JP2020511467A5 - - Google Patents

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Publication number
JP2020511467A5
JP2020511467A5 JP2019550651A JP2019550651A JP2020511467A5 JP 2020511467 A5 JP2020511467 A5 JP 2020511467A5 JP 2019550651 A JP2019550651 A JP 2019550651A JP 2019550651 A JP2019550651 A JP 2019550651A JP 2020511467 A5 JP2020511467 A5 JP 2020511467A5
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JP
Japan
Prior art keywords
cancer
crystal form
powder
compound
ray diffraction
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Pending
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JP2019550651A
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English (en)
Japanese (ja)
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JP2020511467A (ja
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Priority claimed from PCT/US2018/023127 external-priority patent/WO2018175311A1/en
Publication of JP2020511467A publication Critical patent/JP2020511467A/ja
Publication of JP2020511467A5 publication Critical patent/JP2020511467A5/ja
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JP2019550651A 2017-03-20 2018-03-19 ブロモドメインを阻害する4−(1−(1,1−ジ(ピリジン−2−イル)エチル)−6−(3,5−ジメチルイソオキサゾール−4−イル)−1H−ピロロ[3,2−b]ピリジン−3−イル)安息香酸の結晶形 Pending JP2020511467A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762473903P 2017-03-20 2017-03-20
US62/473,903 2017-03-20
PCT/US2018/023127 WO2018175311A1 (en) 2017-03-20 2018-03-19 Crystalline forms of 4-(1-(1,1-di(pyridin-2-yl)ethyl)-6-(3,5-dimethylisoxazol-4-yl)-1h- pyrrolo[3,2-b]pyridin-3-yl)benzoic acid that inhibits bromodomain

Publications (2)

Publication Number Publication Date
JP2020511467A JP2020511467A (ja) 2020-04-16
JP2020511467A5 true JP2020511467A5 (US07585860-20090908-C00112.png) 2021-04-15

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JP2019550651A Pending JP2020511467A (ja) 2017-03-20 2018-03-19 ブロモドメインを阻害する4−(1−(1,1−ジ(ピリジン−2−イル)エチル)−6−(3,5−ジメチルイソオキサゾール−4−イル)−1H−ピロロ[3,2−b]ピリジン−3−イル)安息香酸の結晶形

Country Status (7)

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US (1) US10577366B2 (US07585860-20090908-C00112.png)
EP (1) EP3601281B1 (US07585860-20090908-C00112.png)
JP (1) JP2020511467A (US07585860-20090908-C00112.png)
AU (1) AU2018237047A1 (US07585860-20090908-C00112.png)
CA (1) CA3056777A1 (US07585860-20090908-C00112.png)
ES (1) ES2896502T3 (US07585860-20090908-C00112.png)
WO (1) WO2018175311A1 (US07585860-20090908-C00112.png)

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