JP2022504780A5 - - Google Patents
Info
- Publication number
- JP2022504780A5 JP2022504780A5 JP2021520147A JP2021520147A JP2022504780A5 JP 2022504780 A5 JP2022504780 A5 JP 2022504780A5 JP 2021520147 A JP2021520147 A JP 2021520147A JP 2021520147 A JP2021520147 A JP 2021520147A JP 2022504780 A5 JP2022504780 A5 JP 2022504780A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- iii
- compound
- amine
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2018/110852 | 2018-10-18 | ||
| CN2018110852 | 2018-10-18 | ||
| PCT/EP2019/078208 WO2020079145A1 (en) | 2018-10-18 | 2019-10-17 | Scalable synthesis of optically active 1-cyclopropylalkyl-1-amines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022504780A JP2022504780A (ja) | 2022-01-13 |
| JP2022504780A5 true JP2022504780A5 (https=) | 2022-10-20 |
Family
ID=68290245
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021520147A Pending JP2022504780A (ja) | 2018-10-18 | 2019-10-17 | 光学活性１－シクロプロピルアルキル－１－アミンのスケーラブルな合成 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20210395185A1 (https=) |
| EP (1) | EP3867224A1 (https=) |
| JP (1) | JP2022504780A (https=) |
| CN (1) | CN112930336A (https=) |
| WO (1) | WO2020079145A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112552184B (zh) * | 2020-12-18 | 2022-05-10 | 诚达药业股份有限公司 | 一种含环丙基手性胺盐酸盐的合成方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4287703B2 (ja) * | 2003-06-11 | 2009-07-01 | セントラル硝子株式会社 | 光学活性１−アルキル置換−２，２，２−トリフルオロエチルアミンの製造方法 |
| EP1778620A1 (en) * | 2004-07-22 | 2007-05-02 | DSMIP Assets B.V. | Process for the preparation of a diastereomerically enriched compound |
| GB0510546D0 (en) * | 2005-05-24 | 2005-06-29 | Astrazeneca Ab | New process |
| AU2008335761B2 (en) | 2007-12-13 | 2014-04-24 | Merck Sharp & Dohme Corp. | Inhibitors of janus kinases |
| BRPI0916544A2 (pt) * | 2008-07-23 | 2015-08-04 | Dsm Ip Assets Bv | Rotas de síntese para 2(s), 4(s), 5(s), 7(s) - 2, 7 dialquil-4-hidroxi-2-amino-8-aril-octanoil amida |
| WO2011076744A1 (en) * | 2009-12-21 | 2011-06-30 | Novartis Ag | Disubstituted heteroaryl-fused pyridines |
| NZ723530A (en) | 2014-04-14 | 2023-05-26 | Boehringer Ingelheim Int | Compounds as modulators of ror gamma |
| EP3356366B1 (en) | 2015-10-01 | 2019-08-28 | Boehringer Ingelheim International GmbH | Pteridine derivatives as modulators of ror gamma |
| US11358967B2 (en) | 2016-01-20 | 2022-06-14 | Boehringer Ingelheim International Gmbh | Substituted pyrazino[2,3-b]pyrazines and pyrazino[2,3-c]pyridazines as modulators of ROR gamma |
-
2019
- 2019-10-17 JP JP2021520147A patent/JP2022504780A/ja active Pending
- 2019-10-17 US US17/285,564 patent/US20210395185A1/en not_active Abandoned
- 2019-10-17 WO PCT/EP2019/078208 patent/WO2020079145A1/en not_active Ceased
- 2019-10-17 CN CN201980069158.5A patent/CN112930336A/zh active Pending
- 2019-10-17 EP EP19790192.9A patent/EP3867224A1/en not_active Withdrawn
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