JP2023514280A5 - - Google Patents

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Publication number
JP2023514280A5
JP2023514280A5 JP2022549325A JP2022549325A JP2023514280A5 JP 2023514280 A5 JP2023514280 A5 JP 2023514280A5 JP 2022549325 A JP2022549325 A JP 2022549325A JP 2022549325 A JP2022549325 A JP 2022549325A JP 2023514280 A5 JP2023514280 A5 JP 2023514280A5
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JP
Japan
Prior art keywords
alkyl
group
cycloalkyl
hydroxy
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022549325A
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English (en)
Japanese (ja)
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JP2023514280A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/018863 external-priority patent/WO2021168313A1/en
Publication of JP2023514280A publication Critical patent/JP2023514280A/ja
Publication of JP2023514280A5 publication Critical patent/JP2023514280A5/ja
Pending legal-status Critical Current

Links

JP2022549325A 2020-02-19 2021-02-19 setd2阻害剤、および関連する方法と使用(併用療法を含む) Pending JP2023514280A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062978692P 2020-02-19 2020-02-19
US62/978,692 2020-02-19
PCT/US2021/018863 WO2021168313A1 (en) 2020-02-19 2021-02-19 Setd2 inhibitors and related methods and uses, including combination therapies

Publications (2)

Publication Number Publication Date
JP2023514280A JP2023514280A (ja) 2023-04-05
JP2023514280A5 true JP2023514280A5 (enExample) 2024-02-27

Family

ID=77391740

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022549325A Pending JP2023514280A (ja) 2020-02-19 2021-02-19 setd2阻害剤、および関連する方法と使用(併用療法を含む)

Country Status (11)

Country Link
US (1) US12691111B2 (enExample)
EP (1) EP4107157A4 (enExample)
JP (1) JP2023514280A (enExample)
KR (1) KR20220143116A (enExample)
CN (2) CN121695288A (enExample)
AU (1) AU2021224855A1 (enExample)
BR (1) BR112022016573A2 (enExample)
CA (1) CA3168069A1 (enExample)
IL (1) IL295654A (enExample)
MX (1) MX2022010171A (enExample)
WO (1) WO2021168313A1 (enExample)

Families Citing this family (8)

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CN121695288A (zh) 2020-02-19 2026-03-20 Epizyme股份有限公司 Setd2抑制剂和相关方法和用途,包括组合疗法
EP4351552A4 (en) * 2021-06-09 2025-06-18 Epizyme, Inc. COMBINATION THERAPIES WITH SETD2 INHIBITORS
CN117956995A (zh) * 2021-08-30 2024-04-30 江苏恒瑞医药股份有限公司 一种ezh2抑制剂用于制备治疗t细胞淋巴瘤的药物的用途
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CN117486779A (zh) * 2023-09-26 2024-02-02 青岛海洋生物医药研究院股份有限公司 一种3-羟基-2-氧化吲哚类化合物及其在制备抗肿瘤药物中的应用

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