JP2024505063A5 - - Google Patents

Info

Publication number
JP2024505063A5
JP2024505063A5 JP2023545957A JP2023545957A JP2024505063A5 JP 2024505063 A5 JP2024505063 A5 JP 2024505063A5 JP 2023545957 A JP2023545957 A JP 2023545957A JP 2023545957 A JP2023545957 A JP 2023545957A JP 2024505063 A5 JP2024505063 A5 JP 2024505063A5
Authority
JP
Japan
Prior art keywords
methyl
crystalline
measured
ray diffraction
pattern
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023545957A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024505063A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/014261 external-priority patent/WO2022165141A1/en
Publication of JP2024505063A publication Critical patent/JP2024505063A/ja
Publication of JP2024505063A5 publication Critical patent/JP2024505063A5/ja
Pending legal-status Critical Current

Links

JP2023545957A 2021-01-29 2022-01-28 6-(シクロプロパンカルボキサミド)-4-((2-メトキシ-3-(1-メチル-1H-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-N-(メチル-d3)ピリダジン-3-カルボキサミドの結晶形態 Pending JP2024505063A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163143769P 2021-01-29 2021-01-29
US63/143,769 2021-01-29
PCT/US2022/014261 WO2022165141A1 (en) 2021-01-29 2022-01-28 Crystal form of 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyl-d3)pyridazine-3-carboxamide

Publications (2)

Publication Number Publication Date
JP2024505063A JP2024505063A (ja) 2024-02-02
JP2024505063A5 true JP2024505063A5 (https=) 2025-01-30

Family

ID=80447586

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023545957A Pending JP2024505063A (ja) 2021-01-29 2022-01-28 6-(シクロプロパンカルボキサミド)-4-((2-メトキシ-3-(1-メチル-1H-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-N-(メチル-d3)ピリダジン-3-カルボキサミドの結晶形態

Country Status (11)

Country Link
US (2) US12129245B2 (https=)
EP (1) EP4284796B1 (https=)
JP (1) JP2024505063A (https=)
KR (1) KR20230137962A (https=)
CN (1) CN116829549A (https=)
AU (1) AU2022214313A1 (https=)
CA (1) CA3206254A1 (https=)
ES (1) ES3026120T3 (https=)
IL (1) IL304597A (https=)
MX (1) MX2023008651A (https=)
WO (1) WO2022165141A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7113023B2 (ja) * 2017-03-30 2022-08-04 ブリストル-マイヤーズ スクイブ カンパニー 6-(シクロプロパンアミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキシアミドの製造方法
EP4387968B1 (en) * 2021-08-20 2025-11-12 Bristol-Myers Squibb Company Crystal forms of 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyl-d3)pyridazine-3-carboxamide
EP4423086A1 (en) 2021-10-25 2024-09-04 Kymera Therapeutics, Inc. Tyk2 degraders and uses thereof
CN116574056A (zh) * 2023-04-10 2023-08-11 五邑大学 一种氟代异喹啉酮类化合物的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3495358T (lt) * 2012-11-08 2022-05-25 Bristol-Myers Squibb Company Amidais pakeisti heterocikliniai junginiai, naudingi kaip il-12, il-23 ir (arba) ifn alfa atsako moduliatoriai
JP7113023B2 (ja) * 2017-03-30 2022-08-04 ブリストル-マイヤーズ スクイブ カンパニー 6-(シクロプロパンアミド)-4-((2-メトキシ-3-(1-メチル-1h-1,2,4-トリアゾール-3-イル)フェニル)アミノ)-n-(メチル-d3)ピリダジン-3-カルボキシアミドの製造方法
KR102848769B1 (ko) * 2018-05-31 2025-08-20 브리스톨-마이어스 스큅 컴퍼니 6-(시클로프로판카르복스아미도)-4-((2-메톡시-3-(1-메틸-1h-1,2,4-트리아졸-3-일)페닐)아미노)-n-(메틸-d3) 피리다진-3-카르복스아미드의 결정질 형태
US12570637B2 (en) * 2019-06-12 2026-03-10 Bristol-Myers Squibb Company Crystalline salt forms 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyld3) pyridazine-3-carboxamide

Similar Documents

Publication Publication Date Title
JP2024505063A5 (https=)
JP6966590B2 (ja) オメカムチブメカルビルの塩及び塩を調製するプロセス
JP4624667B2 (ja) 1−4−(5−シアノインドール−3−イル)ブチル−4−(2−カルバモイルベンゾフラン−5−イル)ピペラジン塩酸塩の多形相
JP2024514090A5 (https=)
JP2023036708A5 (https=)
JP2012527442A5 (https=)
JP2022551316A5 (https=)
JP3665053B2 (ja) 純結晶形態の5−クロロ−3−(4−メタンスルホニルフェニル)−6’−メチル−[2,3’]ビピリジニルおよび合成方法
JP2024521412A5 (https=)
ZA200106371B (en) 3-Phenylpyridine derivatives and their use as NK-1 receptor antagonist.
JP2024540922A5 (https=)
TW202200594A (zh) 一種glp-1受體激動劑的晶型a及其製備方法
CA2505361A1 (en) Phenyl or heteroaryl amino alkane derivatives as ip receptor antagonist
JP2015516968A5 (https=)
JP2022533340A5 (https=)
JP2009521414A5 (https=)
AU2001264804A1 (en) 5-chloro-3-(4-methanesulfonylphenyl)-6'-methyl- [2,3']bipyridinyl in pure crystalline form and process for synthesis
JP2024547113A5 (https=)
JP2024529763A5 (https=)
CN115819257A (zh) 维兰特罗三苯乙酸盐的新结晶形式及其制备方法
JP2018522945A5 (https=)
KR20180036722A (ko) 빌라스틴의 결정형 및 그의 제조 방법
CN111793074B (zh) K-5a2化合物的晶型及其制备方法和应用
JP2023521411A5 (https=)
JP2025508792A5 (https=)