JP2022549169A5 - - Google Patents

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Publication number
JP2022549169A5
JP2022549169A5 JP2022517438A JP2022517438A JP2022549169A5 JP 2022549169 A5 JP2022549169 A5 JP 2022549169A5 JP 2022517438 A JP2022517438 A JP 2022517438A JP 2022517438 A JP2022517438 A JP 2022517438A JP 2022549169 A5 JP2022549169 A5 JP 2022549169A5
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JP
Japan
Prior art keywords
inhibitors
pharmaceutically acceptable
acceptable salt
compound according
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2022517438A
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English (en)
Japanese (ja)
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JP2022549169A (ja
JP7652434B2 (ja
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Priority claimed from PCT/US2020/051430 external-priority patent/WO2021055705A1/en
Publication of JP2022549169A publication Critical patent/JP2022549169A/ja
Publication of JP2022549169A5 publication Critical patent/JP2022549169A5/ja
Priority to JP2025036781A priority Critical patent/JP2025094953A/ja
Application granted granted Critical
Publication of JP7652434B2 publication Critical patent/JP7652434B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022517438A 2019-09-18 2020-09-18 がん治療のためのビアミノキノリンとナノ製剤 Active JP7652434B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025036781A JP2025094953A (ja) 2019-09-18 2025-03-07 がん治療のためのビアミノキノリンとナノ製剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962902156P 2019-09-18 2019-09-18
US62/902,156 2019-09-18
PCT/US2020/051430 WO2021055705A1 (en) 2019-09-18 2020-09-18 Biaminoquinolines and nanoformulations for cancer treatment

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025036781A Division JP2025094953A (ja) 2019-09-18 2025-03-07 がん治療のためのビアミノキノリンとナノ製剤

Publications (3)

Publication Number Publication Date
JP2022549169A JP2022549169A (ja) 2022-11-24
JP2022549169A5 true JP2022549169A5 (https=) 2023-09-25
JP7652434B2 JP7652434B2 (ja) 2025-03-27

Family

ID=74884705

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022517438A Active JP7652434B2 (ja) 2019-09-18 2020-09-18 がん治療のためのビアミノキノリンとナノ製剤
JP2025036781A Pending JP2025094953A (ja) 2019-09-18 2025-03-07 がん治療のためのビアミノキノリンとナノ製剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025036781A Pending JP2025094953A (ja) 2019-09-18 2025-03-07 がん治療のためのビアミノキノリンとナノ製剤

Country Status (6)

Country Link
US (1) US20230348419A1 (https=)
EP (1) EP4031543A4 (https=)
JP (2) JP7652434B2 (https=)
CN (2) CN115023418B (https=)
CA (1) CA3154678A1 (https=)
WO (1) WO2021055705A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3099155A1 (en) 2018-05-14 2019-11-21 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds
CA3138197A1 (en) 2019-05-14 2020-11-19 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds
CN115023418B (zh) * 2019-09-18 2024-11-19 加利福尼亚大学董事会 用于癌症治疗的双氨基喹啉和纳米制剂
EP4058464A1 (en) 2019-11-13 2022-09-21 Nuvation Bio Inc. Anti-cancer nuclear hormone receptor-targeting compounds
MX2023011241A (es) 2021-03-23 2023-10-03 Nuvation Bio Inc Compuestos dirigidos a receptores de hormonas nucleares contra el cancer.
JP2024516024A (ja) 2021-05-03 2024-04-11 ニューベイション・バイオ・インコーポレイテッド 抗がん核内ホルモン受容体標的化化合物
CN114948938B (zh) * 2022-02-22 2023-08-11 江苏省中医院 白术内酯i在制备预防和/或治疗宫颈癌的药物中的用途
CN114948901B (zh) * 2022-05-06 2023-04-21 郑州大学第一附属医院 一种协同治疗乳腺癌的依西美坦纳米粒、制剂及其制备方法
CN116059172B (zh) * 2023-02-01 2025-05-13 中山大学附属第八医院(深圳福田) 一种纳米递药系统及其制备方法与应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006522814A (ja) * 2003-04-11 2006-10-05 タイゲン・バイオテクノロジー アミノキノリン化合物
WO2011115555A1 (en) * 2010-03-16 2011-09-22 Ge Healthcare Bio-Sciences Ab System for improved delivery of gene modulating compounds
US20140050696A1 (en) * 2011-04-29 2014-02-20 Ravi K. Amaravadi Novel bisaminoquinoline compounds, pharmaceutical compositions prepared therefrom and their use
WO2015068142A2 (en) * 2013-11-11 2015-05-14 Cellworks Group, Inc. Compositions, process of preparation of said compositions, uses and method of management of myeloproliferative disorder
ES2881048T3 (es) * 2014-08-08 2021-11-26 Univ Pennsylvania Bisaminoquinolinas asimétricas y bisaminoquinolinas con enlazadores variados como inhibidores de la autofagia para el cáncer y otras terapias
US10774047B2 (en) * 2015-04-17 2020-09-15 The Trustees Of The University Of Pennsylvania Dimeric quinacrine derivatives as autophagy inhibitors for cancer therapy
GB2555270A (en) * 2015-05-29 2018-04-25 Presage Biosciences Inc Autophagy-inhibiting compounds and uses thereof
US20180280372A1 (en) * 2016-11-22 2018-10-04 Washington University Compositions and methods for inhibiting autophagy and contraception
CN115023418B (zh) * 2019-09-18 2024-11-19 加利福尼亚大学董事会 用于癌症治疗的双氨基喹啉和纳米制剂

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