JP2020506878A5 - - Google Patents

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Publication number
JP2020506878A5
JP2020506878A5 JP2019530506A JP2019530506A JP2020506878A5 JP 2020506878 A5 JP2020506878 A5 JP 2020506878A5 JP 2019530506 A JP2019530506 A JP 2019530506A JP 2019530506 A JP2019530506 A JP 2019530506A JP 2020506878 A5 JP2020506878 A5 JP 2020506878A5
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JP
Japan
Prior art keywords
alkyl
ring
trek
haloalkoxy
haloalkyl
Prior art date
Application number
JP2019530506A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2018110669A5 (https=
JP7120549B2 (ja
JP2020506878A (ja
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Priority claimed from PCT/JP2017/044975 external-priority patent/WO2018110669A1/en
Publication of JP2020506878A publication Critical patent/JP2020506878A/ja
Publication of JP2020506878A5 publication Critical patent/JP2020506878A5/ja
Publication of JPWO2018110669A5 publication Critical patent/JPWO2018110669A5/ja
Application granted granted Critical
Publication of JP7120549B2 publication Critical patent/JP7120549B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2019530506A 2016-12-15 2017-12-14 Trek(twik関連kチャネル)チャネルのアクチベータ Active JP7120549B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662434524P 2016-12-15 2016-12-15
US62/434,524 2016-12-15
PCT/JP2017/044975 WO2018110669A1 (en) 2016-12-15 2017-12-14 Activator of trek (twik related k+ channels) channels

Publications (4)

Publication Number Publication Date
JP2020506878A JP2020506878A (ja) 2020-03-05
JP2020506878A5 true JP2020506878A5 (https=) 2022-03-28
JPWO2018110669A5 JPWO2018110669A5 (https=) 2022-03-28
JP7120549B2 JP7120549B2 (ja) 2022-08-17

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019530506A Active JP7120549B2 (ja) 2016-12-15 2017-12-14 Trek(twik関連kチャネル)チャネルのアクチベータ

Country Status (4)

Country Link
US (2) US11046683B2 (https=)
EP (1) EP3558992A4 (https=)
JP (1) JP7120549B2 (https=)
WO (1) WO2018110669A1 (https=)

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CN111978319B (zh) 2014-06-27 2023-08-11 诺格拉制药有限公司 芳基受体调制剂及其制备和使用方法
WO2018232264A1 (en) * 2017-06-15 2018-12-20 The Board Of Regents Of The University Of Oklahoma Benzamide derivatives for inhibiting endoplasmic reticulum (er) stress
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CN114031601B (zh) * 2022-01-12 2022-03-18 南京桦冠生物技术有限公司 一种盐酸兰地洛尔的制备方法
CN118695860A (zh) * 2022-02-23 2024-09-24 拜奥海芬治疗学有限公司 作为kv7通道激活剂的吡唑基化合物
AU2023225967A1 (en) * 2022-02-23 2024-08-29 Biohaven Therapeutics Ltd. Pyrazolyl compounds as kv7 channel activators
WO2023164538A1 (en) * 2022-02-23 2023-08-31 Biohaven Therapeutics Ltd. Pyrazolyl compounds as kv7 channel activators
CN114805233A (zh) * 2022-03-30 2022-07-29 华南理工大学 苯基四氮唑类xor抑制剂及其制备方法与应用

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