JP2022505670A5 - - Google Patents

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Publication number
JP2022505670A5
JP2022505670A5 JP2021522086A JP2021522086A JP2022505670A5 JP 2022505670 A5 JP2022505670 A5 JP 2022505670A5 JP 2021522086 A JP2021522086 A JP 2021522086A JP 2021522086 A JP2021522086 A JP 2021522086A JP 2022505670 A5 JP2022505670 A5 JP 2022505670A5
Authority
JP
Japan
Prior art keywords
crystalline salt
salt
xrpd
pattern
theta
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021522086A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022505670A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/059385 external-priority patent/WO2020092898A1/en
Publication of JP2022505670A publication Critical patent/JP2022505670A/ja
Publication of JP2022505670A5 publication Critical patent/JP2022505670A5/ja
Priority to JP2024085295A priority Critical patent/JP2024109860A/ja
Pending legal-status Critical Current

Links

JP2021522086A 2018-11-02 2019-11-01 血漿カリクレイン阻害剤の結晶塩 Pending JP2022505670A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2024085295A JP2024109860A (ja) 2018-11-02 2024-05-27 血漿カリクレイン阻害剤の結晶塩

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862754983P 2018-11-02 2018-11-02
US62/754,983 2018-11-02
PCT/US2019/059385 WO2020092898A1 (en) 2018-11-02 2019-11-01 Crystalline salts of a plasma kallikrein inhibitor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2024085295A Division JP2024109860A (ja) 2018-11-02 2024-05-27 血漿カリクレイン阻害剤の結晶塩

Publications (2)

Publication Number Publication Date
JP2022505670A JP2022505670A (ja) 2022-01-14
JP2022505670A5 true JP2022505670A5 (https=) 2022-10-17

Family

ID=70457981

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021522086A Pending JP2022505670A (ja) 2018-11-02 2019-11-01 血漿カリクレイン阻害剤の結晶塩
JP2024085295A Pending JP2024109860A (ja) 2018-11-02 2024-05-27 血漿カリクレイン阻害剤の結晶塩

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024085295A Pending JP2024109860A (ja) 2018-11-02 2024-05-27 血漿カリクレイン阻害剤の結晶塩

Country Status (22)

Country Link
US (11) US10662160B1 (https=)
EP (1) EP3873463A4 (https=)
JP (2) JP2022505670A (https=)
KR (1) KR102810837B1 (https=)
CN (1) CN112969458A (https=)
AR (1) AR116951A1 (https=)
AU (1) AU2019374115B8 (https=)
BR (1) BR112021008249A2 (https=)
CA (1) CA3117123A1 (https=)
CL (1) CL2021001094A1 (https=)
CO (1) CO2021007172A2 (https=)
EA (1) EA202191192A1 (https=)
IL (2) IL322896A (https=)
MA (1) MA54087A (https=)
MX (1) MX2021004917A (https=)
PE (1) PE20211280A1 (https=)
PH (1) PH12021550883A1 (https=)
PY (1) PY1991831A (https=)
SG (1) SG11202103804TA (https=)
TW (1) TW202031255A (https=)
UY (1) UY38438A (https=)
WO (1) WO2020092898A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102736869B1 (ko) 2014-03-07 2024-12-02 바이오크리스트파마슈티컬즈,인코포레이티드 인간 혈장 칼리크레인 저해제
UY38438A (es) 2018-11-02 2020-05-29 Biocryst Pharm Inc Sales cristalinas de un inhibidor de calicreína plasmática
WO2021025969A1 (en) * 2019-08-02 2021-02-11 Teva Pharmaceuticals International Gmbh Solid state forms of berotralstat
CN116375648A (zh) * 2023-03-22 2023-07-04 苏州农平科技发展有限公司 贝罗司他中间体的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4559157A (en) * 1983-04-21 1985-12-17 Creative Products Resource Associates, Ltd. Cosmetic applicator useful for skin moisturizing
BRPI0519331A2 (pt) 2004-12-15 2009-01-20 Bristol Myers Squibb Co formas cristalina de um inibidor de fator xa
CN101495468A (zh) * 2006-07-31 2009-07-29 艾克提弗赛特制药股份有限公司 血浆激肽释放酶抑制剂
WO2008016883A2 (en) 2006-07-31 2008-02-07 Activesite Pharmaceuticals, Inc. Inhibitors of plasma kallikrein
RU2585683C2 (ru) * 2010-05-19 2016-06-10 Сандоз Аг Очистка позаконазола и промежуточных продуктов для синтеза позаконазола
US9012464B2 (en) 2010-11-25 2015-04-21 Ratiopharm Gmbh Salts and polymorphic forms of Afatinib
GB201212081D0 (en) * 2012-07-06 2012-08-22 Kalvista Pharmaceuticals Ltd New polymorph
KR102736869B1 (ko) * 2014-03-07 2024-12-02 바이오크리스트파마슈티컬즈,인코포레이티드 인간 혈장 칼리크레인 저해제
DK4019022T3 (en) 2015-10-01 2024-02-19 Biocryst Pharm Inc Human plasma kallikrein inhibitors
UY38438A (es) 2018-11-02 2020-05-29 Biocryst Pharm Inc Sales cristalinas de un inhibidor de calicreína plasmática
CN114206839B (zh) 2019-08-06 2025-03-07 拜奥克里斯特制药公司 血浆激肽释放酶抑制剂的生产规模合成

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