JP2022502495A5 - - Google Patents

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Publication number
JP2022502495A5
JP2022502495A5 JP2021540390A JP2021540390A JP2022502495A5 JP 2022502495 A5 JP2022502495 A5 JP 2022502495A5 JP 2021540390 A JP2021540390 A JP 2021540390A JP 2021540390 A JP2021540390 A JP 2021540390A JP 2022502495 A5 JP2022502495 A5 JP 2022502495A5
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JP
Japan
Prior art keywords
amino acid
positions
seq
acid sequence
egfr
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021540390A
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English (en)
Japanese (ja)
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JP2022502495A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/052784 external-priority patent/WO2020068867A1/en
Publication of JP2022502495A publication Critical patent/JP2022502495A/ja
Publication of JP2022502495A5 publication Critical patent/JP2022502495A5/ja
Pending legal-status Critical Current

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JP2021540390A 2018-09-25 2019-09-24 チロシンキナーゼ阻害剤としてのキナゾリン誘導体、組成物、それらの作製方法、およびそれらの使用 Pending JP2022502495A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862736293P 2018-09-25 2018-09-25
US62/736,293 2018-09-25
US201962903592P 2019-09-20 2019-09-20
US62/903,592 2019-09-20
PCT/US2019/052784 WO2020068867A1 (en) 2018-09-25 2019-09-24 Quinazoline derivatives as tyrosine kinase inhibitor, compositions, methods of making them and their use

Publications (2)

Publication Number Publication Date
JP2022502495A JP2022502495A (ja) 2022-01-11
JP2022502495A5 true JP2022502495A5 (https=) 2022-10-03

Family

ID=68165800

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021540390A Pending JP2022502495A (ja) 2018-09-25 2019-09-24 チロシンキナーゼ阻害剤としてのキナゾリン誘導体、組成物、それらの作製方法、およびそれらの使用

Country Status (12)

Country Link
US (2) US11034672B1 (https=)
EP (1) EP3856726A1 (https=)
JP (1) JP2022502495A (https=)
KR (1) KR20210137422A (https=)
CN (1) CN113382986A (https=)
AU (1) AU2019346550A1 (https=)
BR (1) BR112021005513A2 (https=)
CA (1) CA3113241A1 (https=)
IL (1) IL281805A (https=)
MX (1) MX2021003517A (https=)
SG (1) SG11202102981SA (https=)
WO (1) WO2020068867A1 (https=)

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CN116655599B (zh) * 2023-05-17 2025-07-29 江南大学 一类egfr别构抑制剂的合成及其用途
EP4724436A1 (en) * 2023-06-12 2026-04-15 Remix Therapeutics Inc. Compounds and methods for modulating splicing
WO2025096300A1 (en) * 2023-10-30 2025-05-08 Eli Lilly And Company Novel methods for the preparation of 3-azabicylco[3.1,0]hexane-6-carboxamide derivatives
CN118084767B (zh) * 2024-04-02 2025-06-17 康龙化成手性医药技术(宁波)有限公司 一种外型-6-氟甲基-3-氮杂双环[3,1,0]己烷盐酸盐及其衍生物的合成方法
CN118652239A (zh) * 2024-05-29 2024-09-17 江南大学 一类egfr别构抑制剂的合成及其用途

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