JP2022546861A5 - - Google Patents

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Publication number
JP2022546861A5
JP2022546861A5 JP2022515704A JP2022515704A JP2022546861A5 JP 2022546861 A5 JP2022546861 A5 JP 2022546861A5 JP 2022515704 A JP2022515704 A JP 2022515704A JP 2022515704 A JP2022515704 A JP 2022515704A JP 2022546861 A5 JP2022546861 A5 JP 2022546861A5
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JP
Japan
Application number
JP2022515704A
Other languages
Japanese (ja)
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JPWO2021050580A5 (https=
JP2022546861A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/049986 external-priority patent/WO2021050580A1/en
Publication of JP2022546861A publication Critical patent/JP2022546861A/ja
Publication of JPWO2021050580A5 publication Critical patent/JPWO2021050580A5/ja
Publication of JP2022546861A5 publication Critical patent/JP2022546861A5/ja
Priority to JP2025061710A priority Critical patent/JP2025102940A/ja
Pending legal-status Critical Current

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JP2022515704A 2019-09-10 2020-09-09 マルチチロシンキナーゼ阻害剤の結晶形、調製方法およびその使用 Pending JP2022546861A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025061710A JP2025102940A (ja) 2019-09-10 2025-04-03 マルチチロシンキナーゼ阻害剤の結晶形、調製方法およびその使用

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962898469P 2019-09-10 2019-09-10
US62/898,469 2019-09-10
PCT/US2020/049986 WO2021050580A1 (en) 2019-09-10 2020-09-09 Crystalline form of a multi-tyrosine kinase inhibitor, method of preparation, and use thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025061710A Division JP2025102940A (ja) 2019-09-10 2025-04-03 マルチチロシンキナーゼ阻害剤の結晶形、調製方法およびその使用

Publications (3)

Publication Number Publication Date
JP2022546861A JP2022546861A (ja) 2022-11-09
JPWO2021050580A5 JPWO2021050580A5 (https=) 2023-06-16
JP2022546861A5 true JP2022546861A5 (https=) 2023-06-16

Family

ID=74866002

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022515704A Pending JP2022546861A (ja) 2019-09-10 2020-09-09 マルチチロシンキナーゼ阻害剤の結晶形、調製方法およびその使用
JP2025061710A Pending JP2025102940A (ja) 2019-09-10 2025-04-03 マルチチロシンキナーゼ阻害剤の結晶形、調製方法およびその使用

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025061710A Pending JP2025102940A (ja) 2019-09-10 2025-04-03 マルチチロシンキナーゼ阻害剤の結晶形、調製方法およびその使用

Country Status (6)

Country Link
US (1) US12466838B2 (https=)
EP (1) EP4027999B1 (https=)
JP (2) JP2022546861A (https=)
CN (1) CN114401720A (https=)
CA (1) CA3150267A1 (https=)
WO (1) WO2021050580A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202302597A (zh) * 2021-03-10 2023-01-16 美商米拉蒂醫療公司 多重酪胺酸激酶抑制劑之結晶鹽、其製備方法及用途
WO2022240802A1 (en) 2021-05-10 2022-11-17 Teva Pharmaceuticals International Gmbh Solid state forms of sitravatinib salts and processes for preparation thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101125932B1 (ko) 2006-12-06 2012-03-22 아이디유엔 파마슈티칼즈, 인코포레이티드 (3s)-3-[n-(n'-(2-tert-부틸페닐)옥사밀)알라니닐]아미노-5-(2',3',5',6'-테트라플루오로페녹시)-4-옥소펜탄산의 결정 형태
BRPI0816064B8 (pt) * 2007-08-29 2021-05-25 Methylgene Inc composto inibidor da atividade de proteína tirosina quinase, seu uso, e composição farmacêutica
US8907091B2 (en) * 2007-08-29 2014-12-09 Methylgene Inc. Processes and intermediates for preparing fused heterocyclic kinase inhibitors
US20180237378A1 (en) * 2015-08-19 2018-08-23 Sandoz Ag Asymmetric Bisamidation of Malonic Ester Derivatives
EP3740491A1 (en) * 2018-01-18 2020-11-25 Array Biopharma, Inc. Substituted pyrrolo[2,3-d]pyrimidines compounds as ret kinase inhibitors
CN109384799B (zh) * 2018-11-12 2020-07-14 深圳海王医药科技研究院有限公司 一种多靶点激酶抑制剂化合物的晶型a及制备方法和含有其的药物组合物

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