JP2023510918A5 - - Google Patents

Info

Publication number
JP2023510918A5
JP2023510918A5 JP2022543496A JP2022543496A JP2023510918A5 JP 2023510918 A5 JP2023510918 A5 JP 2023510918A5 JP 2022543496 A JP2022543496 A JP 2022543496A JP 2022543496 A JP2022543496 A JP 2022543496A JP 2023510918 A5 JP2023510918 A5 JP 2023510918A5
Authority
JP
Japan
Prior art keywords
cycloalkyl
alkyl
pharmaceutically acceptable
acceptable salt
bonded
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022543496A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023510918A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/013359 external-priority patent/WO2021146370A1/en
Publication of JP2023510918A publication Critical patent/JP2023510918A/ja
Publication of JP2023510918A5 publication Critical patent/JP2023510918A5/ja
Pending legal-status Critical Current

Links

JP2022543496A 2020-01-15 2021-01-14 Map4k1阻害剤 Pending JP2023510918A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062961463P 2020-01-15 2020-01-15
US62/961,463 2020-01-15
PCT/US2021/013359 WO2021146370A1 (en) 2020-01-15 2021-01-14 Map4k1 inhibitors

Publications (2)

Publication Number Publication Date
JP2023510918A JP2023510918A (ja) 2023-03-15
JP2023510918A5 true JP2023510918A5 (enExample) 2024-01-23

Family

ID=74557263

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022543496A Pending JP2023510918A (ja) 2020-01-15 2021-01-14 Map4k1阻害剤

Country Status (7)

Country Link
US (2) US11534441B2 (enExample)
EP (1) EP4090663A1 (enExample)
JP (1) JP2023510918A (enExample)
CN (1) CN115279771B (enExample)
AR (1) AR121047A1 (enExample)
TW (1) TW202140473A (enExample)
WO (1) WO2021146370A1 (enExample)

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WO2020092528A1 (en) 2018-10-31 2020-05-07 Gilead Sciences, Inc. Substituted 6-azabenzimidazole compounds having hpk1 inhibitory activity
EP3972695A1 (en) 2019-05-23 2022-03-30 Gilead Sciences, Inc. Substituted exo-methylene-oxindoles which are hpk1/map4k1 inhibitors
MX2022007969A (es) 2019-12-23 2022-12-13 Blueprint Medicines Corp Inhibidores de egfr.
TW202140473A (zh) 2020-01-15 2021-11-01 美商纜圖藥品公司 Map4k1抑制劑
CN117295748A (zh) * 2021-03-08 2023-12-26 缆图药品公司 Map4k1抑制剂
EP4305041A1 (en) * 2021-03-08 2024-01-17 Blueprint Medicines Corporation Map4k1 inhibitors
WO2023288254A1 (en) * 2021-07-14 2023-01-19 Blueprint Medicines Corporation Heterocyclic compounds as map4k1 inhibitors
US20240336630A1 (en) * 2021-07-15 2024-10-10 Blueprint Medicines Corporation Map4k1 inhibitors
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WO2024196841A1 (en) * 2023-03-21 2024-09-26 Athos Therapeutics, Inc. Vanin-1 inhibitors
CN121548580A (zh) * 2023-05-15 2026-02-17 亚历克西亚治疗公司 Cdk抑制剂化合物
WO2025080099A1 (ko) * 2023-10-13 2025-04-17 주식회사유한양행 7,7-다이메틸푸로[3,4-b]피리딘-5(7h)-온 유도체 또는 이의 염 및 이를 포함하는 약학 조성물

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TW202140473A (zh) 2020-01-15 2021-11-01 美商纜圖藥品公司 Map4k1抑制劑
EP4305041A1 (en) 2021-03-08 2024-01-17 Blueprint Medicines Corporation Map4k1 inhibitors
WO2023288254A1 (en) 2021-07-14 2023-01-19 Blueprint Medicines Corporation Heterocyclic compounds as map4k1 inhibitors

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