MA46361A - Traitement du cancer de la prostate - Google Patents

Traitement du cancer de la prostate

Info

Publication number
MA46361A
MA46361A MA046361A MA46361A MA46361A MA 46361 A MA46361 A MA 46361A MA 046361 A MA046361 A MA 046361A MA 46361 A MA46361 A MA 46361A MA 46361 A MA46361 A MA 46361A
Authority
MA
Morocco
Prior art keywords
treatment
prostate cancer
prostate
cancer
Prior art date
Application number
MA046361A
Other languages
English (en)
Inventor
Brendan Mark Johnson
David B Maclean
Paul N Mudd Jr
Vijaykumar Reddy Rajasekhar
Lynn Seely
Original Assignee
Myovant Sciences Gmbh
Takeda Pharmaceuticals Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Myovant Sciences Gmbh, Takeda Pharmaceuticals Co filed Critical Myovant Sciences Gmbh
Publication of MA46361A publication Critical patent/MA46361A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • A61K31/501Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41661,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA046361A 2016-09-30 2017-09-29 Traitement du cancer de la prostate MA46361A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662402004P 2016-09-30 2016-09-30
US201662402150P 2016-09-30 2016-09-30

Publications (1)

Publication Number Publication Date
MA46361A true MA46361A (fr) 2021-03-31

Family

ID=60915459

Family Applications (1)

Application Number Title Priority Date Filing Date
MA046361A MA46361A (fr) 2016-09-30 2017-09-29 Traitement du cancer de la prostate

Country Status (12)

Country Link
US (4) US10449191B2 (fr)
EP (1) EP3518932A2 (fr)
JP (1) JP7062673B2 (fr)
CN (1) CN110248661A (fr)
AU (2) AU2017334035B2 (fr)
BR (1) BR112019006228A2 (fr)
CA (1) CA3038875A1 (fr)
IL (3) IL308528A (fr)
MA (1) MA46361A (fr)
MX (2) MX2019003733A (fr)
NZ (1) NZ752918A (fr)
WO (1) WO2018060463A2 (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2912929T3 (es) 2016-09-30 2022-05-30 Myovant Sciences Gmbh Métodos de tratamiento de fibromas uterinos y endometriosis
AU2017334035B2 (en) * 2016-09-30 2022-11-24 Sumitomo Pharma Switzerland Gmbh Treatment of prostate cancer
CN110194776B (zh) * 2019-06-27 2021-05-28 四川伊诺达博医药科技有限公司 一种瑞卢戈利的合成方法
JP2022551316A (ja) * 2019-10-10 2022-12-08 ミオバント サイエンシズ ゲーエムベーハー N-(4-(1-(2,6-ジフルオロベンジル)-5-((ジメチルアミノ)メチル)-3-(6-メトキシ-3-ピリダジニル)-2,4-ジオキソ-1,2,3,4-テトラヒドロチエノ[2,3-d]ピリミジン-6-イル)フェニル)-N’-メトキシ尿素の結晶形
WO2021069700A1 (fr) * 2019-10-10 2021-04-15 Myovant Sciences Gmbh Formes cristallines solvatées de n-(4-(1-(2,6-difluorobenzyle)-5- ((diméthylamino)méthyle)-3-(6-méthoxy-3-pyridazinyle)-2,4-dioxo -1,2,3,4-tétrahydrothiéno[2,3-d]pyrimidine-6-yl) phényle)-n'-méthoxyurée
MX2022015003A (es) 2020-05-29 2023-03-03 Myovant Sciences Gmbh Formas de dosificacion oral solidas de combinacion de antagonistas de la hormona liberadora de gonadotropina.
EP4232164A1 (fr) * 2020-10-20 2023-08-30 Baylor College of Medicine Marqueurs métaboliques multiplexes dans le plasma pour la détection précoce du cancer de la prostate chez les afro-américains
EP4243829A1 (fr) 2020-11-11 2023-09-20 Myovant Sciences GmbH Méthodes d'administration du rélugolix
WO2023066941A1 (fr) 2021-10-18 2023-04-27 Myovant Sciences Gmbh Forme cristalline d'un solvate d'éthanol de n-(4-(1-(2,6-difluorobenzyle)-5-((diméthylamino)méthyle)-3-(6-méthoxy-3-pyridazinyl)-2,4-dioxo-1,2,3,4-tétrahydrothiéno[2,3-d]pyrimidin-6-yl)phényle)-n'-méthoxyurée
WO2023152611A1 (fr) * 2022-02-11 2023-08-17 Aragon Pharmaceuticals, Inc. Apalutamide et relugolix pour le traitement du cancer de la prostate

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2233284C2 (ru) 1999-03-24 2004-07-27 Такеда Кемикал Индастриз, Лтд. Тиенопиримидиновые производные, способ их получения, фармацевтическая композиция и способ антагонизации гонадотропин-рилизинг гормона
TWI225863B (en) 1999-03-24 2005-01-01 Takeda Chemical Industries Ltd Thienopyrimidine compounds, their production and use
US6849738B2 (en) 2000-02-29 2005-02-01 Takeda Chemical Industries, Ltd. Processes for the production of thienopyrimidine derivatives
US7569570B2 (en) 2002-01-30 2009-08-04 Takeda Pharmaceutical Company Limited Thienopyrimidines, process for preparing the same and use thereof
NZ541772A (en) 2003-01-29 2009-10-30 Takeda Pharmaceutical Thienopyrimidine compounds and use thereof
MXPA06000297A (es) 2003-07-07 2006-03-28 Neurocrine Biosciences Inc Derivados de pirimidina-2,4-diona como antagonistas del receptor de la hormona de liberacion de gonadotropina.
BRPI0613643A2 (pt) 2005-07-22 2012-11-06 Takeda Pharmaceutical inibidor de ovulação prematura, método de inibir ovulação prematura e uso de um composto
PE20090044A1 (es) 2007-04-06 2009-01-23 Neurocrine Biosciences Inc Antagonistas del receptor de la hormona liberadora de gonadotropina y procedimientos relacionados con los mismos
WO2009062087A1 (fr) 2007-11-07 2009-05-14 Neurocrine Biosciences, Inc. Procédés de préparation de dérivés d'uracile
EP2329823A4 (fr) 2008-09-03 2013-04-03 Takeda Pharmaceutical Procédé pour améliorer la capacité d'une préparation à être absorbée et préparation dont la capacité à être absorbée est améliorée
PL2900675T3 (pl) 2012-09-28 2019-08-30 Takeda Pharmaceutical Company Limited Sposób wytwarzania pochodnej tienopirymidyny
CN107249590A (zh) 2015-02-26 2017-10-13 武田药品工业株式会社 固体制剂
US20180044977A1 (en) 2016-08-12 2018-02-15 Raynor Mfg. Co. Rolling door construction for controlling air leakage
AU2017334035B2 (en) 2016-09-30 2022-11-24 Sumitomo Pharma Switzerland Gmbh Treatment of prostate cancer
ES2912929T3 (es) 2016-09-30 2022-05-30 Myovant Sciences Gmbh Métodos de tratamiento de fibromas uterinos y endometriosis

Also Published As

Publication number Publication date
IL265697A (en) 2019-05-30
EP3518932A2 (fr) 2019-08-07
US20190224196A1 (en) 2019-07-25
JP7062673B2 (ja) 2022-05-06
CA3038875A1 (fr) 2018-04-05
US20220401443A1 (en) 2022-12-22
WO2018060463A2 (fr) 2018-04-05
WO2018060463A3 (fr) 2018-05-11
US10449191B2 (en) 2019-10-22
MX2019003733A (es) 2019-09-26
MX2023001468A (es) 2023-03-03
CN110248661A (zh) 2019-09-17
AU2023201047A1 (en) 2023-03-23
JP2019529574A (ja) 2019-10-17
US11583526B2 (en) 2023-02-21
IL300071A (en) 2023-03-01
US10786501B2 (en) 2020-09-29
BR112019006228A2 (pt) 2019-06-18
US20210205303A1 (en) 2021-07-08
IL265697B2 (en) 2023-07-01
AU2017334035A1 (en) 2019-05-16
IL265697B1 (en) 2023-03-01
AU2017334035B2 (en) 2022-11-24
NZ752918A (en) 2022-09-30
IL308528A (en) 2024-01-01
US20200129507A1 (en) 2020-04-30

Similar Documents

Publication Publication Date Title
MA46361A (fr) Traitement du cancer de la prostate
MA49144A (fr) Polythérapies pour le traitement du cancer
MA43374A (fr) Méthodes de traitement de tumeurs malignes
HK1258098A1 (zh) 治療癌症的方法
MA50056A (fr) Procédés de traitement de tumeur
MA47501A (fr) Dérivé de di-nucléotides cycliques pour le traitement du cancer
MA43135A (fr) Compositions et méthodes pour le du traitement du cancer
MA43190A (fr) Traitement de la dyslipidémie mixte
MA41449A (fr) Polythérapies pour le traitement de cancers
MA48637A (fr) Polythérapies pour le traitement du cancer
MA47408A (fr) Traitement du cancer
MA50409A (fr) Polythérapies pour le traitement du cancer
DK3458052T3 (da) Kombinationsbehandling af cancer
MA45780A (fr) Méthodes de traitement du cancer de la prostate
MA44612A (fr) Méthodes de traitement de cancers pédiatriques
MA45675A (fr) Méthodes et compositions permettant le traitement du cancer
IL262342A (en) Cancer treatment methods
MA49059A (fr) Traitement des cancers positifs à her2
MA52627A (fr) Traitement du cancer
MA42930A (fr) Traitement de maladies neurodégénératives
DK3525774T3 (da) Lasofoxifen behandling af er+ brystcancer
IL263835A (en) Exosome-guided treatment of cancer
DK3576740T3 (da) Cancerbehandling
MA42444A (fr) Traitement du prurit
DK3407909T3 (da) Cancerbehandling