JP4630662B2 - Ｉ．Ａ．慢性関節リウマチの治療においてｐ３８キナーゼ阻害剤として使用される縮合ヘテロアリール誘導体 - Google Patents

Ｉ．Ａ．慢性関節リウマチの治療においてｐ３８キナーゼ阻害剤として使用される縮合ヘテロアリール誘導体 Download PDF

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JP4630662B2
JP4630662B2 JP2004523985A JP2004523985A JP4630662B2 JP 4630662 B2 JP4630662 B2 JP 4630662B2 JP 2004523985 A JP2004523985 A JP 2004523985A JP 2004523985 A JP2004523985 A JP 2004523985A JP 4630662 B2 JP4630662 B2 JP 4630662B2
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cyclopropyl
methyl
indazol
alkyl
optionally substituted
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JP2005538100A5 (https=
JP2005538100A (ja
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アンゲル，リチャード，マーティン
ボールドウィン，イアン，ロバート
バムボロー，ポール
デボエック，ニゲル，マーク
ロングスタッフ，ティモシー
スワンソン，スティーブン
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スミスクライン ビーチャム コーポレーション
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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
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    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Biomedical Technology (AREA)
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  • Tropical Medicine & Parasitology (AREA)
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JP2004523985A 2002-07-31 2003-07-30 Ｉ．Ａ．慢性関節リウマチの治療においてｐ３８キナーゼ阻害剤として使用される縮合ヘテロアリール誘導体 Expired - Fee Related JP4630662B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0217757.4A GB0217757D0 (en) 2002-07-31 2002-07-31 Novel compounds
PCT/GB2003/003316 WO2004010995A1 (en) 2002-07-31 2003-07-30 Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of i.a. rheumatoid arthristis

Publications (3)

Publication Number Publication Date
JP2005538100A JP2005538100A (ja) 2005-12-15
JP2005538100A5 JP2005538100A5 (https=) 2006-07-27
JP4630662B2 true JP4630662B2 (ja) 2011-02-09

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JP2004523985A Expired - Fee Related JP4630662B2 (ja) 2002-07-31 2003-07-30 Ｉ．Ａ．慢性関節リウマチの治療においてｐ３８キナーゼ阻害剤として使用される縮合ヘテロアリール誘導体

Country Status (9)

Country Link
US (1) US7642276B2 (https=)
EP (1) EP1531812B1 (https=)
JP (1) JP4630662B2 (https=)
AT (1) ATE365551T1 (https=)
AU (1) AU2003248978A1 (https=)
DE (1) DE60314639T2 (https=)
ES (1) ES2289336T3 (https=)
GB (1) GB0217757D0 (https=)
WO (1) WO2004010995A1 (https=)

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