JP2023082086A5 - - Google Patents

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Publication number
JP2023082086A5
JP2023082086A5 JP2023052465A JP2023052465A JP2023082086A5 JP 2023082086 A5 JP2023082086 A5 JP 2023082086A5 JP 2023052465 A JP2023052465 A JP 2023052465A JP 2023052465 A JP2023052465 A JP 2023052465A JP 2023082086 A5 JP2023082086 A5 JP 2023082086A5
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Japan
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crystalline form
powder
ray diffraction
pharmaceutical composition
composition
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JP2023052465A
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English (en)
Japanese (ja)
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JP7763203B2 (ja
JP2023082086A (ja
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Priority claimed from JP2019538551A external-priority patent/JP7253491B2/ja
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JP2023052465A 2016-09-29 2023-03-28 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用 Active JP7763203B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CN201610866253 2016-09-29
CN201610866253.6 2016-09-29
JP2019538551A JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用
PCT/CN2017/104506 WO2018059556A1 (zh) 2016-09-29 2017-09-29 激酶抑制剂化合物的多晶型、含其的药物组合物及其制备方法和应用

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2019538551A Division JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用

Publications (3)

Publication Number Publication Date
JP2023082086A JP2023082086A (ja) 2023-06-13
JP2023082086A5 true JP2023082086A5 (https=) 2023-07-28
JP7763203B2 JP7763203B2 (ja) 2025-10-31

Family

ID=61763329

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2019538551A Active JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用
JP2023052465A Active JP7763203B2 (ja) 2016-09-29 2023-03-28 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2019538551A Active JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用

Country Status (17)

Country Link
US (3) US11053224B2 (https=)
EP (1) EP3502105B8 (https=)
JP (2) JP7253491B2 (https=)
KR (1) KR102289684B1 (https=)
CN (1) CN108884080B (https=)
AU (1) AU2017336889B2 (https=)
CA (2) CA3253105A1 (https=)
EA (1) EA201990688A1 (https=)
ES (1) ES2914294T3 (https=)
IL (2) IL265266B2 (https=)
MY (1) MY194364A (https=)
PH (1) PH12019500681A1 (https=)
PL (1) PL3502105T3 (https=)
SG (1) SG11201901962QA (https=)
TW (1) TWI647224B (https=)
WO (1) WO2018059556A1 (https=)
ZA (1) ZA201901717B (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2018059556A1 (zh) * 2016-09-29 2018-04-05 贝达药业股份有限公司 激酶抑制剂化合物的多晶型、含其的药物组合物及其制备方法和应用
KR102195348B1 (ko) 2018-11-15 2020-12-24 에이치케이이노엔 주식회사 단백질 키나제 억제제로서의 신규 화합물 및 이를 포함하는 약제학적 조성물
PT3884929T (pt) 2020-03-25 2023-08-09 Ocular Therapeutix Inc Implante ocular contendo um inibidor da tirosina cinase
AU2021340733A1 (en) 2020-09-14 2023-05-18 EyePoint Pharmaceuticals, Inc. Bioerodible ocular drug delivery insert and therapeutic method
CA3212253A1 (en) * 2021-03-16 2022-09-22 Young Ju Kim Crystalline form of heterocyclic compound as protein kinase inhibitor
JP7138982B1 (ja) 2021-09-24 2022-09-20 東海物産株式会社 アンセリンの結晶及びその製造方法
WO2023173093A1 (en) 2022-03-11 2023-09-14 EyePoint Pharmaceuticals, Inc. Continuous dosing regimen for treatment of a condition of the eye
CA3245207A1 (en) 2022-03-11 2023-09-14 EyePoint Pharmaceuticals, Inc. TREATMENT METHOD FOR MOISTURE-RELATED MACULAR DEGENERATION
KR20250002220A (ko) 2022-03-11 2025-01-07 아이포인트 파마슈티컬스, 인코포레이티드 안구 약물 전달 삽입물을 투여하여 연령 관련 황반 변성을 예방하는 방법
PE20260040A1 (es) 2023-04-11 2026-01-09 Ocular Therapeutix Inc Implante ocular que contiene un inhibidor de la tirosina cinasa
CN117143083B (zh) * 2023-08-30 2026-02-27 沈阳药科大学 VEGFR抑制剂Vorolanib的合成方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0213185A (pt) * 2001-10-10 2004-09-14 Sugen Inc Derivados de 3-[4-(heterociclila substituìda)-pirrol-2-ilmetilideno]2-indolinona como inibidores de cinase
ES2565683T3 (es) * 2006-09-15 2016-04-06 Xcovery, Inc. Compuestos inhibidores de quinasa
WO2008134909A1 (de) * 2007-05-07 2008-11-13 Baumer Electric Ag Akustischer wandler
US20100256392A1 (en) * 2007-11-21 2010-10-07 Teva Pharmaceutical Industries Ltd. Polymorphs of sunitinib base and processes for preparation thereof
WO2009128083A1 (en) * 2008-04-16 2009-10-22 Natco Pharma Limited Novel polymorphic forms of sunitinib base
RU2468022C2 (ru) * 2008-05-23 2012-11-27 Шанхай Инститьют Оф Фармасьютикал Индастри Производные дигидроиндолона
EP2186809A1 (en) * 2008-11-13 2010-05-19 LEK Pharmaceuticals D.D. New crystal form of sunitinib malate
EP2264027A1 (en) * 2009-05-27 2010-12-22 Ratiopharm GmbH Process for the preparation of N-[2-(Diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene) methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
CN106928114B (zh) * 2015-12-31 2020-07-28 韶远科技(上海)有限公司 含有脲基的环状手性氨基类化合物及其可放大工艺和用途
WO2018059556A1 (zh) * 2016-09-29 2018-04-05 贝达药业股份有限公司 激酶抑制剂化合物的多晶型、含其的药物组合物及其制备方法和应用

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