JP2023532330A5 - - Google Patents

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Publication number
JP2023532330A5
JP2023532330A5 JP2022581465A JP2022581465A JP2023532330A5 JP 2023532330 A5 JP2023532330 A5 JP 2023532330A5 JP 2022581465 A JP2022581465 A JP 2022581465A JP 2022581465 A JP2022581465 A JP 2022581465A JP 2023532330 A5 JP2023532330 A5 JP 2023532330A5
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JP
Japan
Prior art keywords
compound
formula
free base
salt
item
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022581465A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023532330A (ja
JP7792920B2 (ja
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Priority claimed from PCT/US2021/039305 external-priority patent/WO2022005928A1/en
Publication of JP2023532330A publication Critical patent/JP2023532330A/ja
Publication of JP2023532330A5 publication Critical patent/JP2023532330A5/ja
Priority to JP2025195295A priority Critical patent/JP2026027462A/ja
Application granted granted Critical
Publication of JP7792920B2 publication Critical patent/JP7792920B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022581465A 2020-06-30 2021-06-28 ピリジン-3-カルボン酸2-[4-[(2,3,4-トリメトキシフェニル)メチル]ピペラジン-1-イル]エチルの結晶形態および合成方法 Active JP7792920B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025195295A JP2026027462A (ja) 2020-06-30 2025-11-14 ピリジン-3-カルボン酸2-[4-[(2,3,4-トリメトキシフェニル)メチル]ピペラジン-1-イル]エチルの結晶形態および合成方法

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202063046123P 2020-06-30 2020-06-30
US202063046120P 2020-06-30 2020-06-30
US63/046,120 2020-06-30
US63/046,123 2020-06-30
PCT/US2021/039305 WO2022005928A1 (en) 2020-06-30 2021-06-28 Crystal forms of 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin -1-yl]ethyl pyridine-3-carboxylate and methods of synthesis

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025195295A Division JP2026027462A (ja) 2020-06-30 2025-11-14 ピリジン-3-カルボン酸2-[4-[(2,3,4-トリメトキシフェニル)メチル]ピペラジン-1-イル]エチルの結晶形態および合成方法

Publications (3)

Publication Number Publication Date
JP2023532330A JP2023532330A (ja) 2023-07-27
JP2023532330A5 true JP2023532330A5 (https=) 2024-06-21
JP7792920B2 JP7792920B2 (ja) 2025-12-26

Family

ID=79314883

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022581465A Active JP7792920B2 (ja) 2020-06-30 2021-06-28 ピリジン-3-カルボン酸2-[4-[(2,3,4-トリメトキシフェニル)メチル]ピペラジン-1-イル]エチルの結晶形態および合成方法
JP2025195295A Pending JP2026027462A (ja) 2020-06-30 2025-11-14 ピリジン-3-カルボン酸2-[4-[(2,3,4-トリメトキシフェニル)メチル]ピペラジン-1-イル]エチルの結晶形態および合成方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025195295A Pending JP2026027462A (ja) 2020-06-30 2025-11-14 ピリジン-3-カルボン酸2-[4-[(2,3,4-トリメトキシフェニル)メチル]ピペラジン-1-イル]エチルの結晶形態および合成方法

Country Status (8)

Country Link
EP (1) EP4171233A4 (https=)
JP (2) JP7792920B2 (https=)
KR (1) KR20230031320A (https=)
CN (1) CN116056711B (https=)
AU (1) AU2021299266A1 (https=)
CA (1) CA3188286A1 (https=)
IL (1) IL299547A (https=)
WO (1) WO2022005928A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023235297A1 (en) * 2022-06-03 2023-12-07 Imbria Pharmaceuticals, Inc. Compounds and methods for increasing efficiency of cardiac metabolism

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9169279B2 (en) * 2009-07-31 2015-10-27 Thar Pharmaceuticals, Inc. Crystallization method and bioavailability
CN102850296B (zh) * 2012-09-29 2015-01-07 瑞阳制药有限公司 曲美他嗪的制备方法
IL283725B2 (en) * 2017-06-20 2024-04-01 Imbria Pharmaceuticals Inc Compositions and methods for increasing efficiency of cardiac metabolism
EP3976103A4 (en) * 2019-05-31 2023-06-28 Imbria Pharmaceuticals, Inc. Methods of altering cardiac remodeling using compounds that promote glucose oxidation
EP3976101A4 (en) * 2019-05-31 2023-06-21 Imbria Pharmaceuticals, Inc. FIBROSIS TREATMENT METHODS USING COMPOUNDS THAT PROMOTE GLUCOSE OXIDATION

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