JP2025511122A5 - - Google Patents

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Publication number
JP2025511122A5
JP2025511122A5 JP2024557915A JP2024557915A JP2025511122A5 JP 2025511122 A5 JP2025511122 A5 JP 2025511122A5 JP 2024557915 A JP2024557915 A JP 2024557915A JP 2024557915 A JP2024557915 A JP 2024557915A JP 2025511122 A5 JP2025511122 A5 JP 2025511122A5
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JP
Japan
Prior art keywords
alkyl
substituted
cancer
optionally substituted
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024557915A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025511122A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/064984 external-priority patent/WO2023192817A1/en
Publication of JP2025511122A publication Critical patent/JP2025511122A/ja
Publication of JP2025511122A5 publication Critical patent/JP2025511122A5/ja
Pending legal-status Critical Current

Links

JP2024557915A 2022-03-28 2023-03-27 リジンアセチルトランスフェラーゼのmystファミリーの阻害剤 Pending JP2025511122A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202263324624P 2022-03-28 2022-03-28
US202263324619P 2022-03-28 2022-03-28
US63/324,624 2022-03-28
US63/324,619 2022-03-28
US202263476826P 2022-12-22 2022-12-22
US63/476,826 2022-12-22
PCT/US2023/064984 WO2023192817A1 (en) 2022-03-28 2023-03-27 Inhibitors of the myst family of lysine acetyl transferases

Publications (2)

Publication Number Publication Date
JP2025511122A JP2025511122A (ja) 2025-04-15
JP2025511122A5 true JP2025511122A5 (https=) 2026-04-06

Family

ID=86099757

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024557915A Pending JP2025511122A (ja) 2022-03-28 2023-03-27 リジンアセチルトランスフェラーゼのmystファミリーの阻害剤

Country Status (11)

Country Link
US (3) US12187732B2 (https=)
EP (1) EP4499609A1 (https=)
JP (1) JP2025511122A (https=)
KR (1) KR20250006833A (https=)
CN (1) CN119301096A (https=)
AU (1) AU2023241822A1 (https=)
CA (1) CA3255313A1 (https=)
IL (1) IL315930A (https=)
MX (1) MX2024011828A (https=)
TW (1) TW202400593A (https=)
WO (1) WO2023192817A1 (https=)

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CN118556053A (zh) 2021-11-16 2024-08-27 英矽智能科技知识产权有限公司 赖氨酸乙酰基转移酶6a(kat6a)抑制剂及其用途
KR20250006833A (ko) * 2022-03-28 2025-01-13 아이소스테릭스, 인코포레이티드 라이신 아세틸 전이효소의 myst 계열의 억제제
JP2026512835A (ja) * 2023-03-27 2026-04-21 ベイジン・コンランズ・ファーマシューティカル・カンパニー・リミテッド スルホンアミド化合物、その医薬組成物及び応用
AU2024325442A1 (en) * 2023-08-14 2026-03-26 Shanghai Henlius Biologics Co., Ltd. Sulfonamide compound, and preparation method therefor and use thereof
TW202530223A (zh) * 2023-09-27 2025-08-01 美商艾索司特瑞克斯公司 Myst抑制劑
WO2025098417A1 (zh) * 2023-11-08 2025-05-15 再和医药科技(苏州)有限公司 磺酰胺类化合物及其应用
WO2026053122A1 (en) * 2024-09-04 2026-03-12 Dana-Farber Cancer Institute, Inc. Methods of treating retinoid responsive cancers

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