JP2024511832A5 - - Google Patents
Info
- Publication number
- JP2024511832A5 JP2024511832A5 JP2023560282A JP2023560282A JP2024511832A5 JP 2024511832 A5 JP2024511832 A5 JP 2024511832A5 JP 2023560282 A JP2023560282 A JP 2023560282A JP 2023560282 A JP2023560282 A JP 2023560282A JP 2024511832 A5 JP2024511832 A5 JP 2024511832A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- membered
- deuterium
- independently selected
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (17)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2021/083783 | 2021-03-30 | ||
| CN2021083783 | 2021-03-30 | ||
| CNPCT/CN2021/090945 | 2021-04-29 | ||
| CN2021090945 | 2021-04-29 | ||
| CN2021111479 | 2021-08-09 | ||
| CNPCT/CN2021/111479 | 2021-08-09 | ||
| CN2021128942 | 2021-11-05 | ||
| CNPCT/CN2021/128942 | 2021-11-05 | ||
| CNPCT/CN2021/130097 | 2021-11-11 | ||
| CN2021130097 | 2021-11-11 | ||
| CNPCT/CN2021/138806 | 2021-12-16 | ||
| CN2021138806 | 2021-12-16 | ||
| CN2021143043 | 2021-12-30 | ||
| CNPCT/CN2021/143043 | 2021-12-30 | ||
| CNPCT/CN2022/071548 | 2022-01-12 | ||
| CN2022071548 | 2022-01-12 | ||
| PCT/CN2022/083557 WO2022206725A1 (en) | 2021-03-30 | 2022-03-29 | Novel compounds useful as sting agonists and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024511832A JP2024511832A (ja) | 2024-03-15 |
| JP2024511832A5 true JP2024511832A5 (https=) | 2025-04-07 |
Family
ID=83457956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023560282A Pending JP2024511832A (ja) | 2021-03-30 | 2022-03-29 | Stingアゴニストとして有用な新規化合物およびその使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20240116909A1 (https=) |
| EP (1) | EP4313962A4 (https=) |
| JP (1) | JP2024511832A (https=) |
| CN (1) | CN117203194A (https=) |
| AR (1) | AR125608A1 (https=) |
| TW (1) | TW202302579A (https=) |
| UY (1) | UY39705A (https=) |
| WO (1) | WO2022206725A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN118524854A (zh) * | 2021-12-17 | 2024-08-20 | 北京加科思新药研发有限公司 | 包含可用作sting激动剂的新型化合物的化合物-连接基构建体及其用途 |
| WO2024032782A1 (en) * | 2022-08-12 | 2024-02-15 | Jacobio Pharmaceuticals Co.Ltd. | Vaccine adjuvants and uses thereof |
| WO2026001915A1 (en) * | 2024-06-24 | 2026-01-02 | Jacobio Pharmaceuticals Co., Ltd. | Drug linker, conjugate thereof, and uses thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3774765A4 (en) * | 2018-04-03 | 2021-12-29 | Merck Sharp & Dohme Corp. | Aza-benzothiophene compounds as sting agonists |
| JP7326319B2 (ja) * | 2018-04-03 | 2023-08-15 | メルク・シャープ・アンド・ドーム・エルエルシー | Stingアゴニストとしてのベンゾチオフェン類及び関連する化合物 |
| CR20220029A (es) * | 2019-07-22 | 2022-03-14 | Lupin Ltd | Compuestos macrocíclicos como agonistas de sting y métodos y usos de los mismos |
-
2022
- 2022-03-29 WO PCT/CN2022/083557 patent/WO2022206725A1/en not_active Ceased
- 2022-03-29 AR ARP220100748A patent/AR125608A1/es not_active Application Discontinuation
- 2022-03-29 EP EP22778907.0A patent/EP4313962A4/en active Pending
- 2022-03-29 JP JP2023560282A patent/JP2024511832A/ja active Pending
- 2022-03-29 CN CN202280023908.7A patent/CN117203194A/zh active Pending
- 2022-03-29 TW TW111112050A patent/TW202302579A/zh unknown
- 2022-03-29 US US18/284,897 patent/US20240116909A1/en active Pending
- 2022-03-29 UY UY0001039705A patent/UY39705A/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2024511832A5 (https=) | ||
| CN114174303B (zh) | 作为sting激动剂的大环化合物及其方法和用途 | |
| JP2021534124A5 (https=) | ||
| JP2022515197A5 (https=) | ||
| JP2014505660A5 (https=) | ||
| JP2024512154A5 (https=) | ||
| RU2014114973A (ru) | Пиразол-4-ил-гетероциклил-карбоксамидные соединения и способы применения | |
| EA031030B1 (ru) | Ингибиторы фактора в комплемента на основе производных пиперидинилиндола и их применение | |
| JP2006528700A5 (https=) | ||
| JP2013510883A5 (https=) | ||
| JP2022505645A5 (https=) | ||
| RU2014122340A (ru) | Ингибиторы вируса гепатита с, имеющие жесткую вытянутую цепь и содержащие фрагмент {2-[4-(бифенил-4-ил)-1н-имидазо-2-ил]пирролидин-1-карбонилметил}амина | |
| RU2014153800A (ru) | Соединения 5-азаиндазола и способы их применения | |
| JP2014528467A5 (https=) | ||
| RU2012117398A (ru) | Бензоксазепиновые ингибиторы pi3 и способы применения | |
| JP2016509047A5 (https=) | ||
| RU2009148320A (ru) | Производные пиперидина/пиперазина | |
| JP2015501833A5 (https=) | ||
| JP2013520473A5 (https=) | ||
| JP2024546951A5 (https=) | ||
| JP2014532716A5 (https=) | ||
| RU2010101611A (ru) | Полициклические производные гуанина и способы их применения | |
| JP2017519754A5 (https=) | ||
| JP2004517843A5 (https=) | ||
| JP2024517861A5 (https=) |