JP2022541772A5 - - Google Patents

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Publication number
JP2022541772A5
JP2022541772A5 JP2022502485A JP2022502485A JP2022541772A5 JP 2022541772 A5 JP2022541772 A5 JP 2022541772A5 JP 2022502485 A JP2022502485 A JP 2022502485A JP 2022502485 A JP2022502485 A JP 2022502485A JP 2022541772 A5 JP2022541772 A5 JP 2022541772A5
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JP
Japan
Prior art keywords
disease
compound
following formula
given
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022502485A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022541772A (ja
JP7618642B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/041876 external-priority patent/WO2021011513A1/en
Publication of JP2022541772A publication Critical patent/JP2022541772A/ja
Publication of JP2022541772A5 publication Critical patent/JP2022541772A5/ja
Application granted granted Critical
Publication of JP7618642B2 publication Critical patent/JP7618642B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022502485A 2019-07-16 2020-07-14 インターロイキンの調節におけるプロドラッグ Active JP7618642B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962874531P 2019-07-16 2019-07-16
US62/874,531 2019-07-16
PCT/US2020/041876 WO2021011513A1 (en) 2019-07-16 2020-07-14 Prodrugs in the modulation of interleukin

Publications (3)

Publication Number Publication Date
JP2022541772A JP2022541772A (ja) 2022-09-27
JP2022541772A5 true JP2022541772A5 (https=) 2023-07-24
JP7618642B2 JP7618642B2 (ja) 2025-01-21

Family

ID=71995065

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022502485A Active JP7618642B2 (ja) 2019-07-16 2020-07-14 インターロイキンの調節におけるプロドラッグ

Country Status (7)

Country Link
US (1) US12528782B2 (https=)
EP (1) EP3999499B1 (https=)
JP (1) JP7618642B2 (https=)
KR (1) KR20220034853A (https=)
CN (1) CN114364665B (https=)
ES (1) ES2991171T3 (https=)
WO (1) WO2021011513A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115466289A (zh) * 2021-06-11 2022-12-13 爱科诺生物医药(香港)有限公司 具有tyk2抑制活性的化合物,包含其的药物组合物,及其应用
CN117362343A (zh) * 2022-07-08 2024-01-09 爱科诺生物医药(香港)有限公司 具有选择性抑制tyk2/jak1活性的化合物,包含其的药物组合物,及其应用
CN118593504B (zh) * 2024-06-03 2025-03-18 北京大学第三医院(北京大学第三临床医学院) 氘可来昔替尼或其盐在制备pvns药物方面的新用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LT3495358T (lt) 2012-11-08 2022-05-25 Bristol-Myers Squibb Company Amidais pakeisti heterocikliniai junginiai, naudingi kaip il-12, il-23 ir (arba) ifn alfa atsako moduliatoriai
TWI582077B (zh) 2013-11-07 2017-05-11 必治妥美雅史谷比公司 作爲IL-12、IL-23及/或IFNα反應調節劑之經烷基-醯胺取代之吡啶化合物
PL3125894T3 (pl) 2014-04-01 2021-02-08 Merck Sharp & Dohme Corp. Proleki inhibitorów odwrotnej transkryptazy hiv
EP3625214B1 (en) 2017-05-16 2022-07-06 Vertex Pharmaceuticals Incorporated Deuterated pyridone amides and prodrugs thereof as modulators of sodium channels
JP7631193B2 (ja) * 2018-10-22 2025-02-18 アルミス インコーポレイテッド Tyk2阻害剤およびその使用

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