JP2023533037A5 - - Google Patents

Info

Publication number
JP2023533037A5
JP2023533037A5 JP2023501220A JP2023501220A JP2023533037A5 JP 2023533037 A5 JP2023533037 A5 JP 2023533037A5 JP 2023501220 A JP2023501220 A JP 2023501220A JP 2023501220 A JP2023501220 A JP 2023501220A JP 2023533037 A5 JP2023533037 A5 JP 2023533037A5
Authority
JP
Japan
Prior art keywords
substituted
alkyl
hydrogen
halo
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023501220A
Other languages
English (en)
Japanese (ja)
Other versions
JP7771157B2 (ja
JP2023533037A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/040798 external-priority patent/WO2022011084A1/en
Publication of JP2023533037A publication Critical patent/JP2023533037A/ja
Publication of JP2023533037A5 publication Critical patent/JP2023533037A5/ja
Application granted granted Critical
Publication of JP7771157B2 publication Critical patent/JP7771157B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023501220A 2020-07-09 2021-07-08 オキソピロリジン fpr2アゴニスト Active JP7771157B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063049838P 2020-07-09 2020-07-09
US63/049,838 2020-07-09
PCT/US2021/040798 WO2022011084A1 (en) 2020-07-09 2021-07-08 Oxopyrrolidine fpr2 agonists

Publications (3)

Publication Number Publication Date
JP2023533037A JP2023533037A (ja) 2023-08-01
JP2023533037A5 true JP2023533037A5 (https=) 2024-07-12
JP7771157B2 JP7771157B2 (ja) 2025-11-17

Family

ID=77207241

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023501220A Active JP7771157B2 (ja) 2020-07-09 2021-07-08 オキソピロリジン fpr2アゴニスト

Country Status (8)

Country Link
US (1) US20230348426A1 (https=)
EP (1) EP4178946A1 (https=)
JP (1) JP7771157B2 (https=)
KR (1) KR20230038515A (https=)
CN (1) CN116034104B (https=)
AR (1) AR122912A1 (https=)
TW (1) TW202216664A (https=)
WO (1) WO2022011084A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7802765B2 (ja) 2020-08-12 2026-01-20 ブリストル-マイヤーズ スクイブ カンパニー オキソピロリジン尿素fpr2アゴニスト

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2752733T3 (es) * 2013-11-28 2020-04-06 Kyorin Seiyaku Kk Derivados de urea deuterados o marcados isotópicamente o sales farmacológicamente aceptables de los mismos útiles como agonistas de FPRL-1
WO2018227067A1 (en) * 2017-06-09 2018-12-13 Bristol-Myers Squibb Company Cyclopropyl urea formyl peptide 2 receptor and formyl peptide 1 receptor agonists
US10676431B2 (en) * 2018-03-05 2020-06-09 Bristol-Myers Squibb Company Phenylpyrrolidinone formyl peptide 2 receptor agonists
AR114383A1 (es) * 2018-03-09 2020-08-26 Gruenenthal Gmbh Piperidinas o piperidonas sustituidas con urea y fenilo
EP3880655A1 (en) * 2018-11-16 2021-09-22 Bristol-Myers Squibb Company Synthetic processes for the production of 1-((3s,4r)-4-(2,6-difluoro-4-methoxyphenyl)-2-oxopyrrolidin-3-yl)-3-phenylurea
CN113166134B (zh) * 2018-11-26 2024-06-14 百时美施贵宝公司 作为甲酰肽2受体激动剂的吡咯烷酮衍生物

Similar Documents

Publication Publication Date Title
JP2024050527A5 (https=)
RU2007124681A (ru) Производные тетрагидропирана в качестве противодиабетических средств
FI89356B (fi) Foerfarande foer framstaellnig av blodsockerhalten saenkande samt atherosklerosis hindrande tiazolidindioner
JP2024540163A5 (https=)
JP2023538408A5 (https=)
JP2023540609A5 (https=)
JP2021535174A5 (https=)
JP2025509281A5 (https=)
JP2021514001A5 (https=)
JP2022544714A5 (https=)
US20120165288A1 (en) Azapeptide derivatives
JP2021535177A5 (https=)
JP2012530703A5 (https=)
JP2023544476A5 (https=)
JP2024540164A5 (https=)
JP2024513227A5 (https=)
JP2021528451A5 (https=)
JP2024543013A5 (https=)
JP2023533037A5 (https=)
JP2022545158A5 (https=)
JP2023537410A5 (https=)
JP2021520394A5 (https=)
JP2022522890A5 (https=)
JPS60208975A (ja) 血小板活性化因子拮抗剤である新規2,5−ジアリ−ルテトラヒドロチオフエン類及びその類縁体
JP2022537350A5 (https=)