JP2021529805A5 - - Google Patents

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Publication number
JP2021529805A5
JP2021529805A5 JP2021500178A JP2021500178A JP2021529805A5 JP 2021529805 A5 JP2021529805 A5 JP 2021529805A5 JP 2021500178 A JP2021500178 A JP 2021500178A JP 2021500178 A JP2021500178 A JP 2021500178A JP 2021529805 A5 JP2021529805 A5 JP 2021529805A5
Authority
JP
Japan
Prior art keywords
ivosidenib
powder
ray diffraction
diffraction pattern
dsc
Prior art date
Application number
JP2021500178A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021529805A (ja
JPWO2020010058A5 (https=
JP7621242B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/040257 external-priority patent/WO2020010058A1/en
Publication of JP2021529805A publication Critical patent/JP2021529805A/ja
Publication of JPWO2020010058A5 publication Critical patent/JPWO2020010058A5/ja
Publication of JP2021529805A5 publication Critical patent/JP2021529805A5/ja
Priority to JP2024131926A priority Critical patent/JP2024150784A/ja
Application granted granted Critical
Publication of JP7621242B2 publication Critical patent/JP7621242B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021500178A 2018-07-06 2019-07-02 イボシデニブ形態および医薬組成物 Active JP7621242B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024131926A JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862694596P 2018-07-06 2018-07-06
US62/694,596 2018-07-06
PCT/US2019/040257 WO2020010058A1 (en) 2018-07-06 2019-07-02 Ivosidenib forms and pharmaceutical compositions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024131926A Division JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Publications (4)

Publication Number Publication Date
JP2021529805A JP2021529805A (ja) 2021-11-04
JPWO2020010058A5 JPWO2020010058A5 (https=) 2022-07-12
JP2021529805A5 true JP2021529805A5 (https=) 2022-07-12
JP7621242B2 JP7621242B2 (ja) 2025-01-24

Family

ID=69059942

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021500178A Active JP7621242B2 (ja) 2018-07-06 2019-07-02 イボシデニブ形態および医薬組成物
JP2024131926A Withdrawn JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024131926A Withdrawn JP2024150784A (ja) 2018-07-06 2024-08-08 イボシデニブ形態および医薬組成物

Country Status (18)

Country Link
US (1) US12264148B2 (https=)
EP (2) EP3817744A4 (https=)
JP (2) JP7621242B2 (https=)
KR (2) KR102919157B1 (https=)
CN (1) CN112367995A (https=)
AU (2) AU2019299352B2 (https=)
BR (1) BR112021000156A2 (https=)
CA (1) CA3103498A1 (https=)
EA (1) EA202190217A1 (https=)
IL (2) IL315423B1 (https=)
MA (1) MA53099A (https=)
MX (2) MX2021000068A (https=)
PH (1) PH12021550017A1 (https=)
SG (1) SG11202012763TA (https=)
TW (2) TWI902665B (https=)
UA (1) UA129800C2 (https=)
WO (1) WO2020010058A1 (https=)
ZA (1) ZA202008034B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT4010331T (pt) 2019-08-08 2024-01-08 Servier Lab Um método de preparação do ivosidenib e de um seu intermediário
GB201912411D0 (en) * 2019-08-29 2019-10-16 Johnson Matthey Plc Crystalline forms of ivosidenib
AR133410A1 (es) 2023-08-01 2025-09-24 Servier Lab Cocristal de un inhibidor de idh1, proceso de preparación del mismo, composiciones farmacéuticas del mismo, y métodos de tratamiento que implican el mismo

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010223919B2 (en) 2009-03-13 2016-03-31 Les Laboratoires Servier Methods and compositions for cell-proliferation-related disorders
EP3561077B1 (en) 2009-10-21 2022-12-21 Les Laboratoires Servier Methods for cell-proliferation-related disorders
RU2013144975A (ru) * 2011-04-08 2015-05-20 Пфайзер Инк. Кристаллические и некристаллические формы тофацитиниба и фармацевтическая композиция, содержащая тофацитиниб, и усилитель проникновения
US9474779B2 (en) 2012-01-19 2016-10-25 Agios Pharmaceuticals, Inc. Therapeutically active compositions and their methods of use
UY35006A (es) * 2012-09-06 2014-03-31 Bayer Healthcare Llc Composición farmacéutica recubierta que contiene regorafenib
BR122023021436A2 (pt) * 2014-03-14 2023-12-12 Les Laboratoires Servier Formas cristalinas e composição farmacêutica de compostos terapeuticamente ativos
KR20240010105A (ko) * 2014-03-14 2024-01-23 아지오스 파마슈티컬스 아이엔씨. 치료적으로 활성인 화합물의 약제학적 조성물
PT3362066T (pt) 2015-10-15 2021-11-16 Celgene Corp Terapia de combinação para tratar malignidades
ES2912909T3 (es) * 2016-02-26 2022-05-30 Celgene Corp Enasidenib para su uso en el tratamiento de la leucemia mieloide aguda recidivante o refractaria
WO2019104318A1 (en) 2017-11-27 2019-05-31 Teva Pharmaceuticals Usa, Inc. Solid state forms of ivosidenib

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