JP2023500408A5 - - Google Patents

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Publication number
JP2023500408A5
JP2023500408A5 JP2022527081A JP2022527081A JP2023500408A5 JP 2023500408 A5 JP2023500408 A5 JP 2023500408A5 JP 2022527081 A JP2022527081 A JP 2022527081A JP 2022527081 A JP2022527081 A JP 2022527081A JP 2023500408 A5 JP2023500408 A5 JP 2023500408A5
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JP
Japan
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alkyl
compound
compound according
disease
substituted
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JP2022527081A
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English (en)
Japanese (ja)
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JP7721517B2 (ja
JP2023500408A (ja
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Priority claimed from PCT/US2020/060180 external-priority patent/WO2021097057A1/en
Publication of JP2023500408A publication Critical patent/JP2023500408A/ja
Publication of JP2023500408A5 publication Critical patent/JP2023500408A5/ja
Priority to JP2025126773A priority Critical patent/JP2025160375A/ja
Application granted granted Critical
Publication of JP7721517B2 publication Critical patent/JP7721517B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022527081A 2019-11-12 2020-11-12 Cftr活性の欠損が介在する状態を治療するための5員ヘテロアリールアミノスルホンアミド Active JP7721517B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025126773A JP2025160375A (ja) 2019-11-12 2025-07-30 Cftr活性の欠損が介在する状態を治療するための5員ヘテロアリールアミノスルホンアミド

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962934293P 2019-11-12 2019-11-12
US62/934,293 2019-11-12
PCT/US2020/060180 WO2021097057A1 (en) 2019-11-12 2020-11-12 5-membered heteroarylaminosulfonamides for treating conditions mediated by deficient cftr activity

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025126773A Division JP2025160375A (ja) 2019-11-12 2025-07-30 Cftr活性の欠損が介在する状態を治療するための5員ヘテロアリールアミノスルホンアミド

Publications (3)

Publication Number Publication Date
JP2023500408A JP2023500408A (ja) 2023-01-05
JP2023500408A5 true JP2023500408A5 (enExample) 2023-11-20
JP7721517B2 JP7721517B2 (ja) 2025-08-12

Family

ID=73740547

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022527081A Active JP7721517B2 (ja) 2019-11-12 2020-11-12 Cftr活性の欠損が介在する状態を治療するための5員ヘテロアリールアミノスルホンアミド
JP2025126773A Pending JP2025160375A (ja) 2019-11-12 2025-07-30 Cftr活性の欠損が介在する状態を治療するための5員ヘテロアリールアミノスルホンアミド

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025126773A Pending JP2025160375A (ja) 2019-11-12 2025-07-30 Cftr活性の欠損が介在する状態を治療するための5員ヘテロアリールアミノスルホンアミド

Country Status (17)

Country Link
US (1) US20240002374A1 (enExample)
EP (1) EP4058439A1 (enExample)
JP (2) JP7721517B2 (enExample)
KR (2) KR20260078949A (enExample)
CN (2) CN122562796A (enExample)
AU (1) AU2020384279A1 (enExample)
BR (1) BR112022009185A2 (enExample)
CA (1) CA3158057A1 (enExample)
CL (1) CL2022001245A1 (enExample)
CO (1) CO2022007953A2 (enExample)
EC (1) ECSP22046050A (enExample)
IL (1) IL292966A (enExample)
JO (1) JOP20220105A1 (enExample)
MX (1) MX2022005809A (enExample)
PE (1) PE20221461A1 (enExample)
PH (1) PH12022551139A1 (enExample)
WO (1) WO2021097057A1 (enExample)

Families Citing this family (17)

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Publication number Priority date Publication date Assignee Title
RS64018B1 (sr) 2018-02-15 2023-03-31 Vertex Pharma Makrocikli kao modulatori transmembranskog regulatora provodnosti cistične fibroze, njihove farmaceutske kompozicije, njihova upotreba u lečenju cistične fibroze i proces njihove izrade
TWI848092B (zh) 2019-04-03 2024-07-11 美商維泰克斯製藥公司 囊腫纖維化跨膜傳導調節蛋白調節劑
US11873300B2 (en) 2019-08-14 2024-01-16 Vertex Pharmaceuticals Incorporated Crystalline forms of CFTR modulators
TWI867024B (zh) 2019-08-14 2024-12-21 美商維泰克斯製藥公司 囊腫纖維化跨膜傳導調節蛋白之調節劑
TWI899097B (zh) 2019-08-14 2025-10-01 美商維泰克斯製藥公司 製備cftr調節劑之方法
MX2022005810A (es) 2019-11-12 2022-06-08 Genzyme Corp Heteroarilaminosulfonamidas de 6 miembros para tratar enfermedades y afecciones mediadas por la actividad de regulador de la conductancia transmembrana de la fibrosis quistica (cftr) deficiente.
WO2021113806A1 (en) 2019-12-05 2021-06-10 Genzyme Corporation Arylamides and methods of use thereof
WO2021113808A1 (en) 2019-12-05 2021-06-10 Genzyme Corporation Cftr-modulating arylamides
WO2021113809A1 (en) 2019-12-05 2021-06-10 Genzyme Corporation Arylamides and methods of use thereof
WO2022076628A1 (en) * 2020-10-07 2022-04-14 Vertex Pharmaceuticals Incorporated Modulators of cystic fibrosis transmembrane conductance regulator
MX2023006770A (es) 2020-12-10 2023-08-14 Vertex Pharma Metodos de tratamiento para fibrosis quistica.
CN113480416B (zh) * 2021-07-12 2023-03-21 重庆大学 一种芳基酮的制备方法
IL315190A (en) 2022-03-30 2024-10-01 Ishihara Sangyo Kaisha A pyridazinone compound or a salt thereof and a pesticide containing them
CN114835655A (zh) * 2022-04-14 2022-08-02 河南师范大学 一种合成光学活性三氟甲基丙烯酸酯类化合物的方法
EP4611742A1 (en) 2022-10-31 2025-09-10 Sionna Therapeutics Inc. Methods of treating cftr-mediated diseases or disorders
EP4746882A1 (en) * 2023-07-20 2026-05-27 CeMM - Forschungszentrum für Molekulare Medizin GmbH Inhibitors of smndc1 and their therapeutic use
CN122374316A (zh) 2023-10-04 2026-07-10 弗特克斯药品有限公司 囊性纤维化跨膜传导调控因子的调节剂

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU654125B2 (en) * 1991-03-07 1994-10-27 Hisamitsu Pharmaceutical Co., Inc. Novel diphenylthyazole derivative
EP0790057B1 (en) * 1994-11-29 2002-06-05 Hisamitsu Pharmaceutical Co., Inc. Antibacterial or bactericide comprising 2-aminothiazole derivative and salts thereof
JP2005510508A (ja) * 2001-11-08 2005-04-21 藤沢薬品工業株式会社 アデノシンアンタゴニストとしてのチアゾールピリダジノン類
US7973169B2 (en) 2003-09-06 2011-07-05 Vertex Pharmaceuticals Incorporated Modulators of ATP-Binding Cassette transporters
AU2012267732A1 (en) 2011-06-10 2014-01-09 Medimmune Limited Anti-Pseudomonas Psl binding molecules and uses thereof
WO2016183173A1 (en) * 2015-05-12 2016-11-17 Avista Pharma Solutions Antiparasitic compounds
US10138227B2 (en) * 2016-06-03 2018-11-27 Abbvie S.Á.R.L. Heteroaryl substituted pyridines and methods of use
TW201811766A (zh) * 2016-08-29 2018-04-01 瑞士商諾華公司 N-(吡啶-2-基)吡啶-磺醯胺衍生物及其用於疾病治療之用途
EP4611742A1 (en) * 2022-10-31 2025-09-10 Sionna Therapeutics Inc. Methods of treating cftr-mediated diseases or disorders

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