JP2020083892A5 - - Google Patents
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- Publication number
- JP2020083892A5 JP2020083892A5 JP2019212064A JP2019212064A JP2020083892A5 JP 2020083892 A5 JP2020083892 A5 JP 2020083892A5 JP 2019212064 A JP2019212064 A JP 2019212064A JP 2019212064 A JP2019212064 A JP 2019212064A JP 2020083892 A5 JP2020083892 A5 JP 2020083892A5
- Authority
- JP
- Japan
- Prior art keywords
- beraprost
- monohydrate
- solvent
- type
- following
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16/199,471 | 2018-11-26 | ||
| US16/199,471 US10577341B1 (en) | 2018-11-26 | 2018-11-26 | Beraprost-314d monohydrate crystals and methods for preparation thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020083892A JP2020083892A (ja) | 2020-06-04 |
| JP2020083892A5 true JP2020083892A5 (https=) | 2021-03-25 |
| JP6894489B2 JP6894489B2 (ja) | 2021-06-30 |
Family
ID=68655416
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2019212064A Active JP6894489B2 (ja) | 2018-11-26 | 2019-11-25 | ベラプロスト−314d・一水和物結晶及びその製造方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US10577341B1 (https=) |
| EP (1) | EP3656767A1 (https=) |
| JP (1) | JP6894489B2 (https=) |
| KR (1) | KR102317032B1 (https=) |
| CN (1) | CN111217782A (https=) |
| TW (1) | TWI724651B (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11447440B2 (en) * | 2020-10-29 | 2022-09-20 | Chirogate International Inc. | Treprostinil monohydrate crystals and methods for preparation thereof |
| CN115611838A (zh) * | 2021-07-15 | 2023-01-17 | 四川国为制药有限公司 | 一种前列环素衍生物的晶型 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS59134787A (ja) * | 1983-01-19 | 1984-08-02 | Toray Ind Inc | 5,6,7−トリノル−4,8−インタ−m−フエニレンPGI↓2誘導体の製造法 |
| JP4503942B2 (ja) * | 2003-06-11 | 2010-07-14 | 大正製薬株式会社 | 止痒剤 |
| CN103717585B (zh) * | 2011-06-16 | 2015-11-25 | 琅歌生物技术股份有限公司 | 贝前列素的生产方法 |
| JP2016512833A (ja) * | 2013-03-15 | 2016-05-09 | ゲームス・ファーマ・インコーポレイテッド | ウイルス感染症の治療薬としてのベラプロスト異性体 |
| CN103242274B (zh) * | 2013-05-22 | 2014-11-05 | 孙威 | 一种贝前列素钠化合物及其制备方法 |
| KR20170012314A (ko) * | 2014-05-20 | 2017-02-02 | 렁 바이오테크놀로지 인크. | 베라프로스트 및 그의 유도체의 제조 방법 |
| KR101986966B1 (ko) * | 2015-08-12 | 2019-06-07 | 유나이티드 쎄러퓨틱스 코포레이션 | 베라프로스트의 제조 방법 |
| HU231080B1 (hu) * | 2016-04-05 | 2020-07-28 | CHINOIN Gyógyszer és Vegyészeti Termékek Gyára Zrt. | Eljárás optikailag aktív Beraprost előállítására |
| KR101777632B1 (ko) * | 2016-04-11 | 2017-09-12 | 연성정밀화학(주) | 베라프로스트 나트륨 결정형 및 이의 제조방법 |
-
2018
- 2018-11-26 US US16/199,471 patent/US10577341B1/en active Active
-
2019
- 2019-11-25 EP EP19211276.1A patent/EP3656767A1/en active Pending
- 2019-11-25 KR KR1020190152168A patent/KR102317032B1/ko active Active
- 2019-11-25 JP JP2019212064A patent/JP6894489B2/ja active Active
- 2019-11-26 TW TW108143007A patent/TWI724651B/zh active
- 2019-11-26 CN CN201911176459.6A patent/CN111217782A/zh active Pending
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