JP2022508642A5 - - Google Patents
Info
- Publication number
- JP2022508642A5 JP2022508642A5 JP2021544096A JP2021544096A JP2022508642A5 JP 2022508642 A5 JP2022508642 A5 JP 2022508642A5 JP 2021544096 A JP2021544096 A JP 2021544096A JP 2021544096 A JP2021544096 A JP 2021544096A JP 2022508642 A5 JP2022508642 A5 JP 2022508642A5
- Authority
- JP
- Japan
- Prior art keywords
- independently
- heteroatoms
- membered
- ring containing
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024179311A JP2025020149A (ja) | 2018-10-05 | 2024-10-11 | モノマーおよびマルチマー抗hbv薬 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862741822P | 2018-10-05 | 2018-10-05 | |
| US62/741,822 | 2018-10-05 | ||
| PCT/US2019/054790 WO2020072955A1 (en) | 2018-10-05 | 2019-10-04 | Monomer and multimeric anti-hbv agents |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024179311A Division JP2025020149A (ja) | 2018-10-05 | 2024-10-11 | モノマーおよびマルチマー抗hbv薬 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022508642A JP2022508642A (ja) | 2022-01-19 |
| JP2022508642A5 true JP2022508642A5 (enExample) | 2023-06-27 |
| JP7648528B2 JP7648528B2 (ja) | 2025-03-18 |
Family
ID=70055532
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021544096A Active JP7648528B2 (ja) | 2018-10-05 | 2019-10-04 | モノマーおよびマルチマー抗hbv薬 |
| JP2024179311A Pending JP2025020149A (ja) | 2018-10-05 | 2024-10-11 | モノマーおよびマルチマー抗hbv薬 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024179311A Pending JP2025020149A (ja) | 2018-10-05 | 2024-10-11 | モノマーおよびマルチマー抗hbv薬 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20230056135A1 (enExample) |
| EP (1) | EP3860991A4 (enExample) |
| JP (2) | JP7648528B2 (enExample) |
| KR (2) | KR20210072015A (enExample) |
| CN (2) | CN122404196A (enExample) |
| AU (1) | AU2019355218B2 (enExample) |
| BR (1) | BR112021006403A2 (enExample) |
| CA (1) | CA3113109A1 (enExample) |
| IL (2) | IL328538A (enExample) |
| MX (1) | MX2021003150A (enExample) |
| PH (1) | PH12021550632A1 (enExample) |
| SG (1) | SG11202102661UA (enExample) |
| WO (1) | WO2020072955A1 (enExample) |
| ZA (1) | ZA202102589B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL328538A (en) * | 2018-10-05 | 2026-07-01 | Univ Emory | Monomeric and multimeric hepatitis B antivirals |
| IL286902B2 (en) | 2019-04-03 | 2025-03-01 | Aligos Therapeutics Inc | Pyrrole compounds |
| KR20230021121A (ko) * | 2020-06-05 | 2023-02-13 | 파티오스 테라퓨틱스 리미티드 | Gpr65의 조절제로서 n-페닐아미노카보닐 피리디노-, 피리미디노 및 벤조-트로판 |
| WO2022156758A1 (zh) * | 2021-01-22 | 2022-07-28 | 广东东阳光药业有限公司 | 新型酰胺吡咯类化合物及其在药物中的用途 |
| WO2023174351A1 (zh) * | 2022-03-17 | 2023-09-21 | 成都微芯药业有限公司 | 吡咯酰胺类化合物及其制备方法和用途 |
| CN116120219A (zh) * | 2022-12-27 | 2023-05-16 | 吉斯凯(苏州)制药有限公司 | 一种多取代吡咯类化合物及其制备方法和在制备hbv衣壳蛋白抑制剂中的应用 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AUPP913999A0 (en) * | 1999-03-12 | 1999-04-01 | Biota Scientific Management Pty Ltd | Novel chemical compounds and their use |
| US20060100233A1 (en) * | 2002-07-25 | 2006-05-11 | Manuela Villa | Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them |
| US9242981B2 (en) * | 2010-09-16 | 2016-01-26 | Merck Sharp & Dohme Corp. | Fused pyrazole derivatives as novel ERK inhibitors |
| WO2013006394A1 (en) * | 2011-07-01 | 2013-01-10 | Institute For Hepatitis And Virus Research | Sulfamoylbenzamide derivatives as antiviral agents against hbv infection |
| CA2881057C (en) * | 2012-08-28 | 2020-10-27 | Janssen Sciences Ireland Uc | Sulfamoyl-arylamides and the use thereof as medicaments for the treatment of hepatitis b |
| HK1215030A1 (zh) * | 2012-11-09 | 2016-08-12 | Indiana University Research And Technology Corporation | 用於hbv組裝效應劑的替代用途 |
| HK1217649A1 (zh) * | 2012-12-27 | 2017-01-20 | 德雷克塞尔大学 | 針對hbv感染的新型抗病毒劑 |
| WO2015011281A1 (en) * | 2013-07-25 | 2015-01-29 | Janssen R&D Ireland | Glyoxamide substituted pyrrolamide derivatives and the use thereof as medicaments for the treatment of hepatitis b |
| EP3150600B1 (en) * | 2014-05-30 | 2018-06-27 | Qilu Pharmaceutical Co., Ltd. | Dihydropyrimido loop derivative as hbv inhibitor |
| WO2016109689A2 (en) * | 2014-12-30 | 2016-07-07 | Novira Therapeutics, Inc. | Derivatives and methods of treating hepatitis b infections |
| CN106317055A (zh) * | 2015-07-02 | 2017-01-11 | 中国科学院上海药物研究所 | 一类具有激酶抑制活性的化合物、制备方法和用途 |
| BR112018068177B1 (pt) * | 2016-03-09 | 2024-02-27 | Emory University | Composto, uso do composto e composição para eliminação do vírus da hepatite b com agentes antivirais |
| JOP20190024A1 (ar) | 2016-08-26 | 2019-02-19 | Gilead Sciences Inc | مركبات بيروليزين بها استبدال واستخداماتها |
| WO2019185016A1 (zh) | 2018-03-30 | 2019-10-03 | 正大天晴药业集团股份有限公司 | 含有n杂五元环的衣壳蛋白装配抑制剂、其药物组合物和用途 |
| WO2019241292A1 (en) | 2018-06-11 | 2019-12-19 | VenatoRx Pharmaceuticals, Inc. | Hepatitis b capsid assembly modulators |
| WO2020001592A1 (zh) * | 2018-06-28 | 2020-01-02 | 河南天晟泰丰医药科技有限公司 | 二氢嘧啶衍生物及其用途 |
| IL328538A (en) * | 2018-10-05 | 2026-07-01 | Univ Emory | Monomeric and multimeric hepatitis B antivirals |
-
2019
- 2019-10-04 IL IL328538A patent/IL328538A/en unknown
- 2019-10-04 SG SG11202102661UA patent/SG11202102661UA/en unknown
- 2019-10-04 AU AU2019355218A patent/AU2019355218B2/en active Active
- 2019-10-04 KR KR1020217012512A patent/KR20210072015A/ko active Pending
- 2019-10-04 EP EP19868793.1A patent/EP3860991A4/en active Pending
- 2019-10-04 CN CN202511985696.2A patent/CN122404196A/zh active Pending
- 2019-10-04 BR BR112021006403A patent/BR112021006403A2/pt unknown
- 2019-10-04 JP JP2021544096A patent/JP7648528B2/ja active Active
- 2019-10-04 KR KR1020257021884A patent/KR20250107952A/ko active Pending
- 2019-10-04 CN CN201980081049.5A patent/CN113166115A/zh active Pending
- 2019-10-04 CA CA3113109A patent/CA3113109A1/en active Pending
- 2019-10-04 US US17/281,940 patent/US20230056135A1/en active Pending
- 2019-10-04 MX MX2021003150A patent/MX2021003150A/es unknown
- 2019-10-04 WO PCT/US2019/054790 patent/WO2020072955A1/en not_active Ceased
-
2021
- 2021-03-19 PH PH12021550632A patent/PH12021550632A1/en unknown
- 2021-03-21 IL IL281698A patent/IL281698A/en unknown
- 2021-04-19 ZA ZA2021/02589A patent/ZA202102589B/en unknown
-
2024
- 2024-10-11 JP JP2024179311A patent/JP2025020149A/ja active Pending
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