JP2022524111A5 - - Google Patents
Info
- Publication number
- JP2022524111A5 JP2022524111A5 JP2021553136A JP2021553136A JP2022524111A5 JP 2022524111 A5 JP2022524111 A5 JP 2022524111A5 JP 2021553136 A JP2021553136 A JP 2021553136A JP 2021553136 A JP2021553136 A JP 2021553136A JP 2022524111 A5 JP2022524111 A5 JP 2022524111A5
- Authority
- JP
- Japan
- Prior art keywords
- compound according
- alkyl
- disease
- compound
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024173169A JP2025016465A (ja) | 2019-03-11 | 2024-10-02 | Ｒａｒ活性化のための合成レチノイド |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1903242.4 | 2019-03-11 | ||
| GBGB1903242.4A GB201903242D0 (en) | 2019-03-11 | 2019-03-11 | Synthetic retinoids for use in rar activation |
| PCT/GB2020/050607 WO2020183173A2 (en) | 2019-03-11 | 2020-03-11 | Synthetic retinoids for use in rar activation |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024173169A Division JP2025016465A (ja) | 2019-03-11 | 2024-10-02 | Ｒａｒ活性化のための合成レチノイド |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022524111A JP2022524111A (ja) | 2022-04-27 |
| JP2022524111A5 true JP2022524111A5 (https=) | 2023-02-14 |
| JP7566765B2 JP7566765B2 (ja) | 2024-10-15 |
Family
ID=66380503
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021553136A Active JP7566765B2 (ja) | 2019-03-11 | 2020-03-11 | Ｒａｒ活性化のための合成レチノイド |
| JP2024173169A Pending JP2025016465A (ja) | 2019-03-11 | 2024-10-02 | Ｒａｒ活性化のための合成レチノイド |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024173169A Pending JP2025016465A (ja) | 2019-03-11 | 2024-10-02 | Ｒａｒ活性化のための合成レチノイド |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US12344587B2 (https=) |
| EP (2) | EP4414355A3 (https=) |
| JP (2) | JP7566765B2 (https=) |
| KR (2) | KR102722925B1 (https=) |
| CN (2) | CN113677667B (https=) |
| AU (1) | AU2020235464B2 (https=) |
| BR (1) | BR112021017045A2 (https=) |
| CA (1) | CA3131108A1 (https=) |
| ES (1) | ES2985674T3 (https=) |
| GB (1) | GB201903242D0 (https=) |
| MX (1) | MX2021011028A (https=) |
| PL (1) | PL3937923T3 (https=) |
| SG (1) | SG11202109075WA (https=) |
| WO (1) | WO2020183173A2 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201903242D0 (en) * | 2019-03-11 | 2019-04-24 | Univ Durham | Synthetic retinoids for use in rar activation |
| CN115974860B (zh) * | 2022-12-15 | 2024-09-24 | 复旦大学附属中山医院 | 维甲酸类化合物及其制备方法和用途、含该化合物的药物组合物 |
| GB2638262A (en) | 2024-02-16 | 2025-08-20 | Univ Durham | Synthetic retinoids for use in RAR activation |
| GB2642547A (en) * | 2024-07-12 | 2026-01-14 | Univ Durham | Compounds for use in senotherapy |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5149705A (en) | 1987-03-13 | 1992-09-22 | Allergan, Inc. | Acetylenes disubstituted with a heteroaromatic group and a tetralin group and having retinoid like activity |
| ATE68486T1 (de) * | 1988-07-28 | 1991-11-15 | Uriach & Cia Sa J | 1-((2-fluorophenyl)(4-fluorophenyl)phenylmethyl - 1h-imidazol. |
| JP2003081834A (ja) * | 2001-09-10 | 2003-03-19 | Shiseido Co Ltd | ざ瘡治療剤、及びざ瘡治療用皮膚外用剤 |
| RU2010136954A (ru) * | 2008-02-06 | 2012-03-20 | Носсира С.А. (Es) | Фенилпрениловые производные морского и синтетического происхождения для лечения нарушения познавательной способности, нейродегенеративных или нервных заболеваний или нарушений |
| CN107176945B (zh) | 2016-03-11 | 2021-06-08 | 中国科学院上海有机化学研究所 | 一种视黄酸类化合物、其制备方法、中间体及应用 |
| WO2017152725A1 (zh) * | 2016-03-11 | 2017-09-14 | 中国科学院上海有机化学研究所 | 一种视黄酸类化合物、其制备方法、中间体及应用 |
| WO2017174999A1 (en) * | 2016-04-07 | 2017-10-12 | High Force Research Limited | Synthetic retinoids for use in rar mediated conditions |
| GB201903242D0 (en) * | 2019-03-11 | 2019-04-24 | Univ Durham | Synthetic retinoids for use in rar activation |
-
2019
- 2019-03-11 GB GBGB1903242.4A patent/GB201903242D0/en not_active Ceased
-
2020
- 2020-03-11 KR KR1020217032599A patent/KR102722925B1/ko active Active
- 2020-03-11 BR BR112021017045A patent/BR112021017045A2/pt unknown
- 2020-03-11 ES ES20715434T patent/ES2985674T3/es active Active
- 2020-03-11 EP EP24184646.8A patent/EP4414355A3/en active Pending
- 2020-03-11 SG SG11202109075WA patent/SG11202109075WA/en unknown
- 2020-03-11 CA CA3131108A patent/CA3131108A1/en active Pending
- 2020-03-11 JP JP2021553136A patent/JP7566765B2/ja active Active
- 2020-03-11 CN CN202080018638.1A patent/CN113677667B/zh active Active
- 2020-03-11 WO PCT/GB2020/050607 patent/WO2020183173A2/en not_active Ceased
- 2020-03-11 EP EP20715434.5A patent/EP3937923B1/en active Active
- 2020-03-11 US US17/435,939 patent/US12344587B2/en active Active
- 2020-03-11 CN CN202510439129.0A patent/CN120271434A/zh active Pending
- 2020-03-11 MX MX2021011028A patent/MX2021011028A/es unknown
- 2020-03-11 PL PL20715434.5T patent/PL3937923T3/pl unknown
- 2020-03-11 KR KR1020247035311A patent/KR20240159014A/ko not_active Ceased
- 2020-03-11 AU AU2020235464A patent/AU2020235464B2/en active Active
-
2024
- 2024-10-02 JP JP2024173169A patent/JP2025016465A/ja active Pending
-
2025
- 2025-06-06 US US19/231,208 patent/US20260000631A1/en active Pending
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