JP2005511625A5 - - Google Patents
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- Publication number
- JP2005511625A5 JP2005511625A5 JP2003544044A JP2003544044A JP2005511625A5 JP 2005511625 A5 JP2005511625 A5 JP 2005511625A5 JP 2003544044 A JP2003544044 A JP 2003544044A JP 2003544044 A JP2003544044 A JP 2003544044A JP 2005511625 A5 JP2005511625 A5 JP 2005511625A5
- Authority
- JP
- Japan
- Prior art keywords
- treatment
- diseases
- compounds
- formula
- present
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 238000011282 treatment Methods 0.000 description 9
- 150000001875 compounds Chemical class 0.000 description 8
- 150000003839 salts Chemical class 0.000 description 5
- 239000012453 solvate Substances 0.000 description 5
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 description 4
- 201000010099 disease Diseases 0.000 description 3
- 239000003814 drug Substances 0.000 description 3
- 208000031295 Animal disease Diseases 0.000 description 2
- 206010036618 Premenstrual syndrome Diseases 0.000 description 2
- 208000028017 Psychotic disease Diseases 0.000 description 2
- 208000006011 Stroke Diseases 0.000 description 2
- 206010008118 cerebral infarction Diseases 0.000 description 2
- 230000002265 prevention Effects 0.000 description 2
- 238000011321 prophylaxis Methods 0.000 description 2
- 239000002464 receptor antagonist Substances 0.000 description 2
- 229940044551 receptor antagonist Drugs 0.000 description 2
- 206010000599 Acromegaly Diseases 0.000 description 1
- 208000024827 Alzheimer disease Diseases 0.000 description 1
- 201000000736 Amenorrhea Diseases 0.000 description 1
- 206010001928 Amenorrhoea Diseases 0.000 description 1
- 208000019901 Anxiety disease Diseases 0.000 description 1
- 241000416162 Astragalus gummifer Species 0.000 description 1
- 201000006474 Brain Ischemia Diseases 0.000 description 1
- 208000014644 Brain disease Diseases 0.000 description 1
- 206010008120 Cerebral ischaemia Diseases 0.000 description 1
- 229920002261 Corn starch Polymers 0.000 description 1
- 208000017701 Endocrine disease Diseases 0.000 description 1
- 206010020772 Hypertension Diseases 0.000 description 1
- 206010058359 Hypogonadism Diseases 0.000 description 1
- 208000019695 Migraine disease Diseases 0.000 description 1
- CZMRCDWAGMRECN-UGDNZRGBSA-N Sucrose Chemical compound O[C@H]1[C@H](O)[C@@H](CO)O[C@@]1(CO)O[C@@H]1[C@H](O)[C@@H](O)[C@H](O)[C@@H](CO)O1 CZMRCDWAGMRECN-UGDNZRGBSA-N 0.000 description 1
- 229930006000 Sucrose Natural products 0.000 description 1
- 229920001615 Tragacanth Polymers 0.000 description 1
- 230000001270 agonistic effect Effects 0.000 description 1
- CJCSPKMFHVPWAR-JTQLQIEISA-N alpha-methyl-L-dopa Chemical compound OC(=O)[C@](N)(C)CC1=CC=C(O)C(O)=C1 CJCSPKMFHVPWAR-JTQLQIEISA-N 0.000 description 1
- 231100000540 amenorrhea Toxicity 0.000 description 1
- 230000036506 anxiety Effects 0.000 description 1
- 210000003169 central nervous system Anatomy 0.000 description 1
- 230000003931 cognitive performance Effects 0.000 description 1
- 239000003086 colorant Substances 0.000 description 1
- 239000008120 corn starch Substances 0.000 description 1
- 208000035475 disorder Diseases 0.000 description 1
- 230000000694 effects Effects 0.000 description 1
- 229960003133 ergot alkaloid Drugs 0.000 description 1
- 230000006651 lactation Effects 0.000 description 1
- 238000004519 manufacturing process Methods 0.000 description 1
- 206010027599 migraine Diseases 0.000 description 1
- 230000001575 pathological effect Effects 0.000 description 1
- 239000008194 pharmaceutical composition Substances 0.000 description 1
- 208000020016 psychiatric disease Diseases 0.000 description 1
- 230000000698 schizophrenic effect Effects 0.000 description 1
- 239000003723 serotonin 1A agonist Substances 0.000 description 1
- 239000005720 sucrose Substances 0.000 description 1
- 208000024891 symptom Diseases 0.000 description 1
- 239000000454 talc Substances 0.000 description 1
- 229910052623 talc Inorganic materials 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01126531 | 2001-11-14 | ||
| PCT/EP2002/011464 WO2003042208A1 (en) | 2001-11-14 | 2002-10-14 | Pyrazole derivatives as psychopharmaceuticals |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005511625A JP2005511625A (ja) | 2005-04-28 |
| JP2005511625A5 true JP2005511625A5 (https=) | 2006-01-05 |
Family
ID=8179188
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003544044A Pending JP2005511625A (ja) | 2001-11-14 | 2002-10-14 | 向精神薬としてのピラゾール誘導体 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20050026927A1 (https=) |
| EP (1) | EP1444229A1 (https=) |
| JP (1) | JP2005511625A (https=) |
| KR (1) | KR20050036882A (https=) |
| CN (1) | CN1585768A (https=) |
| BR (1) | BR0214046A (https=) |
| CA (1) | CA2467081A1 (https=) |
| HU (1) | HUP0402124A2 (https=) |
| MX (1) | MXPA04004443A (https=) |
| PL (1) | PL369674A1 (https=) |
| WO (1) | WO2003042208A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0320320D0 (en) * | 2003-08-29 | 2003-10-01 | Glaxo Group Ltd | Novel compounds |
| GB0321473D0 (en) | 2003-09-12 | 2003-10-15 | Glaxo Group Ltd | Novel compounds |
| US20050282818A1 (en) * | 2004-06-22 | 2005-12-22 | Rigel Pharmaceuticals, Inc. | Ubiquitin ligase inhibitors |
| US9893294B2 (en) | 2010-11-22 | 2018-02-13 | The Regents Of The University Of California | Organic small molecule semiconducting chromophores for use in organic electronic devices |
| US11309499B2 (en) | 2012-02-14 | 2022-04-19 | Next Energy Technologies, Inc. | Electronic devices using organic small molecule semiconducting compounds |
| WO2013123508A2 (en) * | 2012-02-17 | 2013-08-22 | Next Energy Technologies, Inc. | Organic semiconducting compounds for use in organic electronic devices |
| MX365851B (es) * | 2012-08-24 | 2019-06-17 | Treventis Corp | Compuestos de benzofurazano anti-amiloides y metodos. |
| CN104854175A (zh) * | 2012-12-18 | 2015-08-19 | 默克专利股份有限公司 | 包含噻二唑基的聚合物、这种聚合物的制备和它在有机电子器件中的用途 |
| RS58976B1 (sr) * | 2014-02-27 | 2019-08-30 | Treventis Corp | Antiamiloidna jedinjenja koja sadrže benzofuran |
| PT3889145T (pt) | 2015-12-17 | 2024-04-02 | Merck Patent Gmbh | 8-ciano-5-piperidino-quinolinas como antagonistas de tlr7/8 e suas utilizações para tratamento de distúrbios imunitários |
| EP4198031A1 (en) | 2016-08-08 | 2023-06-21 | Merck Patent GmbH | Tlr7/8 antagonists and uses thereof |
| WO2024124439A1 (zh) * | 2022-12-14 | 2024-06-20 | 苏州大学 | 一种抗菌抗肿瘤增效剂及其合成方法与应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6114334A (en) * | 1995-07-13 | 2000-09-05 | Knoll Aktiengesellschaft | Piperazine derivatives as therapeutic agents |
| DE19602505A1 (de) * | 1996-01-25 | 1997-07-31 | Merck Patent Gmbh | 1-(Pyrazol-4-Indol-3-yl)-Piperidine |
-
2002
- 2002-10-14 MX MXPA04004443A patent/MXPA04004443A/es unknown
- 2002-10-14 WO PCT/EP2002/011464 patent/WO2003042208A1/en not_active Ceased
- 2002-10-14 US US10/495,456 patent/US20050026927A1/en not_active Abandoned
- 2002-10-14 EP EP02785208A patent/EP1444229A1/en not_active Withdrawn
- 2002-10-14 PL PL02369674A patent/PL369674A1/xx unknown
- 2002-10-14 BR BR0214046-2A patent/BR0214046A/pt not_active Application Discontinuation
- 2002-10-14 CA CA002467081A patent/CA2467081A1/en not_active Abandoned
- 2002-10-14 HU HU0402124A patent/HUP0402124A2/hu unknown
- 2002-10-14 JP JP2003544044A patent/JP2005511625A/ja active Pending
- 2002-10-14 CN CNA02822566XA patent/CN1585768A/zh active Pending
- 2002-10-14 KR KR1020047006057A patent/KR20050036882A/ko not_active Withdrawn
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