JP2020536944A5 - - Google Patents

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Publication number
JP2020536944A5
JP2020536944A5 JP2020521319A JP2020521319A JP2020536944A5 JP 2020536944 A5 JP2020536944 A5 JP 2020536944A5 JP 2020521319 A JP2020521319 A JP 2020521319A JP 2020521319 A JP2020521319 A JP 2020521319A JP 2020536944 A5 JP2020536944 A5 JP 2020536944A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020521319A
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Japanese (ja)
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JP2020536944A (ja
JPWO2019079299A5 (https=
JP7776258B2 (ja
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Publication date
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Priority claimed from PCT/US2018/056083 external-priority patent/WO2019079299A1/en
Publication of JP2020536944A publication Critical patent/JP2020536944A/ja
Priority to JP2023151499A priority Critical patent/JP2024001040A/ja
Publication of JP2020536944A5 publication Critical patent/JP2020536944A5/ja
Publication of JPWO2019079299A5 publication Critical patent/JPWO2019079299A5/ja
Application granted granted Critical
Publication of JP7776258B2 publication Critical patent/JP7776258B2/ja
Active legal-status Critical Current
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JP2020521319A 2017-10-16 2018-10-16 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態 Active JP7776258B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023151499A JP2024001040A (ja) 2017-10-16 2023-09-19 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762572603P 2017-10-16 2017-10-16
US62/572,603 2017-10-16
PCT/US2018/056083 WO2019079299A1 (en) 2017-10-16 2018-10-16 SOLID FORMS OF 3- (5-FLUOROBENZOFURAN-3-YL) -4- (5-METHYL-5H- [1,3] DIOXOLO [4,5-F] INDOL-7-YL) PYRROLE-2,5-DIONE

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023151499A Division JP2024001040A (ja) 2017-10-16 2023-09-19 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Publications (4)

Publication Number Publication Date
JP2020536944A JP2020536944A (ja) 2020-12-17
JP2020536944A5 true JP2020536944A5 (https=) 2025-09-10
JPWO2019079299A5 JPWO2019079299A5 (https=) 2025-09-10
JP7776258B2 JP7776258B2 (ja) 2025-11-26

Family

ID=64110166

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020521319A Active JP7776258B2 (ja) 2017-10-16 2018-10-16 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態
JP2023151499A Pending JP2024001040A (ja) 2017-10-16 2023-09-19 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023151499A Pending JP2024001040A (ja) 2017-10-16 2023-09-19 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Country Status (16)

Country Link
US (3) US11407759B2 (https=)
EP (1) EP3697794B1 (https=)
JP (2) JP7776258B2 (https=)
KR (1) KR102891811B1 (https=)
CN (1) CN111315748B (https=)
AU (1) AU2018352384B2 (https=)
CA (1) CA3074037A1 (https=)
DK (1) DK3697794T3 (https=)
ES (1) ES3064009T3 (https=)
FI (1) FI3697794T3 (https=)
IL (1) IL273920B2 (https=)
MX (1) MX2020003431A (https=)
PL (1) PL3697794T3 (https=)
PT (1) PT3697794T (https=)
WO (1) WO2019079299A1 (https=)
ZA (1) ZA202002740B (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL3697794T3 (pl) * 2017-10-16 2026-04-07 Actuate Therapeutics Inc. Stałe postacie 3-(5-fluorobenzofuran-3-ylo)-4-(5-metylo-5h-[1,3]dioksolo[4,5-f]indol-7-ilo)pirolo-2,5-dionu
WO2019222483A1 (en) * 2018-05-17 2019-11-21 Board Of Regents, The University Of Texas System Treatment of idiopathic pulmonary fibrosis with glycogen synthase kinase 3 form beta inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2673368C (en) 2006-12-19 2014-10-28 The Board Of Trustees Of The University Of Illinois 3-benzofuranyl-4-indolyl maleimides as potent gsk3 inhibitors for neurogenerative disorders
EP3665176B1 (en) * 2017-08-11 2024-01-24 Actuate Therapeutics Inc. Solid forms of 3-(5-fluorobenzofuran-3-yl)-4-(5-methyl-5h[1,3]dioxolo[4,5-f]indol-7-yl)pyrrole-2,5-dione
PL3697794T3 (pl) * 2017-10-16 2026-04-07 Actuate Therapeutics Inc. Stałe postacie 3-(5-fluorobenzofuran-3-ylo)-4-(5-metylo-5h-[1,3]dioksolo[4,5-f]indol-7-ilo)pirolo-2,5-dionu

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