JP2024540922A5 - - Google Patents

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Publication number
JP2024540922A5
JP2024540922A5 JP2024523525A JP2024523525A JP2024540922A5 JP 2024540922 A5 JP2024540922 A5 JP 2024540922A5 JP 2024523525 A JP2024523525 A JP 2024523525A JP 2024523525 A JP2024523525 A JP 2024523525A JP 2024540922 A5 JP2024540922 A5 JP 2024540922A5
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JP
Japan
Application number
JP2024523525A
Other languages
Japanese (ja)
Other versions
JPWO2023066941A5 (https=
JP2024540922A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/078989 external-priority patent/WO2023066941A1/en
Publication of JP2024540922A publication Critical patent/JP2024540922A/ja
Publication of JPWO2023066941A5 publication Critical patent/JPWO2023066941A5/ja
Publication of JP2024540922A5 publication Critical patent/JP2024540922A5/ja
Pending legal-status Critical Current

Links

JP2024523525A 2021-10-18 2022-10-18 N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素のエタノール溶媒和物の結晶形 Pending JP2024540922A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163257073P 2021-10-18 2021-10-18
US63/257,073 2021-10-18
PCT/EP2022/078989 WO2023066941A1 (en) 2021-10-18 2022-10-18 Crystalline form of an ethanol solvate of n-(4-(1-(2,6-difluorobenzyl)-5-((dimethylamino)methyl)-3-(6-methoxy-3-pyridazinyl)-2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-n'-methoxyurea

Publications (3)

Publication Number Publication Date
JP2024540922A JP2024540922A (ja) 2024-11-06
JPWO2023066941A5 JPWO2023066941A5 (https=) 2025-10-27
JP2024540922A5 true JP2024540922A5 (https=) 2025-10-27

Family

ID=84359608

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024523525A Pending JP2024540922A (ja) 2021-10-18 2022-10-18 N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素のエタノール溶媒和物の結晶形

Country Status (5)

Country Link
US (1) US20250066382A1 (https=)
EP (1) EP4419530A1 (https=)
JP (1) JP2024540922A (https=)
CN (1) CN118451082A (https=)
WO (1) WO2023066941A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2912929T5 (en) 2016-09-30 2025-05-09 Sumitomo Pharma Switzerland Gmbh Methods of treating uterine fibroids and endometriosis
JP2022551316A (ja) 2019-10-10 2022-12-08 ミオバント サイエンシズ ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形
CA3185151A1 (en) 2020-05-29 2021-12-02 Myovant Sciences Gmbh Combination solid oral dosage forms of gonadotropin-releasing hormone antagonists

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7300935B2 (en) 2003-01-29 2007-11-27 Takeda Pharmaceutical Company Thienopyrimidine compounds and use thereof
AR092707A1 (es) 2012-09-28 2015-04-29 Takeda Pharmaceuticals Co Metodo de produccion de derivado de tienopirimidina
TWI744224B (zh) 2015-02-26 2021-11-01 日商武田藥品工業股份有限公司 固形製劑
ES2912929T5 (en) 2016-09-30 2025-05-09 Sumitomo Pharma Switzerland Gmbh Methods of treating uterine fibroids and endometriosis
MA46361A (fr) 2016-09-30 2021-03-31 Myovant Sciences Gmbh Traitement du cancer de la prostate
US11306104B2 (en) * 2018-03-14 2022-04-19 Teva Pharmaceuticals International Gmbh Solid state forms of Relugolix
WO2021069700A1 (en) 2019-10-10 2021-04-15 Myovant Sciences Gmbh Crystalline solvated forms of n-(4-(1-(2,6-difluorobenzyl)-5- ((dimethylamino)methyl)-3-(6-methoxy-3-pyridazinyl)-2,4-dioxo-1,2,3,4- tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-n'-methoxyurea
JP2022551316A (ja) 2019-10-10 2022-12-08 ミオバント サイエンシズ ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形

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