JP2023548657A5 - - Google Patents

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Publication number
JP2023548657A5
JP2023548657A5 JP2023521702A JP2023521702A JP2023548657A5 JP 2023548657 A5 JP2023548657 A5 JP 2023548657A5 JP 2023521702 A JP2023521702 A JP 2023521702A JP 2023521702 A JP2023521702 A JP 2023521702A JP 2023548657 A5 JP2023548657 A5 JP 2023548657A5
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JP
Japan
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JP2023521702A
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Japanese (ja)
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JPWO2022076831A5 (https=
JP2023548657A (ja
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Publication date
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Priority claimed from PCT/US2021/054191 external-priority patent/WO2022076831A2/en
Publication of JP2023548657A publication Critical patent/JP2023548657A/ja
Publication of JPWO2022076831A5 publication Critical patent/JPWO2022076831A5/ja
Publication of JP2023548657A5 publication Critical patent/JP2023548657A5/ja
Pending legal-status Critical Current

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JP2023521702A 2020-10-09 2021-10-08 がんの処置に使用するための、egfrおよび/またはher2のヘテロ環阻害剤 Pending JP2023548657A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202063089965P 2020-10-09 2020-10-09
US63/089,965 2020-10-09
US202163151468P 2021-02-19 2021-02-19
US63/151,468 2021-02-19
PCT/US2021/054191 WO2022076831A2 (en) 2020-10-09 2021-10-08 Methods for treating cancer

Publications (3)

Publication Number Publication Date
JP2023548657A JP2023548657A (ja) 2023-11-20
JPWO2022076831A5 JPWO2022076831A5 (https=) 2024-10-15
JP2023548657A5 true JP2023548657A5 (https=) 2024-10-15

Family

ID=78516928

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023521702A Pending JP2023548657A (ja) 2020-10-09 2021-10-08 がんの処置に使用するための、egfrおよび/またはher2のヘテロ環阻害剤

Country Status (13)

Country Link
US (1) US20240101576A1 (https=)
EP (1) EP4225445A2 (https=)
JP (1) JP2023548657A (https=)
KR (1) KR20230107419A (https=)
AU (1) AU2021358596A1 (https=)
BR (1) BR112023006531A2 (https=)
CA (1) CA3198202A1 (https=)
CL (2) CL2023001012A1 (https=)
IL (1) IL301929A (https=)
MX (1) MX2023004085A (https=)
PH (1) PH12023500010A1 (https=)
TW (1) TW202227063A (https=)
WO (1) WO2022076831A2 (https=)

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GB201905721D0 (en) 2019-04-24 2019-06-05 Univ Dundee Compounds
EP4323356A1 (en) 2021-04-13 2024-02-21 Nuvalent, Inc. Amino-substituted heterocycles for treating cancers with egfr mutations
IL321504A (en) * 2022-12-23 2025-08-01 Tay Therapeutics Ltd Selective beta inhibitors and their uses
CN115819418B (zh) * 2023-02-14 2023-04-28 山东绿叶制药有限公司 Plk1激酶抑制剂及其制备方法和应用
CN121909190A (zh) * 2023-06-08 2026-04-21 安塔列斯疗法股份有限公司 1,5-二氢-4H-吡咯并[3,2-c]吡啶-4-酮用于癌症治疗
CN121712773A (zh) 2023-06-08 2026-03-20 安塔列斯疗法股份有限公司 1,5-二氢-4h-吡咯并[3,2-c]吡啶-4-酮用于癌症治疗
CN119528906A (zh) * 2023-08-30 2025-02-28 中国科学院上海药物研究所 氮杂螺环类化合物及其制备方法、药物组合物和应用
EP4534085A1 (en) * 2023-10-03 2025-04-09 Scorpion Therapeutics, Inc. Compounds for use in methods of treating cancer
WO2025251058A1 (en) * 2024-05-31 2025-12-04 Celyn Therapeutics, Inc. Egfr inhibitors in cancer treatment

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US7964729B2 (en) 2006-08-28 2011-06-21 Massachusetts Institute Of Technology Sox-based kinase sensor
ES2570756T3 (es) * 2009-06-15 2016-05-20 Nerviano Medical Sciences Srl Derivados pirimidinilpirrolopiridinona sustituidos, proceso para su preparación y su uso como inhibidores de cinasa
JP5825932B2 (ja) 2011-08-26 2015-12-02 キヤノン株式会社 撮像装置及びその制御方法、プログラム、及び記録媒体
WO2013092512A1 (en) 2011-12-21 2013-06-27 Bayer Intellectual Property Gmbh Substituted benzylpyrazoles
WO2013167698A1 (en) 2012-05-11 2013-11-14 Bayer Pharma Aktiengesellschaft Substituted cycloalkenopyrazoles as bub1 inhibitors for the treatment of cancer
EP2976335A1 (en) 2013-03-21 2016-01-27 Bayer Pharma Aktiengesellschaft Heteroaryl substituted indazoles
EP2976336A1 (en) 2013-03-21 2016-01-27 Bayer Pharma Aktiengesellschaft 3-heteroaryl substituted indazoles
CN105452237A (zh) 2013-06-21 2016-03-30 拜耳制药股份公司 杂芳基取代的吡唑
JP2016525076A (ja) 2013-06-21 2016-08-22 バイエル ファーマ アクチエンゲゼルシャフト 置換されたベンジルピラゾール類
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JP2016526540A (ja) 2013-06-21 2016-09-05 バイエル ファーマ アクチエンゲゼルシャフト 置換ベンジルピラゾール
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EP3143015B1 (en) 2014-05-13 2019-02-20 ARIAD Pharmaceuticals, Inc. Heteroaryl compounds for kinase inhibition
AR100886A1 (es) 2014-06-17 2016-11-09 Bayer Pharma AG 3-amino-1,5,6,7-tetrahidro-4h-indol-4-onas
AU2016212230B2 (en) * 2015-01-28 2019-09-19 Bayer Pharma Aktiengesellschaft 4H-pyrrolo[3,2-c]pyridin-4-one derivatives
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CA3091834A1 (en) 2018-02-23 2019-08-29 The Regents Of The University Of Michigan Egfr dimer disruptors and use of the same
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