricacion de derivados del pirazol
JPS5673069A (en) * 1979-11-16 1981-06-17 Morishita Seiyaku Kk Pyrazolecarboxylic acid derivative
JP2743461B2 (ja) 1989-05-08 1998-04-22 三菱化学株式会社 1―メチル―3―アルキル―5―ピラゾールカルボン酸エステル類の製造法
US5250534A (en) 1990-06-20 1993-10-05 Pfizer Inc. Pyrazolopyrimidinone antianginal agents
JP3006091B2 (ja) * 1990-12-25 2000-02-07 日本ヒドラジン工業株式会社 置換ピラゾールの製造方法
GB9114760D0 (en) 1991-07-09 1991-08-28 Pfizer Ltd Therapeutic agents
GB9311920D0 (en) 1993-06-09 1993-07-28 Pfizer Ltd Therapeutic agents
JP3491344B2 (ja) * 1993-08-31 2004-01-26 宇部興産株式会社 1−アルキル−5−ピラゾールカルボン酸エステル類の製法
DE19701277A1 (de) * 1997-01-16 1998-07-23 Bayer Ag Verfahren zur Herstellung von 1-Alkyl-pyrazol-5-carbonsäureestern

Also Published As

Publication number Publication date
HUP0103116A3 (en) 2002-05-28
CZ2001615A3 (cs) 2001-09-12
ATE310730T1 (de) 2005-12-15
CN1312801A (zh) 2001-09-12
KR20010072709A (ko) 2001-07-31
DE59912831D1 (de) 2005-12-29
HUP0103116A2 (hu) 2002-04-29
IL141281A0 (en) 2002-03-10
CA2340704A1 (en) 2000-03-02
EP1104406B1 (de) 2005-11-23
PL346016A1 (en) 2002-01-14
EP1104406A1 (de) 2001-06-06
WO2000010978A8 (de) 2001-05-10
JP4725939B2 (ja) 2011-07-13
DE19837067A1 (de) 2000-02-24
JP2002523401A (ja) 2002-07-30
WO2000010978A1 (de) 2000-03-02
US6444828B1 (en) 2002-09-03

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C06 Publication
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ASS Succession or assignment of patent right

Owner name: LANXESS DEUTSCHLAND GMBH

Free format text: FORMER OWNER: BAYER AG

Effective date: 20070525

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Effective date of registration: 20070525

Address after: Germany Leverkusen

Patentee after: Lanxess Deutschland GmbH

Address before: Germany Leverkusen

Patentee before: Bayer Aktiengesellschaft

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Owner name: SALTIGO GMBH

Free format text: FORMER OWNER: LANXESS DEUTSCHLAND GMBH

Effective date: 20081024

C41 Transfer of patent application or patent right or utility model
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Effective date of registration: 20081024

Address after: Germany Langenfeld

Patentee after: Saltigo GmbH

Address before: Germany Leverkusen

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CF01 Termination of patent right due to non-payment of annual fee

Granted publication date: 20050309

Termination date: 20150804

EXPY Termination of patent right or utility model