JP2022551316A5 - - Google Patents

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Publication number
JP2022551316A5
JP2022551316A5 JP2022521569A JP2022521569A JP2022551316A5 JP 2022551316 A5 JP2022551316 A5 JP 2022551316A5 JP 2022521569 A JP2022521569 A JP 2022521569A JP 2022521569 A JP2022521569 A JP 2022521569A JP 2022551316 A5 JP2022551316 A5 JP 2022551316A5
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JP
Japan
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JP2022521569A
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Japanese (ja)
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JP2022551316A (ja
JPWO2021069711A5 (https=
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Publication date
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Priority claimed from PCT/EP2020/078493 external-priority patent/WO2021069711A1/en
Publication of JP2022551316A publication Critical patent/JP2022551316A/ja
Publication of JP2022551316A5 publication Critical patent/JP2022551316A5/ja
Publication of JPWO2021069711A5 publication Critical patent/JPWO2021069711A5/ja
Pending legal-status Critical Current

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JP2022521569A 2019-10-10 2020-10-09 N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形 Pending JP2022551316A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962913560P 2019-10-10 2019-10-10
US62/913,560 2019-10-10
PCT/EP2020/078493 WO2021069711A1 (en) 2019-10-10 2020-10-09 Crystalline forms of n-(4-(1-(2,6-difluorobenzyl)-5- ((dimethylamino)methyl)-3-(6-methoxy-3-pyridazinyl)-2,4-dioxo- 1,2,3,4-tetrahydrothieno[2,3-d]pyrimidin-6-yl)phenyl)-n'- methoxyurea

Publications (3)

Publication Number Publication Date
JP2022551316A JP2022551316A (ja) 2022-12-08
JP2022551316A5 true JP2022551316A5 (https=) 2023-10-17
JPWO2021069711A5 JPWO2021069711A5 (https=) 2023-10-17

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ID=72852650

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JP2022521569A Pending JP2022551316A (ja) 2019-10-10 2020-10-09 N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形

Country Status (5)

Country Link
US (2) US12338249B2 (https=)
EP (1) EP4041739A1 (https=)
JP (1) JP2022551316A (https=)
CN (1) CN115279769A (https=)
WO (1) WO2021069711A1 (https=)

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JP2024540922A (ja) 2021-10-18 2024-11-06 スミトモ ファーマ スウィッツァーランド ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素のエタノール溶媒和物の結晶形

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JP2022551316A (ja) 2019-10-10 2022-12-08 ミオバント サイエンシズ ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形
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JP2024540922A (ja) 2021-10-18 2024-11-06 スミトモ ファーマ スウィッツァーランド ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素のエタノール溶媒和物の結晶形
WO2023119333A1 (en) 2021-12-25 2023-06-29 Dr. Reddy’S Laboratories Limited Process for preparation of relugolix and its intermediates
IN202221021078A (https=) 2022-04-08 2023-10-13
CN115417883B (zh) 2022-09-16 2024-08-27 浙江科聚生物医药有限公司 一种瑞卢戈利的晶型及其制备方法

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