JP3719679B2 - プラバスタチンナトリウム錠 - Google Patents
プラバスタチンナトリウム錠 Download PDFInfo
- Publication number
- JP3719679B2 JP3719679B2 JP2003303781A JP2003303781A JP3719679B2 JP 3719679 B2 JP3719679 B2 JP 3719679B2 JP 2003303781 A JP2003303781 A JP 2003303781A JP 2003303781 A JP2003303781 A JP 2003303781A JP 3719679 B2 JP3719679 B2 JP 3719679B2
- Authority
- JP
- Japan
- Prior art keywords
- pravastatin sodium
- tablet
- mannitol
- tablets
- sodium
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
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- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Description
処方例1(1錠あたり)
プラバスチンナトリウム 5mg
乳糖 64mg
リン酸水素カルシウム 15mg
カルボキシメチルセルロースカルシウム 5mg
ヒドロキシプロピルセルロース 2mg
ステアリン酸マグネシウム 1mg
計 92mg
プラバスチンナトリウム 5mg
乳糖 64mg
メタケイ酸アルミン酸マグネシウム 15mg
カルボキシメチルセルロースカルシウム 5mg
ヒドロキシプロピルセルロース 2mg
ステアリン酸マグネシウム 1mg
計 92mg
マンニトールをベースにし、表1の処方により直接打錠法によって1錠中プラバスタンNa5mgを含む錠剤を製造し、硬度、崩壊時間、溶出率を測定した。
プラバスタチンNa 5mg
マンニトール 75mg
微結晶セルロース 10mg
ステアリン酸Mg 1mg
合計 91mg
乳糖をベースにし、表3の処方により直接打錠法によって1錠中プラスバスタチンNa5mgを含む錠剤を製造し、実施例2と同様な測定を行った。
1.溶出試験法:JP13第2法
試験液:37℃の水900mL
回転数:50rpm
測定数:N=3
2.崩壊試験法:JP13
測定数:N=6
Claims (2)
- プラバスタチンナトリウム、マンニトールおよび滑沢剤よりなる混合物を、直接打錠法により打錠することによって得たことを特徴とする、貯蔵安定性にすぐれ、崩壊時間および溶出率にもすぐれたプラバスタチンナトリウム錠剤。
- さらに崩壊剤を含む混合物を打錠することによって得たことを特徴とする請求項1に記載のプラバスタチンナトリウム錠剤。
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2003303781A JP3719679B2 (ja) | 1998-12-07 | 2003-08-28 | プラバスタチンナトリウム錠 |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP36608398 | 1998-12-07 | ||
JP2003303781A JP3719679B2 (ja) | 1998-12-07 | 2003-08-28 | プラバスタチンナトリウム錠 |
Related Parent Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP11117389A Division JP2000229855A (ja) | 1998-12-07 | 1999-04-26 | プラバスタチンナトリウム錠 |
Publications (3)
Publication Number | Publication Date |
---|---|
JP2004002473A JP2004002473A (ja) | 2004-01-08 |
JP2004002473A5 JP2004002473A5 (ja) | 2005-08-25 |
JP3719679B2 true JP3719679B2 (ja) | 2005-11-24 |
Family
ID=30445584
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2003303781A Expired - Fee Related JP3719679B2 (ja) | 1998-12-07 | 2003-08-28 | プラバスタチンナトリウム錠 |
Country Status (1)
Country | Link |
---|---|
JP (1) | JP3719679B2 (ja) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2012002464A1 (ja) | 2010-06-30 | 2012-01-05 | 持田製薬株式会社 | ω3脂肪酸の配合製剤 |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2012056509A1 (ja) * | 2010-10-25 | 2012-05-03 | 興和株式会社 | 医薬組成物 |
JP4981194B2 (ja) * | 2010-10-25 | 2012-07-18 | 興和株式会社 | 医薬組成物 |
JP5988963B2 (ja) * | 2011-04-12 | 2016-09-07 | 沢井製薬株式会社 | ピタバスタチン含有製剤及びその製造方法 |
-
2003
- 2003-08-28 JP JP2003303781A patent/JP3719679B2/ja not_active Expired - Fee Related
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2012002464A1 (ja) | 2010-06-30 | 2012-01-05 | 持田製薬株式会社 | ω3脂肪酸の配合製剤 |
US8609138B2 (en) | 2010-06-30 | 2013-12-17 | Mochida Pharmaceutical Co., Ltd. | ω3 fatty acid compound preparation |
Also Published As
Publication number | Publication date |
---|---|
JP2004002473A (ja) | 2004-01-08 |
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