JP2021512898A5 - - Google Patents

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Publication number
JP2021512898A5
JP2021512898A5 JP2020542580A JP2020542580A JP2021512898A5 JP 2021512898 A5 JP2021512898 A5 JP 2021512898A5 JP 2020542580 A JP2020542580 A JP 2020542580A JP 2020542580 A JP2020542580 A JP 2020542580A JP 2021512898 A5 JP2021512898 A5 JP 2021512898A5
Authority
JP
Japan
Prior art keywords
compound
alkyl
salt according
formula
group
Prior art date
Application number
JP2020542580A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021512898A (ja
JPWO2019157417A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/017422 external-priority patent/WO2019157417A1/en
Publication of JP2021512898A publication Critical patent/JP2021512898A/ja
Publication of JPWO2019157417A5 publication Critical patent/JPWO2019157417A5/ja
Publication of JP2021512898A5 publication Critical patent/JP2021512898A5/ja
Pending legal-status Critical Current

Links

JP2020542580A 2018-02-09 2019-02-11 複素環p2y14受容体拮抗薬 Pending JP2021512898A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862628699P 2018-02-09 2018-02-09
US62/628,699 2018-02-09
PCT/US2019/017422 WO2019157417A1 (en) 2018-02-09 2019-02-11 Heterocyclic p2y14 receptor antagonists

Publications (3)

Publication Number Publication Date
JP2021512898A JP2021512898A (ja) 2021-05-20
JPWO2019157417A5 JPWO2019157417A5 (https=) 2022-02-24
JP2021512898A5 true JP2021512898A5 (https=) 2022-02-24

Family

ID=65529813

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020542580A Pending JP2021512898A (ja) 2018-02-09 2019-02-11 複素環p2y14受容体拮抗薬

Country Status (7)

Country Link
US (1) US11584736B2 (https=)
EP (1) EP3749651A1 (https=)
JP (1) JP2021512898A (https=)
CN (1) CN111868036A (https=)
AU (1) AU2019218256A1 (https=)
CA (1) CA3090788A1 (https=)
WO (1) WO2019157417A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11708346B2 (en) 2019-07-23 2023-07-25 Saint Louis University Treatment and prevention of neuropathic pain with P2Y14 antagonists
WO2022155037A1 (en) * 2021-01-18 2022-07-21 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Heterocyclic p2y 14 receptor antagonists
CN116444482B (zh) * 2023-06-14 2023-09-22 中国药科大学 噻吩-2-羧酸衍生物、其制备方法及医药用途

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4377586A (en) 1981-04-30 1983-03-22 The Upjohn Company Diuretic 2,6-diaryl-4-pyridine carboxylic acids
GB0507200D0 (en) 2005-04-08 2005-05-18 Smithkline Beecham Corp Chemical compounds
CA2706632A1 (en) * 2007-12-04 2009-06-11 Merck Frosst Canada Ltd. Substituted 2-naphthoic acids as antagonists of gpr105 activity
US8580961B2 (en) 2010-12-13 2013-11-12 National Tsing Hua University 2-phenyl-6-azolylpyridine-based ligand and group VIII transition metal complex
US9290453B2 (en) 2010-12-23 2016-03-22 Merck Sharp & Dohme Corp. Quinolines and aza-quinolines as CRTH2 receptor modulators
DE112011105485T5 (de) 2011-08-01 2014-06-12 Mitsubishi Electric Corporation Steuervorrichtung und Steuerverfahren für eine Spritzgussmaschine
EP2774919A1 (en) 2013-03-06 2014-09-10 Pharmeste S.R.L. In Liquidazione Novel sulfonamide TRPA1 receptor antagonists
PE20181366A1 (es) * 2015-08-03 2018-08-27 Bristol Myers Squibb Co Compuestos heterociclicos utiles como moduladores de factor de necrosis tumoral (tnf) alfa
US10683277B2 (en) 2015-09-25 2020-06-16 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Triazole derivatives as P2Y14 receptor antagonists
US11008340B2 (en) 2015-11-20 2021-05-18 Vitae Pharmaceuticals, Llc Modulators of ROR-gamma
US11938114B2 (en) 2017-03-10 2024-03-26 Rutgers, The State University Of New Jersey Bacterial efflux pump inhibitors
CN109096177A (zh) 2018-08-31 2018-12-28 中国药科大学 3-酰胺基苯甲酸衍生物、其制备方法及医药用途

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