BR112020015043A2 - Métodos para tratar doença com inibidores de magl - Google Patents
Métodos para tratar doença com inibidores de magl Download PDFInfo
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- BR112020015043A2 BR112020015043A2 BR112020015043-6A BR112020015043A BR112020015043A2 BR 112020015043 A2 BR112020015043 A2 BR 112020015043A2 BR 112020015043 A BR112020015043 A BR 112020015043A BR 112020015043 A2 BR112020015043 A2 BR 112020015043A2
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- 238000002560 therapeutic procedure Methods 0.000 description 1
- 125000001113 thiadiazolyl group Chemical group 0.000 description 1
- 125000001984 thiazolidinyl group Chemical group 0.000 description 1
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- 125000005985 thienyl[1,3]dithianyl group Chemical group 0.000 description 1
- LBLYYCQCTBFVLH-UHFFFAOYSA-M toluenesulfonate group Chemical group C=1(C(=CC=CC1)S(=O)(=O)[O-])C LBLYYCQCTBFVLH-UHFFFAOYSA-M 0.000 description 1
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Classifications
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Landscapes
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- Chemical Kinetics & Catalysis (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862772554P | 2018-11-28 | 2018-11-28 | |
| US62/772,554 | 2018-11-28 | ||
| PCT/US2019/063451 WO2020112905A1 (en) | 2018-11-28 | 2019-11-26 | Methods of treating disease with magl inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112020015043A2 true BR112020015043A2 (pt) | 2021-08-31 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112020015043-6A BR112020015043A2 (pt) | 2018-11-28 | 2019-11-26 | Métodos para tratar doença com inibidores de magl |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20220031676A1 (https=) |
| EP (1) | EP3886844A4 (https=) |
| JP (1) | JP2022509206A (https=) |
| KR (1) | KR20210097734A (https=) |
| CN (1) | CN113347971A (https=) |
| AU (1) | AU2019389017B2 (https=) |
| BR (1) | BR112020015043A2 (https=) |
| CA (1) | CA3120577A1 (https=) |
| CL (1) | CL2021001363A1 (https=) |
| IL (1) | IL283508A (https=) |
| MA (1) | MA54313A (https=) |
| MX (1) | MX2021006312A (https=) |
| SG (1) | SG11202105320YA (https=) |
| WO (1) | WO2020112905A1 (https=) |
| ZA (1) | ZA202103975B (https=) |
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| DK3630744T3 (da) | 2017-05-23 | 2023-03-06 | H Lundbeck As | Pyrazol-magl-inhibitorer |
| US10927105B1 (en) | 2017-05-23 | 2021-02-23 | Lundbeck La Jolla Research Center, Inc. | Pyrazole MAGL inhibitors |
| CN117177744A (zh) | 2021-01-29 | 2023-12-05 | 塞迪拉治疗股份有限公司 | Cdk2抑制剂及其使用方法 |
| MX2023015436A (es) | 2021-06-26 | 2024-02-21 | Cedilla Therapeutics Inc | Inhibidores de cdk2 y metodos de uso de los mismos. |
| WO2023006893A1 (en) | 2021-07-30 | 2023-02-02 | Confo Therapeutics N.V. | Compounds for the treatment of pain, in particular neuropathic pain, and/or other diseases or disorders that are associated with at2r and/or at2r mediated signaling |
| CA3234430A1 (en) * | 2021-11-02 | 2023-05-11 | Samuel George ANDREW | Crystalline forms of a monoacylglycerol lipase inhibitor |
| CA3242372A1 (en) | 2021-12-29 | 2023-07-06 | Psy Therapeutics, Inc. | Inhibiting monoacylglycerol lipase (magl) |
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| US8455476B2 (en) * | 2009-04-22 | 2013-06-04 | Janssen Pharmaceutica, Nv | Azetidinyl diamides as monoacylglycerol lipase inhibitors |
| US10093630B2 (en) * | 2014-05-21 | 2018-10-09 | Abide Therapeutics, Inc. | Pyrazole compounds and methods of making and using same |
| US10570146B2 (en) * | 2014-07-25 | 2020-02-25 | Northeastern University | Urea/carbamates FAAH MAGL or dual FAAH/MAGL inhibitors and uses thereof |
| WO2017087858A1 (en) * | 2015-11-20 | 2017-05-26 | Abide Therapeutics, Inc. | Pyrazole compounds and methods of making and using same |
| CN108601769B (zh) * | 2015-11-20 | 2021-09-03 | H.隆德贝克有限公司 | 吡唑化合物及其制备和使用方法 |
| KR20170128029A (ko) * | 2016-05-13 | 2017-11-22 | 삼성에스디아이 주식회사 | 태양전지 전극 형성용 조성물 및 이로부터 제조된 전극 |
| CN110198944A (zh) * | 2017-01-23 | 2019-09-03 | 辉瑞大药厂 | 作为单酰基甘油脂肪酶抑制剂的杂环螺环化合物 |
| DK3630744T3 (da) * | 2017-05-23 | 2023-03-06 | H Lundbeck As | Pyrazol-magl-inhibitorer |
| US10927105B1 (en) * | 2017-05-23 | 2021-02-23 | Lundbeck La Jolla Research Center, Inc. | Pyrazole MAGL inhibitors |
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2019
- 2019-11-26 KR KR1020217019736A patent/KR20210097734A/ko not_active Ceased
- 2019-11-26 CA CA3120577A patent/CA3120577A1/en active Pending
- 2019-11-26 US US17/296,489 patent/US20220031676A1/en not_active Abandoned
- 2019-11-26 MX MX2021006312A patent/MX2021006312A/es unknown
- 2019-11-26 BR BR112020015043-6A patent/BR112020015043A2/pt unknown
- 2019-11-26 MA MA054313A patent/MA54313A/fr unknown
- 2019-11-26 SG SG11202105320YA patent/SG11202105320YA/en unknown
- 2019-11-26 WO PCT/US2019/063451 patent/WO2020112905A1/en not_active Ceased
- 2019-11-26 EP EP19889241.6A patent/EP3886844A4/en not_active Withdrawn
- 2019-11-26 JP JP2021529827A patent/JP2022509206A/ja active Pending
- 2019-11-26 AU AU2019389017A patent/AU2019389017B2/en not_active Expired - Fee Related
- 2019-11-26 CN CN201980090281.5A patent/CN113347971A/zh active Pending
-
2021
- 2021-05-25 CL CL2021001363A patent/CL2021001363A1/es unknown
- 2021-05-27 IL IL283508A patent/IL283508A/en unknown
- 2021-06-09 ZA ZA2021/03975A patent/ZA202103975B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| SG11202105320YA (en) | 2021-06-29 |
| CN113347971A (zh) | 2021-09-03 |
| US20220031676A1 (en) | 2022-02-03 |
| MA54313A (fr) | 2022-03-09 |
| AU2019389017A1 (en) | 2021-06-10 |
| IL283508A (en) | 2021-07-29 |
| WO2020112905A1 (en) | 2020-06-04 |
| CA3120577A1 (en) | 2020-06-04 |
| EP3886844A1 (en) | 2021-10-06 |
| CL2021001363A1 (es) | 2021-11-12 |
| MX2021006312A (es) | 2021-08-11 |
| KR20210097734A (ko) | 2021-08-09 |
| AU2019389017B2 (en) | 2025-01-09 |
| JP2022509206A (ja) | 2022-01-20 |
| ZA202103975B (en) | 2023-11-29 |
| EP3886844A4 (en) | 2022-08-24 |
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