JP2018531957A5 - - Google Patents

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Publication number
JP2018531957A5
JP2018531957A5 JP2018521301A JP2018521301A JP2018531957A5 JP 2018531957 A5 JP2018531957 A5 JP 2018531957A5 JP 2018521301 A JP2018521301 A JP 2018521301A JP 2018521301 A JP2018521301 A JP 2018521301A JP 2018531957 A5 JP2018531957 A5 JP 2018531957A5
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Japan
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chloro
carboxylic acid
ene
alkyl
cyclohex
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Ceased
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JP2018521301A
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Japanese (ja)
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JP2018531957A (ja
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Priority claimed from PCT/US2016/059057 external-priority patent/WO2017075178A1/en
Publication of JP2018531957A publication Critical patent/JP2018531957A/ja
Publication of JP2018531957A5 publication Critical patent/JP2018531957A5/ja
Ceased legal-status Critical Current

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JP2018521301A 2015-10-27 2016-10-27 ＲＯＲγＴ阻害薬としての置換二環式ピラゾール化合物及びその使用 Ceased JP2018531957A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562246918P 2015-10-27 2015-10-27
US62/246,918 2015-10-27
PCT/US2016/059057 WO2017075178A1 (en) 2015-10-27 2016-10-27 SUBSTITUTED BICYCLIC PYRAZOLE COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF

Publications (2)

Publication Number Publication Date
JP2018531957A JP2018531957A (ja) 2018-11-01
JP2018531957A5 true JP2018531957A5 (https=) 2019-11-28

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ID=58630774

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JP2018521301A Ceased JP2018531957A (ja) 2015-10-27 2016-10-27 ＲＯＲγＴ阻害薬としての置換二環式ピラゾール化合物及びその使用

Country Status (6)

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US (1) US10344000B2 (https=)
EP (1) EP3368516B1 (https=)
JP (1) JP2018531957A (https=)
AU (1) AU2016344111A1 (https=)
CA (1) CA3002846A1 (https=)
WO (1) WO2017075178A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9809561B2 (en) 2013-12-20 2017-11-07 Merck Sharp & Dohme Corp. Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease
EP3368535B1 (en) 2015-10-27 2020-12-02 Merck Sharp & Dohme Corp. Heteroaryl substituted benzoic acids as rorgammat inhibitors and uses thereof
JP2018535958A (ja) 2015-10-27 2018-12-06 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． ＲＯＲγＴ阻害薬としての置換インダゾール化合物及びその使用
CN110945002B (zh) * 2017-08-01 2021-12-24 正大天晴药业集团股份有限公司 作为RORγ抑制剂的双环化合物

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