JP2024533787A5 - - Google Patents

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Publication number
JP2024533787A5
JP2024533787A5 JP2024519528A JP2024519528A JP2024533787A5 JP 2024533787 A5 JP2024533787 A5 JP 2024533787A5 JP 2024519528 A JP2024519528 A JP 2024519528A JP 2024519528 A JP2024519528 A JP 2024519528A JP 2024533787 A5 JP2024533787 A5 JP 2024533787A5
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JP
Japan
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Pending
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JP2024519528A
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English (en)
Japanese (ja)
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JP2024533787A (ja
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Priority claimed from PCT/CN2022/122205 external-priority patent/WO2023051628A1/zh
Publication of JP2024533787A publication Critical patent/JP2024533787A/ja
Publication of JP2024533787A5 publication Critical patent/JP2024533787A5/ja
Pending legal-status Critical Current

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JP2024519528A 2021-09-29 2022-09-28 ピリド六員環構造を有するsos1阻害剤 Pending JP2024533787A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CN202111155906.7 2021-09-29
CN202111155906 2021-09-29
CN202211141499.9 2022-09-20
CN202211141499 2022-09-20
PCT/CN2022/122205 WO2023051628A1 (zh) 2021-09-29 2022-09-28 一类具有吡啶并六元环结构的sos1抑制剂

Publications (2)

Publication Number Publication Date
JP2024533787A JP2024533787A (ja) 2024-09-12
JP2024533787A5 true JP2024533787A5 (enExample) 2025-10-01

Family

ID=85781333

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024519528A Pending JP2024533787A (ja) 2021-09-29 2022-09-28 ピリド六員環構造を有するsos1阻害剤

Country Status (6)

Country Link
US (1) US20250042857A1 (enExample)
EP (1) EP4410790A4 (enExample)
JP (1) JP2024533787A (enExample)
CN (1) CN117999263A (enExample)
TW (1) TW202320766A (enExample)
WO (1) WO2023051628A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022184116A1 (zh) * 2021-03-05 2022-09-09 江苏先声药业有限公司 新型sos1抑制剂及其制备方法和应用
CN117024404A (zh) * 2022-05-10 2023-11-10 四川汇宇制药股份有限公司 苯并吡啶衍生物及其用途
WO2025188163A1 (ko) * 2024-03-07 2025-09-12 아이리드비엠에스 주식회사 Sos1 억제제 및 이의 용도

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003055866A1 (en) * 2001-12-21 2003-07-10 Bayer Pharmaceuticals Corporation Quinazoline and quinoline derivative compounds as inhibitors of prolylpeptidase, inducers of apoptosis and cancer treatment agents
HUP0302440A3 (en) * 2003-07-31 2007-08-28 Sanofi Aventis Aminoquinoline derivatives, process for producing them and pharmaceutical compositions containing them
EP2581372B1 (en) * 2010-06-09 2017-06-07 Tianjin Hemay Oncology Pharmaceutical Co., Ltd. Cyanoquinoline derivatives
WO2014120995A2 (en) * 2013-02-01 2014-08-07 Wellstat Therapeutics Corporation Amine compounds having anti-inflammatory, antifungal, antiparasitic and anticancer activity
EA033686B1 (ru) * 2015-08-03 2019-11-15 Bristol Myers Squibb Co Гетероциклические соединения, применимые в качестве модуляторов tnf-альфа
CA3156359A1 (en) 2019-11-08 2021-05-14 Adrian Liam Gill Bicyclic heteroaryl compounds and uses thereof
WO2022156792A1 (en) * 2021-01-25 2022-07-28 Guangdong Newopp Biopharmaceuticals Co., Ltd. Heterocyclic compounds as sos1 inhibitors
WO2022161461A1 (zh) * 2021-01-29 2022-08-04 江苏先声药业有限公司 Sos1抑制剂及其制备方法和应用
CN115043842A (zh) * 2021-03-09 2022-09-13 苏州泽璟生物制药股份有限公司 胺基取代双环类抑制剂及其制备方法和应用

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