JP2020514361A5 - - Google Patents
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- JP2020514361A5 JP2020514361A5 JP2019550659A JP2019550659A JP2020514361A5 JP 2020514361 A5 JP2020514361 A5 JP 2020514361A5 JP 2019550659 A JP2019550659 A JP 2019550659A JP 2019550659 A JP2019550659 A JP 2019550659A JP 2020514361 A5 JP2020514361 A5 JP 2020514361A5
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2022200392A JP2023051962A (ja) | 2017-03-16 | 2022-12-15 | ９，１０，１１，１２－テトラヒドロ－８ｈ－［１，４］ジアゼピノ［５’，６’：４，５］チエノ［３，２－ｆ］キノリン－８－オン化合物およびその使用 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762472027P | 2017-03-16 | 2017-03-16 | |
| US62/472,027 | 2017-03-16 | ||
| PCT/US2018/022548 WO2018170204A1 (en) | 2017-03-16 | 2018-03-15 | 9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one compounds and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022200392A Division JP2023051962A (ja) | 2017-03-16 | 2022-12-15 | ９，１０，１１，１２－テトラヒドロ－８ｈ－［１，４］ジアゼピノ［５’，６’：４，５］チエノ［３，２－ｆ］キノリン－８－オン化合物およびその使用 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2020514361A JP2020514361A (ja) | 2020-05-21 |
| JP2020514361A5 true JP2020514361A5 (https=) | 2021-04-22 |
Family
ID=63522566
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019550659A Pending JP2020514361A (ja) | 2017-03-16 | 2018-03-15 | ９，１０，１１，１２−テトラヒドロ−８ｈ−［１，４］ジアゼピノ［５’，６’：４，５］チエノ［３，２−ｆ］キノリン−８−オン化合物およびその使用 |
| JP2022200392A Pending JP2023051962A (ja) | 2017-03-16 | 2022-12-15 | ９，１０，１１，１２－テトラヒドロ－８ｈ－［１，４］ジアゼピノ［５’，６’：４，５］チエノ［３，２－ｆ］キノリン－８－オン化合物およびその使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022200392A Pending JP2023051962A (ja) | 2017-03-16 | 2022-12-15 | ９，１０，１１，１２－テトラヒドロ－８ｈ－［１，４］ジアゼピノ［５’，６’：４，５］チエノ［３，２－ｆ］キノリン－８－オン化合物およびその使用 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US11098057B2 (https=) |
| EP (1) | EP3596084A4 (https=) |
| JP (2) | JP2020514361A (https=) |
| WO (1) | WO2018170204A1 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RS62017B1 (sr) | 2014-09-17 | 2021-07-30 | Celgene Car Llc | Mk2 inhibitori i njihova upotreba |
| US11230551B2 (en) | 2017-03-16 | 2022-01-25 | Celgene Car Llc | Deuterated analogs of MK2 inhibitors and uses thereof |
| JP7282039B2 (ja) | 2017-03-16 | 2023-05-26 | セルジーン シーエーアール エルエルシー | Ｍｋ２阻害剤、その合成、およびそれに至るまでの中間体 |
| JP7200120B2 (ja) | 2017-03-16 | 2023-01-06 | セルジーン シーエーアール エルエルシー | Ｍｋ２阻害剤として有用なヘテロアリール化合物 |
| WO2018170204A1 (en) | 2017-03-16 | 2018-09-20 | Celgene Car Llc | 9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one compounds and uses thereof |
| US10882867B2 (en) | 2017-03-16 | 2021-01-05 | Celgene Car Llc | Forms and compositions of a MK2 inhibitor |
| CN114364681A (zh) * | 2019-05-17 | 2022-04-15 | 西建卡尔有限责任公司 | 治疗mk2介导的病症的方法 |
| KR20230142529A (ko) | 2021-02-01 | 2023-10-11 | 셀진 코포레이션 | Mk2 억제제, 이의 합성, 및 이의 중간체 |
| TW202328141A (zh) * | 2021-08-27 | 2023-07-16 | 大陸商瑞石生物醫藥有限公司 | 喹啉并呋喃衍生物及其用途 |
| CN119998296A (zh) * | 2022-08-31 | 2025-05-13 | 国立大学法人京都大学 | 化合物、内质网应激抑制剂、药物、眼科用药、滴眼剂、组合物、化合物的制备方法 |
| CN115925718A (zh) * | 2022-12-27 | 2023-04-07 | 瑞石生物医药有限公司 | 一种四环内酰胺衍生物及其用途 |
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| CN1087725C (zh) | 1994-03-25 | 2002-07-17 | 同位素技术有限公司 | 用氘代方法增强药物效果 |
| CN1747949A (zh) | 2002-12-20 | 2006-03-15 | 法马西亚公司 | 无环吡唑化合物 |
| WO2005105814A1 (en) | 2004-04-28 | 2005-11-10 | Incyte Corporation | Tetracyclic inhibitors of janus kinases |
| CN101687869A (zh) | 2007-07-16 | 2010-03-31 | 诺瓦提斯公司 | 作为mk2抑制剂的四环内酰胺衍生物 |
| EP2201737A2 (en) * | 2007-10-20 | 2010-06-30 | Penango, Inc. | Methods and systems for indicating trustworthiness of secure communications |
| WO2011153553A2 (en) | 2010-06-04 | 2011-12-08 | The Regents Of The University Of California | Methods and compositions for kinase inhibition |
| HK1210696A1 (en) * | 2012-07-11 | 2016-05-06 | Nimbus Iris, Inc. | Irak inhibitors and uses thereof |
| JP2016518316A (ja) * | 2013-03-15 | 2016-06-23 | セルジーン アビロミクス リサーチ， インコーポレイテッド | Ｍｋ２阻害剤およびそれらの使用 |
| RS62017B1 (sr) | 2014-09-17 | 2021-07-30 | Celgene Car Llc | Mk2 inhibitori i njihova upotreba |
| JP7282039B2 (ja) * | 2017-03-16 | 2023-05-26 | セルジーン シーエーアール エルエルシー | Ｍｋ２阻害剤、その合成、およびそれに至るまでの中間体 |
| WO2018170204A1 (en) | 2017-03-16 | 2018-09-20 | Celgene Car Llc | 9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one compounds and uses thereof |
| JP7200120B2 (ja) * | 2017-03-16 | 2023-01-06 | セルジーン シーエーアール エルエルシー | Ｍｋ２阻害剤として有用なヘテロアリール化合物 |
| US11230551B2 (en) | 2017-03-16 | 2022-01-25 | Celgene Car Llc | Deuterated analogs of MK2 inhibitors and uses thereof |
| US10882867B2 (en) | 2017-03-16 | 2021-01-05 | Celgene Car Llc | Forms and compositions of a MK2 inhibitor |
-
2018
- 2018-03-15 WO PCT/US2018/022548 patent/WO2018170204A1/en not_active Ceased
- 2018-03-15 JP JP2019550659A patent/JP2020514361A/ja active Pending
- 2018-03-15 EP EP18766809.0A patent/EP3596084A4/en not_active Withdrawn
- 2018-03-15 US US16/494,722 patent/US11098057B2/en active Active
-
2022
- 2022-12-15 JP JP2022200392A patent/JP2023051962A/ja active Pending
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