JP2024529763A5 - - Google Patents

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Publication number
JP2024529763A5
JP2024529763A5 JP2024510406A JP2024510406A JP2024529763A5 JP 2024529763 A5 JP2024529763 A5 JP 2024529763A5 JP 2024510406 A JP2024510406 A JP 2024510406A JP 2024510406 A JP2024510406 A JP 2024510406A JP 2024529763 A5 JP2024529763 A5 JP 2024529763A5
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JP
Japan
Prior art keywords
pxrd
pattern
crystalline material
methyl
room temperature
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024510406A
Other languages
English (en)
Japanese (ja)
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JP2024529763A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/040884 external-priority patent/WO2023023322A1/en
Publication of JP2024529763A publication Critical patent/JP2024529763A/ja
Publication of JP2024529763A5 publication Critical patent/JP2024529763A5/ja
Pending legal-status Critical Current

Links

JP2024510406A 2021-08-20 2022-08-19 6-(シクロプロパンカルボキサミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキサミドの結晶体 Pending JP2024529763A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163235635P 2021-08-20 2021-08-20
US63/235,635 2021-08-20
PCT/US2022/040884 WO2023023322A1 (en) 2021-08-20 2022-08-19 Crystal forms of 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyl-d3)pyridazine-3-carboxamide

Publications (2)

Publication Number Publication Date
JP2024529763A JP2024529763A (ja) 2024-08-08
JP2024529763A5 true JP2024529763A5 (https=) 2025-08-26

Family

ID=83283223

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024510406A Pending JP2024529763A (ja) 2021-08-20 2022-08-19 6-(シクロプロパンカルボキサミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキサミドの結晶体

Country Status (7)

Country Link
US (1) US20240368130A1 (https=)
EP (1) EP4387968B1 (https=)
JP (1) JP2024529763A (https=)
KR (1) KR20240050380A (https=)
CN (1) CN118119614A (https=)
ES (1) ES3062193T3 (https=)
WO (1) WO2023023322A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2024241347A1 (en) * 2023-05-25 2024-11-28 Msn Laboratories Private Limited, R&D Center Novel polymorphs of 6-(cyclopropanecarbonylamido)-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-n-(trideuteriomethyl)pyridazine-3-carboxamide
ES3059443A1 (es) * 2024-09-17 2026-03-20 Moehs Iberica Sl Forma solida de 6-(ciclopropanocarboxamido)-4-((2-metoxi-3-(1-metil-1h-1,2,4-triazol-3-il)fenil)amino)piridazine-3-carboxilato de metilo o una sal del mismo, procedimiento para su preparacion y su uso en la sintesis de deucravacitinib

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3495358T (lt) * 2012-11-08 2022-05-25 Bristol-Myers Squibb Company Amidais pakeisti heterocikliniai junginiai, naudingi kaip il-12, il-23 ir (arba) ifn alfa atsako moduliatoriai
JP7113023B2 (ja) 2017-03-30 2022-08-04 ブリストル-マイヤーズ スクイブ カンパニー 6-(シクロプロパンアミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキシアミドの製造方法
KR102848769B1 (ko) 2018-05-31 2025-08-20 브리스톨-마이어스 스큅 컴퍼니 6-(시클로프로판카르복스아미도)-4-((2-메톡시-3-(1-메틸-1h-1,2,4-트리아졸-3-일)페닐)아미노)-n-(메틸-d3) 피리다진-3-카르복스아미드의 결정질 형태
US12570637B2 (en) 2019-06-12 2026-03-10 Bristol-Myers Squibb Company Crystalline salt forms 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyld3) pyridazine-3-carboxamide
KR20230137962A (ko) * 2021-01-29 2023-10-05 브리스톨-마이어스 스큅 컴퍼니 6-(시클로프로판카르복스아미도)-4-((2-메톡시-3-(1-메틸-1h-1,2,4-트리아졸-3-일)페닐)아미노)-n-(메틸-d3)피리다진-3-카르복스아미드의 결정 형태
CN117377667A (zh) * 2021-03-29 2024-01-09 百时美施贵宝公司 6-(环丙烷甲酰胺基)-4-((2-甲氧基-3-(1-甲基-1H-1,2,4-三唑-3-基)苯基)氨基)-N-(甲基-d3)哒嗪-3-甲酰胺的晶型

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