JP2021534158A5 - - Google Patents

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Publication number
JP2021534158A5
JP2021534158A5 JP2021507737A JP2021507737A JP2021534158A5 JP 2021534158 A5 JP2021534158 A5 JP 2021534158A5 JP 2021507737 A JP2021507737 A JP 2021507737A JP 2021507737 A JP2021507737 A JP 2021507737A JP 2021534158 A5 JP2021534158 A5 JP 2021534158A5
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cancer
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substituted
pharmaceutical composition
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JP2021507737A
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Japanese (ja)
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JP2021534158A (ja
JP7433291B2 (ja
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Priority claimed from PCT/US2019/046592 external-priority patent/WO2020037092A1/en
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JP2021507737A 2018-08-16 2019-08-15 イミダゾ[4,5-c]キノリン誘導体のNLRP3モジュレーター Active JP7433291B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862764900P 2018-08-16 2018-08-16
US62/764,900 2018-08-16
PCT/US2019/046592 WO2020037092A1 (en) 2018-08-16 2019-08-15 Imidazo[4,5-c]quinoline derived nlrp3-modulators

Publications (3)

Publication Number Publication Date
JP2021534158A JP2021534158A (ja) 2021-12-09
JP2021534158A5 true JP2021534158A5 (https=) 2022-08-01
JP7433291B2 JP7433291B2 (ja) 2024-02-19

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JP2021507737A Active JP7433291B2 (ja) 2018-08-16 2019-08-15 イミダゾ[4,5-c]キノリン誘導体のNLRP3モジュレーター

Country Status (7)

Country Link
US (1) US12024513B2 (https=)
EP (1) EP3837015B1 (https=)
JP (1) JP7433291B2 (https=)
KR (1) KR102817037B1 (https=)
CN (1) CN112996567A (https=)
ES (1) ES2974964T3 (https=)
WO (1) WO2020037092A1 (https=)

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WO2020037094A1 (en) 2018-08-16 2020-02-20 Innate Tumor Immunity, Inc. Substitued 4-amino-1h-imidazo[4,5-c]quinoline compounds and improved methods for their preparation
US20210269434A1 (en) * 2020-01-10 2021-09-02 Incyte Corporation Tricyclic compounds as inhibitors of kras
WO2021150613A1 (en) 2020-01-20 2021-07-29 Incyte Corporation Spiro compounds as inhibitors of kras
US11739102B2 (en) 2020-05-13 2023-08-29 Incyte Corporation Fused pyrimidine compounds as KRAS inhibitors
US11999752B2 (en) 2020-08-28 2024-06-04 Incyte Corporation Vinyl imidazole compounds as inhibitors of KRAS
US11767320B2 (en) 2020-10-02 2023-09-26 Incyte Corporation Bicyclic dione compounds as inhibitors of KRAS
WO2022204112A1 (en) 2021-03-22 2022-09-29 Incyte Corporation Imidazole and triazole kras inhibitors
MX2024000357A (es) 2021-07-07 2024-02-12 Incyte Corp Compuestos triciclicos como inhibidores de homologo de oncogen viral de sarcoma de rata kirsten (kras).
WO2023287896A1 (en) 2021-07-14 2023-01-19 Incyte Corporation Tricyclic compounds as inhibitors of kras
US12441742B2 (en) 2021-08-31 2025-10-14 Incyte Corporation Naphthyridine compounds as inhibitors of KRAS
WO2023049697A1 (en) 2021-09-21 2023-03-30 Incyte Corporation Hetero-tricyclic compounds as inhibitors of kras
CA3234375A1 (en) 2021-10-01 2023-04-06 Incyte Corporation Pyrazoloquinoline kras inhibitors
CA3235146A1 (en) 2021-10-14 2023-04-20 Incyte Corporation Quinoline compounds as inhibitors of kras

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