JP2023502030A5 - - Google Patents
Info
- Publication number
- JP2023502030A5 JP2023502030A5 JP2022527713A JP2022527713A JP2023502030A5 JP 2023502030 A5 JP2023502030 A5 JP 2023502030A5 JP 2022527713 A JP2022527713 A JP 2022527713A JP 2022527713 A JP2022527713 A JP 2022527713A JP 2023502030 A5 JP2023502030 A5 JP 2023502030A5
- Authority
- JP
- Japan
- Prior art keywords
- peaks
- methyl
- compound
- crystalline
- powder
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025132388A JP2025159062A (ja) | 2019-11-14 | 2025-08-07 | 複素環式化合物およびその使用 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019206311 | 2019-11-14 | ||
| JP2019206311A JP2021080177A (ja) | 2019-11-14 | 2019-11-14 | 複素環化合物及びその用途 |
| PCT/IB2020/000962 WO2021094832A1 (en) | 2019-11-14 | 2020-11-12 | Heterocyclic nmda antagonists |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025132388A Division JP2025159062A (ja) | 2019-11-14 | 2025-08-07 | 複素環式化合物およびその使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023502030A JP2023502030A (ja) | 2023-01-20 |
| JP2023502030A5 true JP2023502030A5 (https=) | 2023-11-20 |
| JP7726879B2 JP7726879B2 (ja) | 2025-08-20 |
Family
ID=74141594
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019206311A Pending JP2021080177A (ja) | 2019-11-14 | 2019-11-14 | 複素環化合物及びその用途 |
| JP2022527713A Active JP7726879B2 (ja) | 2019-11-14 | 2020-11-12 | 複素環式化合物およびその使用 |
| JP2025132388A Pending JP2025159062A (ja) | 2019-11-14 | 2025-08-07 | 複素環式化合物およびその使用 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019206311A Pending JP2021080177A (ja) | 2019-11-14 | 2019-11-14 | 複素環化合物及びその用途 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025132388A Pending JP2025159062A (ja) | 2019-11-14 | 2025-08-07 | 複素環式化合物およびその使用 |
Country Status (21)
| Country | Link |
|---|---|
| US (3) | US20230002318A1 (https=) |
| EP (1) | EP4058430A1 (https=) |
| JP (3) | JP2021080177A (https=) |
| KR (1) | KR20220102629A (https=) |
| CN (1) | CN114728900A (https=) |
| AR (1) | AR120452A1 (https=) |
| AU (1) | AU2020385250A1 (https=) |
| BR (1) | BR112022008367A2 (https=) |
| CA (1) | CA3158352A1 (https=) |
| CL (1) | CL2022001241A1 (https=) |
| CO (1) | CO2022008012A2 (https=) |
| CR (1) | CR20220275A (https=) |
| DO (1) | DOP2022000099A (https=) |
| EC (1) | ECSP22037602A (https=) |
| IL (1) | IL292639A (https=) |
| JO (1) | JOP20220108A1 (https=) |
| MX (1) | MX2022005778A (https=) |
| PE (1) | PE20221767A1 (https=) |
| PH (1) | PH12022551173A1 (https=) |
| TW (1) | TWI908745B (https=) |
| WO (1) | WO2021094832A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CR20220160A (es) | 2019-09-16 | 2022-06-16 | Takeda Pharmaceuticals Co | Derivados de piridazin-3(2h)-ona fusionados con azol |
| JP2021050161A (ja) | 2019-09-25 | 2021-04-01 | 武田薬品工業株式会社 | 複素環化合物及びその用途 |
| JP2021080177A (ja) | 2019-11-14 | 2021-05-27 | 武田薬品工業株式会社 | 複素環化合物及びその用途 |
| WO2026060343A1 (en) | 2024-09-16 | 2026-03-19 | Neurocrine Biosciences, Inc. | Solid forms comprising a nr2b nam antagonist |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2001500852A (ja) | 1996-08-27 | 2001-01-23 | プレーシス ファーマスーティカルズ インコーポレイテッド | D―アミノ酸を含むβ―アミロイドペプチド凝集のモジュレーター |
| WO2000017162A1 (en) * | 1998-09-21 | 2000-03-30 | Takeda Chemical Industries, Ltd. | Novel thiol derivatives, process for producing the same and utilization thereof |
| JP2000159747A (ja) * | 1998-09-21 | 2000-06-13 | Takeda Chem Ind Ltd | 新規チオ―ル誘導体、その製造法および用途 |
| CA2374610A1 (en) | 1999-06-28 | 2001-01-04 | Jordan J. N. Tang | Catalytically active recombinant memapsin and methods of use thereof |
| AU1153601A (en) * | 1999-10-29 | 2001-05-08 | Merck Sharp & Dohme Limited | Method to treat pain utilizing benzimidazole NMDA NR2B antagonists |
| JPWO2003035641A1 (ja) * | 2001-10-22 | 2005-02-10 | 塩野義製薬株式会社 | 新規カルバモイルピロリドン誘導体 |
| JP2004002405A (ja) * | 2002-04-26 | 2004-01-08 | Takeda Chem Ind Ltd | 新規チオール誘導体、その製造法および用途 |
| AU2003235121A1 (en) | 2002-04-26 | 2003-11-10 | Takeda Pharmaceutical Company Limited | Novel thiol derivative, process for producing the same and use thereof |
| TW200732313A (en) * | 2005-12-15 | 2007-09-01 | Astrazeneca Ab | Oxazolidinone compounds and their use as metabotropic glutamate receptor potentiators |
| TWI403320B (zh) | 2005-12-16 | 2013-08-01 | Infinity Discovery Inc | 用於抑制bcl蛋白和結合夥伴間之交互作用的化合物及方法 |
| WO2009004430A1 (en) * | 2007-06-29 | 2009-01-08 | Pfizer Inc. | N-benzyl oxazolidinones and related heterocycleic compounds as potentiators of glutamate receptors |
| PL3110434T3 (pl) | 2014-02-24 | 2019-01-31 | Takeda Gmbh | Białka fuzyjne uti |
| CN107074788B (zh) * | 2014-10-31 | 2019-09-20 | 厦门大学 | 取代杂环衍生物、其制备方法和用途 |
| WO2018205935A1 (zh) | 2017-05-09 | 2018-11-15 | 浙江大学 | 治疗抑郁症的方法和药物组合物 |
| JP6806735B2 (ja) | 2018-05-30 | 2021-01-06 | 矢崎総業株式会社 | 車両用回路体および車両用回路体の製造方法 |
| WO2020081999A1 (en) | 2018-10-18 | 2020-04-23 | Essa Pharma, Inc. | Androgen receptor modulators and methods for their use |
| CA3134545A1 (en) | 2019-03-28 | 2020-10-01 | Essa Pharma, Inc. | Pharmaceutical compositions and combinations comprising inhibitors of the androgen receptor and uses thereof |
| JP2021080177A (ja) | 2019-11-14 | 2021-05-27 | 武田薬品工業株式会社 | 複素環化合物及びその用途 |
-
2019
- 2019-11-14 JP JP2019206311A patent/JP2021080177A/ja active Pending
-
2020
- 2020-11-12 EP EP20838595.5A patent/EP4058430A1/en active Pending
- 2020-11-12 CN CN202080079710.1A patent/CN114728900A/zh active Pending
- 2020-11-12 TW TW109139608A patent/TWI908745B/zh active
- 2020-11-12 MX MX2022005778A patent/MX2022005778A/es unknown
- 2020-11-12 BR BR112022008367A patent/BR112022008367A2/pt unknown
- 2020-11-12 JP JP2022527713A patent/JP7726879B2/ja active Active
- 2020-11-12 US US17/755,907 patent/US20230002318A1/en active Pending
- 2020-11-12 PE PE2022000751A patent/PE20221767A1/es unknown
- 2020-11-12 AR ARP200103139A patent/AR120452A1/es unknown
- 2020-11-12 AU AU2020385250A patent/AU2020385250A1/en active Pending
- 2020-11-12 WO PCT/IB2020/000962 patent/WO2021094832A1/en not_active Ceased
- 2020-11-12 CR CR20220275A patent/CR20220275A/es unknown
- 2020-11-12 PH PH1/2022/551173A patent/PH12022551173A1/en unknown
- 2020-11-12 CA CA3158352A patent/CA3158352A1/en active Pending
- 2020-11-12 KR KR1020227019888A patent/KR20220102629A/ko active Pending
-
2022
- 2022-05-01 IL IL292639A patent/IL292639A/en unknown
- 2022-05-10 JO JOP/2022/0108A patent/JOP20220108A1/ar unknown
- 2022-05-12 EC ECSENADI202237602A patent/ECSP22037602A/es unknown
- 2022-05-12 CL CL2022001241A patent/CL2022001241A1/es unknown
- 2022-05-13 DO DO2022000099A patent/DOP2022000099A/es unknown
- 2022-06-06 CO CONC2022/0008012A patent/CO2022008012A2/es unknown
- 2022-12-22 US US18/087,233 patent/US11834409B2/en active Active
- 2022-12-22 US US18/087,302 patent/US11827601B2/en active Active
-
2025
- 2025-08-07 JP JP2025132388A patent/JP2025159062A/ja active Pending
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