JP2020504707A5 - - Google Patents

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Publication number
JP2020504707A5
JP2020504707A5 JP2019523587A JP2019523587A JP2020504707A5 JP 2020504707 A5 JP2020504707 A5 JP 2020504707A5 JP 2019523587 A JP2019523587 A JP 2019523587A JP 2019523587 A JP2019523587 A JP 2019523587A JP 2020504707 A5 JP2020504707 A5 JP 2020504707A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
solvate
acceptable salt
alkyl
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2019523587A
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English (en)
Japanese (ja)
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JP2020504707A (ja
JP7042547B2 (ja
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Publication date
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Priority claimed from PCT/US2017/061868 external-priority patent/WO2018093947A1/en
Publication of JP2020504707A publication Critical patent/JP2020504707A/ja
Publication of JP2020504707A5 publication Critical patent/JP2020504707A5/ja
Application granted granted Critical
Publication of JP7042547B2 publication Critical patent/JP7042547B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2019523587A 2016-11-16 2017-11-15 Magl阻害剤 Expired - Fee Related JP7042547B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662423099P 2016-11-16 2016-11-16
US62/423,099 2016-11-16
PCT/US2017/061868 WO2018093947A1 (en) 2016-11-16 2017-11-15 Magl inhibitors

Publications (3)

Publication Number Publication Date
JP2020504707A JP2020504707A (ja) 2020-02-13
JP2020504707A5 true JP2020504707A5 (enExample) 2021-02-04
JP7042547B2 JP7042547B2 (ja) 2022-03-28

Family

ID=62106678

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2019523587A Expired - Fee Related JP7042547B2 (ja) 2016-11-16 2017-11-15 Magl阻害剤

Country Status (29)

Country Link
US (1) US10093635B2 (enExample)
EP (1) EP3541821A4 (enExample)
JP (1) JP7042547B2 (enExample)
KR (1) KR20190077544A (enExample)
CN (1) CN110267963B (enExample)
AR (1) AR110089A1 (enExample)
AU (1) AU2017361251B2 (enExample)
BR (1) BR112019009994A2 (enExample)
CA (1) CA3043615A1 (enExample)
CL (1) CL2019001339A1 (enExample)
CO (1) CO2019005059A2 (enExample)
CR (1) CR20190241A (enExample)
DO (1) DOP2019000122A (enExample)
EA (1) EA038090B1 (enExample)
EC (1) ECSP19035077A (enExample)
GE (2) GEAP202215088A (enExample)
IL (1) IL266523B (enExample)
JO (1) JOP20190106A1 (enExample)
MA (1) MA46857A (enExample)
MX (1) MX391117B (enExample)
NI (1) NI201900051A (enExample)
PE (1) PE20191144A1 (enExample)
PH (1) PH12019501097A1 (enExample)
RU (1) RU2754536C1 (enExample)
TN (1) TN2019000153A1 (enExample)
TW (1) TWI756299B (enExample)
UA (1) UA124542C2 (enExample)
WO (1) WO2018093947A1 (enExample)
ZA (1) ZA201903100B (enExample)

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JOP20190107A1 (ar) 2016-11-16 2019-05-09 Lundbeck La Jolla Research Center Inc مثبطات أحادي أسيل جليسرول ليباز (magl)
KR20190085046A (ko) 2016-11-16 2019-07-17 어바이드 테라퓨틱스, 인크. 약학 제제
DK3541807T3 (da) 2016-11-16 2021-12-06 H Lundbeck As Krystallinsk form af en magl-inhibitor
EA201992409A1 (ru) 2017-05-23 2020-03-23 Лундбекк Ла-Хойя Рисерч Сентер, Инк. Ингибиторы magl на основе пиразола
JP7257387B2 (ja) 2017-08-29 2023-04-13 ハー・ルンドベック・アクチエゼルスカベット スピロ環化合物並びにその作製及び使用方法
KR20210010475A (ko) * 2018-05-15 2021-01-27 룬드벡 라 졸라 리서치 센터 인코포레이티드 Magl 저해제
MA54827A (fr) * 2019-01-25 2022-05-04 H Lundbeck As Méthodes de traitement d'une maladie à l'aide d'inhibiteurs de magl
KR20220101095A (ko) * 2019-11-15 2022-07-19 하. 룬드벡 아크티에셀스카브 Magl 억제제의 결정형
IT202000007150A1 (it) * 2020-04-03 2021-10-03 Univ Pisa Inibitori di monoacilglicerolo lipasi (magl)
IL297470A (en) 2020-04-21 2022-12-01 H Lundbeck As Synthesis of a monoacylglycerol lipase inhibitor
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KR20250005229A (ko) 2022-05-04 2025-01-09 하. 룬드벡 아크티에셀스카브 모노아실글리세롤 리파제 억제제로서 1,1,1,3,3,3-헥사플루오로프로판-2-일 (s)-1-(피리다진-3-일카르바모일)-6 아자스피로[2.5]옥탄-6-카르복실레이트의 결정질 형태

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