JP2022509206A5 - - Google Patents

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Publication number
JP2022509206A5
JP2022509206A5 JP2021529827A JP2021529827A JP2022509206A5 JP 2022509206 A5 JP2022509206 A5 JP 2022509206A5 JP 2021529827 A JP2021529827 A JP 2021529827A JP 2021529827 A JP2021529827 A JP 2021529827A JP 2022509206 A5 JP2022509206 A5 JP 2022509206A5
Authority
JP
Japan
Prior art keywords
alkyl
pharmaceutical composition
composition according
pain
heterocycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021529827A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022509206A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/063451 external-priority patent/WO2020112905A1/en
Publication of JP2022509206A publication Critical patent/JP2022509206A/ja
Publication of JP2022509206A5 publication Critical patent/JP2022509206A5/ja
Pending legal-status Critical Current

Links

JP2021529827A 2018-11-28 2019-11-26 Magl阻害剤による疾病の治療方法 Pending JP2022509206A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862772554P 2018-11-28 2018-11-28
US62/772,554 2018-11-28
PCT/US2019/063451 WO2020112905A1 (en) 2018-11-28 2019-11-26 Methods of treating disease with magl inhibitors

Publications (2)

Publication Number Publication Date
JP2022509206A JP2022509206A (ja) 2022-01-20
JP2022509206A5 true JP2022509206A5 (https=) 2022-11-28

Family

ID=70851863

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021529827A Pending JP2022509206A (ja) 2018-11-28 2019-11-26 Magl阻害剤による疾病の治療方法

Country Status (15)

Country Link
US (1) US20220031676A1 (https=)
EP (1) EP3886844A4 (https=)
JP (1) JP2022509206A (https=)
KR (1) KR20210097734A (https=)
CN (1) CN113347971A (https=)
AU (1) AU2019389017B2 (https=)
BR (1) BR112020015043A2 (https=)
CA (1) CA3120577A1 (https=)
CL (1) CL2021001363A1 (https=)
IL (1) IL283508A (https=)
MA (1) MA54313A (https=)
MX (1) MX2021006312A (https=)
SG (1) SG11202105320YA (https=)
WO (1) WO2020112905A1 (https=)
ZA (1) ZA202103975B (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10927105B1 (en) 2017-05-23 2021-02-23 Lundbeck La Jolla Research Center, Inc. Pyrazole MAGL inhibitors
EA201992409A1 (ru) 2017-05-23 2020-03-23 Лундбекк Ла-Хойя Рисерч Сентер, Инк. Ингибиторы magl на основе пиразола
BR112023015210A2 (pt) 2021-01-29 2023-11-07 Cedilla Therapeutics Inc Inibidores de cdk2 e métodos de uso dos mesmos
CA3225439A1 (en) 2021-06-26 2022-12-29 Cedilla Therapeutics, Inc. Cdk2 inhibitors and methods of using the same
PE20241304A1 (es) 2021-07-30 2024-06-24 Confo Therapeutics N V Compuestos para el tratamiento del dolor, en particular el dolor neuropatico, y/u otras enfermedades o trastornos que se asocian con at2r y/o senalizacion mediada por at2r
CN118139863A (zh) * 2021-11-02 2024-06-04 H.隆德贝克有限公司 单酰基甘油脂肪酶抑制剂的结晶形式
CA3242372A1 (en) 2021-12-29 2023-07-06 Psy Therapeutics, Inc. Inhibiting monoacylglycerol lipase (magl)

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012524800A (ja) * 2009-04-22 2012-10-18 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ モノアシルグリセロールリパーゼ阻害剤としてのアゼチジニルジアミド
WO2015179559A2 (en) * 2014-05-21 2015-11-26 Abide Therapeutics, Inc. Pyrazole compounds and methods of making and using same
WO2016014975A2 (en) * 2014-07-25 2016-01-28 Northeastern University Urea/carbamates faah magl or dual faah/magl inhibitors and uses thereof
WO2017087858A1 (en) * 2015-11-20 2017-05-26 Abide Therapeutics, Inc. Pyrazole compounds and methods of making and using same
US10519134B2 (en) * 2015-11-20 2019-12-31 Lundbeck La Jolla Research Center, Inc. Pyrazole compounds and methods of making and using same
KR20170128029A (ko) * 2016-05-13 2017-11-22 삼성에스디아이 주식회사 태양전지 전극 형성용 조성물 및 이로부터 제조된 전극
EP3571202B1 (en) * 2017-01-23 2021-06-30 Pfizer Inc. Heterocyclic spiro compounds as magl inhibitors
US10927105B1 (en) * 2017-05-23 2021-02-23 Lundbeck La Jolla Research Center, Inc. Pyrazole MAGL inhibitors
EA201992409A1 (ru) * 2017-05-23 2020-03-23 Лундбекк Ла-Хойя Рисерч Сентер, Инк. Ингибиторы magl на основе пиразола

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