JP2023554492A5 - - Google Patents

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Publication number
JP2023554492A5
JP2023554492A5 JP2023537470A JP2023537470A JP2023554492A5 JP 2023554492 A5 JP2023554492 A5 JP 2023554492A5 JP 2023537470 A JP2023537470 A JP 2023537470A JP 2023537470 A JP2023537470 A JP 2023537470A JP 2023554492 A5 JP2023554492 A5 JP 2023554492A5
Authority
JP
Japan
Prior art keywords
formula
compound
approximately
mixture
fumarate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023537470A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023554492A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/061895 external-priority patent/WO2022130304A1/en
Publication of JP2023554492A publication Critical patent/JP2023554492A/ja
Publication of JP2023554492A5 publication Critical patent/JP2023554492A5/ja
Pending legal-status Critical Current

Links

JP2023537470A 2020-12-18 2021-12-17 共結晶のcdk阻害剤 Pending JP2023554492A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN202041055174 2020-12-18
IN202041055174 2020-12-18
PCT/IB2021/061895 WO2022130304A1 (en) 2020-12-18 2021-12-17 Cocrystal of a cdk inhibitor

Publications (2)

Publication Number Publication Date
JP2023554492A JP2023554492A (ja) 2023-12-27
JP2023554492A5 true JP2023554492A5 (https=) 2024-12-25

Family

ID=80001496

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023537470A Pending JP2023554492A (ja) 2020-12-18 2021-12-17 共結晶のcdk阻害剤

Country Status (17)

Country Link
US (1) US20240059669A1 (https=)
EP (1) EP4263534A1 (https=)
JP (1) JP2023554492A (https=)
KR (1) KR20230159363A (https=)
CN (1) CN116685326A (https=)
AU (1) AU2021402415A1 (https=)
CA (1) CA3202198A1 (https=)
CL (1) CL2023001753A1 (https=)
CO (1) CO2023009368A2 (https=)
CR (1) CR20230261A (https=)
DO (1) DOP2023000126A (https=)
EC (1) ECSP23054131A (https=)
IL (1) IL303738A (https=)
MX (1) MX2023007218A (https=)
PE (1) PE20231441A1 (https=)
TW (1) TW202241881A (https=)
WO (1) WO2022130304A1 (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022084930A2 (en) * 2020-10-22 2022-04-28 Aurigene Discovery Technologies Limited Cancer therapy using a combination of cdk7 inhibitor with an anti-microtubule agent
US12084453B2 (en) 2021-12-10 2024-09-10 Incyte Corporation Bicyclic amines as CDK12 inhibitors
WO2023224961A1 (en) 2022-05-16 2023-11-23 Exelixis, Inc. Cancer therapy using a combination of a cdk7 inhibitor with an oral serd
TW202508595A (zh) 2023-05-04 2025-03-01 美商銳新醫藥公司 用於ras相關疾病或病症之組合療法
US20250049810A1 (en) 2023-08-07 2025-02-13 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder
AU2024360465A1 (en) 2023-10-12 2026-04-09 Revolution Medicines, Inc. Macrocyclic ras inhibitors
WO2025171296A1 (en) 2024-02-09 2025-08-14 Revolution Medicines, Inc. Ras inhibitors
WO2025217307A1 (en) 2024-04-09 2025-10-16 Revolution Medicines, Inc. Methods for predicting response to a ras(on) inhibitor and combination therapies
TW202547461A (zh) 2024-05-17 2025-12-16 美商銳新醫藥公司 Ras抑制劑
WO2025255438A1 (en) 2024-06-07 2025-12-11 Revolution Medicines, Inc. Methods of treating a ras protein-related disease or disorder
CN118772106A (zh) * 2024-06-07 2024-10-15 山东大学 伊马替尼-没食子酸共晶、其溶剂化物、制备方法和应用
WO2025265060A1 (en) 2024-06-21 2025-12-26 Revolution Medicines, Inc. Therapeutic compositions and methods for managing treatment-related effects
WO2026006747A1 (en) 2024-06-28 2026-01-02 Revolution Medicines, Inc. Ras inhibitors
WO2026015790A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015801A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015796A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2026015825A1 (en) 2024-07-12 2026-01-15 Revolution Medicines, Inc. Use of ras inhibitor for treating pancreatic cancer
WO2026050446A1 (en) 2024-08-29 2026-03-05 Revolution Medicines, Inc. Ras inhibitors
WO2026072904A2 (en) 2024-09-26 2026-04-02 Revolution Medicines, Inc. Compositions and methods for treating lung cancer

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI3302448T1 (sl) 2015-06-04 2024-03-29 Aurigene Oncology Limited Substituirani heterociklični derivati kot inhibitorji cdk

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