JP2019535754A5 - - Google Patents

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JP2019535754A5
JP2019535754A5 JP2019527426A JP2019527426A JP2019535754A5 JP 2019535754 A5 JP2019535754 A5 JP 2019535754A5 JP 2019527426 A JP2019527426 A JP 2019527426A JP 2019527426 A JP2019527426 A JP 2019527426A JP 2019535754 A5 JP2019535754 A5 JP 2019535754A5
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Japan
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formula
compound according
compound
pharmaceutically acceptable
equation
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JP2019527426A
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English (en)
Japanese (ja)
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JP2019535754A (ja
JP7167021B2 (ja
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Priority claimed from PCT/US2017/063182 external-priority patent/WO2018098390A1/en
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Publication of JP2019535754A5 publication Critical patent/JP2019535754A5/ja
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JP2019527426A 2016-11-23 2017-11-24 アルブミン結合psma阻害剤 Active JP7167021B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662425810P 2016-11-23 2016-11-23
US62/425,810 2016-11-23
PCT/US2017/063182 WO2018098390A1 (en) 2016-11-23 2017-11-24 Albumin-binding psma inhibitors

Publications (3)

Publication Number Publication Date
JP2019535754A JP2019535754A (ja) 2019-12-12
JP2019535754A5 true JP2019535754A5 (enExample) 2021-01-07
JP7167021B2 JP7167021B2 (ja) 2022-11-08

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ID=60812130

Family Applications (1)

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JP2019527426A Active JP7167021B2 (ja) 2016-11-23 2017-11-24 アルブミン結合psma阻害剤

Country Status (8)

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US (1) US11147889B2 (enExample)
EP (1) EP3544960A1 (enExample)
JP (1) JP7167021B2 (enExample)
CN (1) CN109982998A (enExample)
BR (1) BR112019010206A2 (enExample)
CA (1) CA3043619A1 (enExample)
MX (1) MX2019005742A (enExample)
WO (1) WO2018098390A1 (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3079906A1 (en) * 2017-10-22 2019-04-25 Provincial Health Services Authority Novel radiometal-binding compounds for diagnosis or treatment of prostate specific membrane antigen-expressing cancer
WO2019246445A1 (en) * 2018-06-20 2019-12-26 The Research Foundation For The State University Of New York Triazamacrocycle-derived chelator compositions for coordination of imaging and therapy metal ions and methods of using same
CA3118762A1 (en) 2018-11-14 2020-05-22 Noria Therapeutics, Inc. Thioamide-containing compositions and methods of use thereof
WO2020108753A1 (en) * 2018-11-28 2020-06-04 ITM Isotopen Technologien München AG Novel tumor antigen binding agents and uses thereof
CA3136979A1 (en) 2019-04-17 2020-10-22 Provincial Health Services Authority Radiolabelled compounds for diagnosis or treatment of prostate-spe cific membrane antigen-expressing cancer
CN114401947B (zh) 2019-06-21 2024-11-29 省卫生服务机构 靶向前列腺特异性膜抗原的放射性标记化合物
WO2021177390A1 (ja) 2020-03-04 2021-09-10 日本メジフィジックス株式会社 化合物及び放射性標識化合物
MX2022013783A (es) * 2020-05-06 2023-04-19 Univ Cornell Compuestos tratanosticos que contienen cobre y metodos de uso.
EP4255891A1 (en) * 2020-12-04 2023-10-11 The Regents of University of California Peptide receptor radionuclide therapy
US20240018110A1 (en) * 2020-12-16 2024-01-18 The University Of British Columbia Radiolabeled compounds targeting the prostate-specific membrane antigen
CN114685599A (zh) * 2020-12-30 2022-07-01 南京江原安迪科正电子研究发展有限公司 一种psma靶向抑制剂及放射性核素标记的psma靶向抑制剂、制备方法和用途
JPWO2022186311A1 (enExample) * 2021-03-04 2022-09-09
CA3244865A1 (en) * 2022-03-04 2023-09-07 Provincial Health Services Authority RADIOLABELLED COMPOUNDS TARGETING PROSTATE-SPECIFIC MEMBRANE ANTIGEN
WO2024126687A1 (en) * 2022-12-16 2024-06-20 Silence Therapeutics Gmbh Nucleic acids conjugated to an albumin binding moiety
CN118496305A (zh) * 2023-02-16 2024-08-16 无锡诺宇医药科技有限公司 Psma靶向放射性药物及其合成和应用
CN116217505B (zh) * 2023-03-17 2024-10-01 南京医科大学 用于诊断或治疗表达前列腺特异性膜抗原癌症的新型标记靶向剂

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0621973D0 (en) * 2006-11-03 2006-12-13 Philogen Spa Binding molecules and uses thereof
HRP20240952T1 (hr) * 2009-03-19 2024-10-11 The Johns Hopkins University Spojevi koji ciljaju psma i njihova uporaba
PL2739316T3 (pl) * 2011-08-05 2019-09-30 Molecular Insight Pharmaceuticals, Inc. Radioznakowane inhibitory antygenu błonowego specyficznego dla prostaty
US10011632B2 (en) * 2011-08-22 2018-07-03 Siemens Medical Solutions Usa, Inc. PSMA imaging agents
US20160257961A1 (en) * 2013-11-06 2016-09-08 Solstice Biologics, Ltd. Polynucleotide constructs having disulfide groups
BR112016010927A2 (pt) * 2013-11-14 2017-08-08 Endocyte Inc Conjugado de fórmula
ES2912753T3 (es) * 2014-08-24 2022-05-27 Max Planck Gesellschaft Zur Foerderung Der Wss Método para la producción de ésteres activos marcados con 18F y su aplicación ejemplificada por la preparación de un marcador de PET específico de PSMA
GEAP202014748A (en) * 2015-09-30 2020-01-27 Univ Heidelberg Ruprecht Karls 18f-tagged inhibitors of prostate specific membrane antigen (psma) and their use as imaging agents for prostate cancer
HUE065327T2 (hu) * 2016-03-22 2024-05-28 Univ Johns Hopkins Prosztata-fajlagos membrán antigénhez célzott nagy affinitású szerek prosztatarák endoradioterápiájához
CA3028978A1 (en) * 2016-06-23 2017-12-28 Cornell University Double targeted constructs to affect tumor kill
DE102016122273B4 (de) * 2016-11-18 2018-06-21 Abx Advanced Biochemical Compounds Gmbh Präkursoren für die Radiofluorierung

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