JP2022524741A5 - - Google Patents
Info
- Publication number
- JP2022524741A5 JP2022524741A5 JP2021552142A JP2021552142A JP2022524741A5 JP 2022524741 A5 JP2022524741 A5 JP 2022524741A5 JP 2021552142 A JP2021552142 A JP 2021552142A JP 2021552142 A JP2021552142 A JP 2021552142A JP 2022524741 A5 JP2022524741 A5 JP 2022524741A5
- Authority
- JP
- Japan
- Prior art keywords
- selinexol
- succinic acid
- cocrystal
- mixed solution
- morphology
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025106508A JP2025134935A (ja) | 2019-03-20 | 2025-06-24 | セリネクソールの共結晶形態 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962821203P | 2019-03-20 | 2019-03-20 | |
| US62/821,203 | 2019-03-20 | ||
| PCT/US2020/023530 WO2020191140A1 (en) | 2019-03-20 | 2020-03-19 | Co-crystal forms of selinexor |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025106508A Division JP2025134935A (ja) | 2019-03-20 | 2025-06-24 | セリネクソールの共結晶形態 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022524741A JP2022524741A (ja) | 2022-05-10 |
| JP2022524741A5 true JP2022524741A5 (https=) | 2024-11-18 |
Family
ID=70293085
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021552142A Pending JP2022524741A (ja) | 2019-03-20 | 2020-03-19 | セリネクソールの共結晶形態 |
| JP2025106508A Pending JP2025134935A (ja) | 2019-03-20 | 2025-06-24 | セリネクソールの共結晶形態 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025106508A Pending JP2025134935A (ja) | 2019-03-20 | 2025-06-24 | セリネクソールの共結晶形態 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US12559478B2 (https=) |
| EP (1) | EP3941588A1 (https=) |
| JP (2) | JP2022524741A (https=) |
| KR (1) | KR20210141936A (https=) |
| CN (1) | CN113423468A (https=) |
| BR (1) | BR112021016762A2 (https=) |
| CA (1) | CA3130107A1 (https=) |
| WO (1) | WO2020191140A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112021016762A2 (pt) | 2019-03-20 | 2021-10-19 | Johnson Matthey Public Limited Company | Cocristal de selinexor, composição farmacêutica, método de tratamento de doenças, e, processo para a preparação de cocristal de selinexor |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN104230936A (zh) * | 2009-12-03 | 2014-12-24 | 阿斯利康(瑞典)有限公司 | 三唑并[4,5-d]嘧啶血小板聚集抑制剂的共晶体 |
| EP4234545A3 (en) | 2011-07-29 | 2023-09-06 | Karyopharm Therapeutics Inc. | Hydrazide containing nuclear transport modulators and uses thereof |
| US9808450B2 (en) * | 2013-03-26 | 2017-11-07 | Celgene Corporation | Solid forms comprising 3-(4-amino-1-OXO-1,3-dihydro-isoindol-2-yl)-piperidine-2,6-dione and a coformer, compositions and methods of use thereof |
| US20180230140A1 (en) * | 2014-06-30 | 2018-08-16 | Basf Se | Multicomponent crystals of dasatinib with menthol or vanillin |
| KR102608259B1 (ko) | 2014-08-15 | 2023-11-29 | 카리오팜 쎄라퓨틱스, 인코포레이티드 | 셀리넥소의 다형태 |
| WO2017118940A1 (en) * | 2016-01-08 | 2017-07-13 | Dr. Reddy's Laboratories Limited | Solid forms of selinexor and process for their preparation |
| EP3565813A1 (en) * | 2017-01-05 | 2019-11-13 | Watson Laboratories, Inc. | Novel crystalline forms of selinexor and process for their preparation |
| CN107089946B (zh) * | 2017-05-05 | 2020-04-03 | 浙江科技学院 | 一种诺氟沙星与香兰素共晶及其制备方法 |
| BR112021016762A2 (pt) | 2019-03-20 | 2021-10-19 | Johnson Matthey Public Limited Company | Cocristal de selinexor, composição farmacêutica, método de tratamento de doenças, e, processo para a preparação de cocristal de selinexor |
-
2020
- 2020-03-19 BR BR112021016762-5A patent/BR112021016762A2/pt not_active Application Discontinuation
- 2020-03-19 JP JP2021552142A patent/JP2022524741A/ja active Pending
- 2020-03-19 EP EP20719832.6A patent/EP3941588A1/en not_active Withdrawn
- 2020-03-19 CA CA3130107A patent/CA3130107A1/en active Pending
- 2020-03-19 KR KR1020217028384A patent/KR20210141936A/ko not_active Withdrawn
- 2020-03-19 WO PCT/US2020/023530 patent/WO2020191140A1/en not_active Ceased
- 2020-03-19 CN CN202080013966.2A patent/CN113423468A/zh active Pending
-
2021
- 2021-09-01 US US17/446,664 patent/US12559478B2/en active Active
-
2025
- 2025-06-24 JP JP2025106508A patent/JP2025134935A/ja active Pending
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